ChemicalBook > CAS DataBase List > GSK5959

GSK5959

Product Name
GSK5959
CAS No.
901245-65-6
Chemical Name
GSK5959
Synonyms
CS-1636;GSK5959;BRPF1-IN-3;GSK-5959;GSK5959;N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide;Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-;BRPF3,GSK5959,bromodomain,Inhibitor,inhibit,BRD1,BRPF1,Epigenetic Reader Domain,GSK-5959,GSK 5959,BRPF2,epigenetics
CBNumber
CB23040788
Molecular Formula
C22H26N4O3
Formula Weight
394.47
MOL File
901245-65-6.mol
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GSK5959 Property

Boiling point:
527.3±50.0 °C(Predicted)
Density 
1.263±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO : 13 mg/mL (32.96 mM; Need ultrasonic and warming)
form 
Powder
pka
13.06±0.20(Predicted)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Cayman Chemical
Product number
18123
Product name
GSK5959
Purity
≥98%
Packaging
1mg
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
18123
Product name
GSK5959
Purity
≥98%
Packaging
5mg
Price
$100
Updated
2024/03/01
Cayman Chemical
Product number
18123
Product name
GSK5959
Purity
≥98%
Packaging
10mg
Price
$184
Updated
2024/03/01
Cayman Chemical
Product number
18123
Product name
GSK5959
Purity
≥98%
Packaging
25mg
Price
$381
Updated
2024/03/01
Tocris
Product number
5385
Product name
GSK5959
Purity
≥99%(HPLC)
Packaging
10
Price
$159
Updated
2021/12/16
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GSK5959 Chemical Properties,Usage,Production

Description

GSK 5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.

Uses

GSK5959 is as elective BRPF1 bromodomain inhibitor.

storage

Store at +4°C

GSK5959 Preparation Products And Raw materials

Raw materials

Preparation Products

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GSK5959 Suppliers

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901245-65-6, GSK5959Related Search:

GSK8612 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S)-3-piperidinylmethoxy]-1H-imidazo[4,5-c]pyridin-4-yl]-2-methyl-3-butyn-2-ol 1-(1-(3-methoxyphenyl)-7-propoxyindolizin-3-yl)ethanone GSK8612 GSK6853 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoicacid GSK620 GSK591 ROR gamma-t-IN-1 GSK872

  • GSK5959
  • BRPF1-IN-3
  • N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
  • GSK-5959;GSK5959
  • CS-1636
  • Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-
  • BRPF3,GSK5959,bromodomain,Inhibitor,inhibit,BRD1,BRPF1,Epigenetic Reader Domain,GSK-5959,GSK 5959,BRPF2,epigenetics
  • 901245-65-6
  • Inhibitors