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5-ISOTHIAZOLECARBOXYLIC ACID

Product Name
5-ISOTHIAZOLECARBOXYLIC ACID
CAS No.
10271-85-9
Chemical Name
5-ISOTHIAZOLECARBOXYLIC ACID
Synonyms
5-ISOTHIAZOLECARBOXYLIC ACID;ISOTHIAZOLE-5-CARBOXYLIC ACID;1,2-thiazole-5-carboxylic acid;8-Isoquinoline-methaneaminedihydrochloride
CBNumber
CB2317896
Molecular Formula
C4H3NO2S
Formula Weight
129.14
MOL File
10271-85-9.mol
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5-ISOTHIAZOLECARBOXYLIC ACID Property

Melting point:
196-200℃ (decomposition)
Boiling point:
178.4±23.0℃ (760 Torr)
Density 
1.525±0.06 g/cm3 (20 ºC 760 Torr)
Flash point:
61.7±22.6℃
storage temp. 
2-8°C
form 
Solid
pka
1.23±0.10(Predicted)
color 
Off-white to light brown
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Safety

HS Code 
2934208090
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P321Specific treatment (see … on this label).

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

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N-Bromosuccinimide Price

TRC
Product number
I917608
Product name
Isothiazole-5-carboxylicacid
Packaging
50mg
Price
$55
Updated
2021/12/16
Usbiological
Product number
280318
Product name
Isothiazole-5-carboxylic acid
Packaging
100mg
Price
$460
Updated
2021/12/16
Apolloscientific
Product number
OR313078
Product name
Isothiazole-5-carboxylic acid
Packaging
250mg
Price
$210
Updated
2021/12/16
AK Scientific
Product number
0659AA
Product name
Isothiazole-5-carboxylicacid
Packaging
1g
Price
$266
Updated
2021/12/16
Apolloscientific
Product number
OR313078
Product name
Isothiazole-5-carboxylic acid
Packaging
1g
Price
$513
Updated
2021/12/16
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5-ISOTHIAZOLECARBOXYLIC ACID Chemical Properties,Usage,Production

Uses

Isothiazole-5-carboxylic acid (8-Isoquinoline-methaneaminedihydrochloride) is an organic compound with antibacterial, anticancer and anti-inflammatory properties. Isothiazole-5-carboxylic acid can be used to develop novel compounds to combat various diseases. Isothiazole-5-carboxylic acid exhibits a wide range of potential pharmacological activities and helps improve existing inhibitory schemes.

Synthesis

15901-66-3

10271-85-9

Methyl isothiazole-5-carboxylate (0.50 g, 3.49 mmol) was dissolved in a THF/MeOH solvent mixture (20 mL/5 mL) at room temperature, followed by slow addition of 1N NaOH solution (5.24 mL, 5.24 mmol). The reaction mixture was stirred continuously for 16 h at room temperature and the completion of the reaction was confirmed by thin layer chromatography (TLC) monitoring. Upon completion of the reaction, the reaction mixture was acidified to pH 2 with 1N HCl solution, at which point a precipitate was observed to be generated. The precipitate was separated by filtration and dried to afford the target product isothiazole-5-carboxylic acid (Compound 2) as a beige solid in a yield of 0.35 g (76% yield). The structure of the product was confirmed by 1H-NMR (400 MHz, DMSO-d6) with chemical shifts of δ 8.69 (d, 1H) and 7.85 (d, 1H), respectively.

References

[1] Patent: US2007/105864, 2007, A1. Location in patent: Page/Page column 151-152
[2] Patent: US2007/117804, 2007, A1. Location in patent: Page/Page column 78

5-ISOTHIAZOLECARBOXYLIC ACID Preparation Products And Raw materials

Raw materials

Preparation Products

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5-ISOTHIAZOLECARBOXYLIC ACID Suppliers

J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Fax
86-10-82849933
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jkinfo@jkchemical.com
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China
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96815
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76
Wuhan Chemwish Technology Co., Ltd
Tel
86-027-67849912
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86-027-87531808
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sales@chemwish.com
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China
ProdList
35896
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56
Shanghai Sinch Parmaceuticals Tech. Co. Ltd.
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sales@sinch.com.cn
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China
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11598
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Beijing Eternalchem Co,. Ltd.
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010-59484199 18611897322
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China
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Wuhan Haizheng Industry & Trade Development Co. Ltd
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027-8866 0053/88660577/88660578
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China
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55
Wuhan TCASChem Technology Co., Ltd.
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027-86697669 13986148687
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China
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3993
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21-33526724 18930996265
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Bide Pharmatech Ltd.
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400-164-7117 13681763483
Fax
+86-21-61629029
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China
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39966
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Modachem Shanghai Co., Ltd
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+86 (0)21 51320687 51371369 1744605818
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+86 (0)21 51371369
Country
China
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1578
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View Lastest Price from 5-ISOTHIAZOLECARBOXYLIC ACID manufacturers

Career Henan Chemical Co
Product
5-ISOTHIAZOLECARBOXYLIC ACID 10271-85-9
Price
US $1.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
Customized
Release date
2019-07-03