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ACETYL-PEPSTATIN

Product Name
ACETYL-PEPSTATIN
CAS No.
28575-34-0
Chemical Name
ACETYL-PEPSTATIN
Synonyms
Aids080613;Aids-080613;Ac-Pepstain;AC-PEPSTATIN;ACETYL-PEPSTATIN;N-Acetyl-Pepstatin;PEPSTATIN, ACETYL-;AC-VAL-VAL-STA-ALA-STA;AC-VAL-VAL-STA-ALA-STA-OH;ACETYL-PEPSTATIN USP/EP/BP
CBNumber
CB2390785
Molecular Formula
C31H57N5O9
Formula Weight
643.81
MOL File
28575-34-0.mol
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ACETYL-PEPSTATIN Property

storage temp. 
−20°C
solubility 
Soluble in DMSO
form 
Solid
color 
White to Off-white
InChIKey
WKYBEGDEGRCZNF-AHXZNPHMNA-N
SMILES
[C@H](CC(C)C)([C@@H](O)CC(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)[C@@H](O)CC(=O)O)NC(=O)[C@H](C(C)C)NC(=O)[C@H](C(C)C)NC(=O)C |&1:0,5,11,16,21,30,37,r|
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Safety

WGK Germany 
3
HS Code 
2924190090
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

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N-Bromosuccinimide Price

Biosynth Carbosynth
Product number
FA111026
Product name
Acetyl-Pepstatin Ac-Val-Val-Sta-Ala-Sta-OH
Packaging
500ug
Price
$90
Updated
2021/12/16
Biosynth Carbosynth
Product number
FA111026
Product name
Acetyl-Pepstatin Ac-Val-Val-Sta-Ala-Sta-OH
Packaging
1mg
Price
$157
Updated
2021/12/16
Biosynth Carbosynth
Product number
FA111026
Product name
Acetyl-Pepstatin Ac-Val-Val-Sta-Ala-Sta-OH
Packaging
2mg
Price
$273
Updated
2021/12/16
Chem-Impex
Product number
32941
Product name
Acetyl-Pepstatin
Packaging
5MG
Price
$384
Updated
2021/12/16
Biosynth Carbosynth
Product number
FA111026
Product name
Acetyl-Pepstatin Ac-Val-Val-Sta-Ala-Sta-OH
Packaging
5mg
Price
$546
Updated
2021/12/16
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ACETYL-PEPSTATIN Chemical Properties,Usage,Production

Uses

Acetyl Pepstatin is an HIV-1 protease inhibitor.

General Description

An aspartyl protease inhibitor that acts as an effective inhibitor of HIV-1 proteinase (Ki = 20 nM at pH 4.7) and HIV-2 proteinase (Ki = 5 nM at pH 4.7).

Biochem/physiol Actions

Target Ki: 20 nM at pH 4.7 against HIV-1 proteinase

in vivo

Pepstatin (Pepstatin A) has a very low toxicity, with LD50s of 1090 mg/kg, 875 mg/kg, 820 mg/kg and 450 mg/kg for mice, rats, rabbits, and dogs by i.p. route, and > 2000 mg/kg for all species by oral route[1].
Pepstatin (0.5-50 mg/kg, p.o.) suppresses stomach ulceration of the pylorus in ligated Shay rats[1].

Animal Model:Pylorus ligated male Wistar rats[1]
Dosage:0.5, 1, 10 and 50 mg/kg
Administration:Oral administration, 15 minutes after pyloric ligation
Result:Effectively prevented stomach ulceration.

ACETYL-PEPSTATIN Preparation Products And Raw materials

Raw materials

Preparation Products

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ACETYL-PEPSTATIN Suppliers

China 71 Europe 1 France 2 Germany 1 Japan 1 Switzerland 1 United Kingdom 3 United States 13 USA 1 Global 94
Hangzhou Peptidego Biotech Co.,Ltd.
Tel
0571-87213919
Email
Eric@peptidego.com
Country
China
ProdList
7408
Advantage
58
J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
Alabiochem Tech.Co., Ltd.
Tel
512-58900862 400-0707518
Fax
0086-512-56765862
Email
sales@alabiochem.com
Country
China
ProdList
970
Advantage
59
GL Biochem (Shanghai) Ltd
Tel
21-61263452 13641803416
Fax
86-21-61263399
Email
ymbetter@glbiochem.com
Country
China
ProdList
9981
Advantage
64
Shanghai Hanhong Scientific Co.,Ltd.
Tel
021-54306202 13764082696
Email
info@hanhongsci.com
Country
China
ProdList
42934
Advantage
64
Chemsky（shanghai）International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
Advantage
50
Nanjing Dulai Biotechnology Co., Ltd.
Tel
025-846993838003-8003 18013301590
Fax
025-84699383-8003
Email
njduly@126.com
Country
China
ProdList
3249
Advantage
55
Wuxi Zhongkun Biochemical Technology Co., Ltd.
Tel
0510-85629785 18013409632
Fax
051085625359
Email
sales@reading-chemicals.com
Country
China
ProdList
15178
Advantage
58
Sigma-Aldrich
Tel
021-61415566 800-8193336
Email
orderCN@merckgroup.com
Country
China
ProdList
51395
Advantage
80
Shanghai YuanYe Biotechnology Co., Ltd.
Tel
021-61312847; 18021002903
Fax
QQ:3008007432
Email
3008007409@qq.com
Country
China
ProdList
71826
Advantage
60
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View Lastest Price from ACETYL-PEPSTATIN manufacturers

WUHAN FORTUNA CHEMICAL CO., LTD
Product
Acetyl pepstatin 28575-34-0
Price
US $0.00/mg
Min. Order
1mg
Purity
≥95% or 98%
Supply Ability
1kg/month
Release date
2021-06-23
Career Henan Chemical Co
Product
ACETYL-PEPSTATIN 28575-34-0
Price
US $7.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
100KG
Release date
2020-02-16

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  • Cell Biology
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  • inhibitor