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a-Hydroxy Tamoxifen

Product Name
a-Hydroxy Tamoxifen
CAS No.
97151-02-5
Chemical Name
a-Hydroxy Tamoxifen
Synonyms
α-OHTAM;α-OHTAM;α-hydroxy Tamoxifen;(E)-α-Hydroxy tamoxifen;(E)-α-Hydroxy Tamoxifen;(E)-(+/-)-alpha-Hydroxytamoxifen;Benzeneethanol,b-[[4-[2-(dimethylamino)ethoxy]phenyl]phenylmethylene]-a-methyl-,(bE)-;Benzeneethanol, β-[[4-[2-(dimethylamino)ethoxy]phenyl]phenylmethylene]-α-methyl-, (βE)-
CBNumber
CB31176114
Molecular Formula
C26H29NO2
Formula Weight
387.52
MOL File
97151-02-5.mol
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a-Hydroxy Tamoxifen Property

Melting point:
115-119°C
Boiling point:
533.8±50.0 °C(Predicted)
Density 
1.094±0.06 g/cm3(Predicted)
storage temp. 
Amber Vial, -20°C Freezer
solubility 
Chloroform (Slightly), Methanol (Slightly)
pka
14.13±0.20(Predicted)
form 
Solid
color 
Pale Yellow to Pale Beige
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H361Suspected of damaging fertility or the unborn child

Precautionary statements

P201Obtain special instructions before use.

P202Do not handle until all safety precautions have been read and understood.

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P308+P313IF exposed or concerned: Get medical advice/attention.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Cayman Chemical
Product number
17204
Product name
α-hydroxy Tamoxifen
Purity
≥98%
Packaging
500μg
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
17204
Product name
α-hydroxy Tamoxifen
Purity
≥98%
Packaging
1mg
Price
$57
Updated
2024/03/01
Cayman Chemical
Product number
17204
Product name
α-hydroxy Tamoxifen
Purity
≥98%
Packaging
5mg
Price
$214
Updated
2024/03/01
Cayman Chemical
Product number
17204
Product name
α-hydroxy Tamoxifen
Purity
≥98%
Packaging
10mg
Price
$335
Updated
2024/03/01
TRC
Product number
H954700
Product name
(E)-α-HydroxyTamoxifen
Packaging
10mg
Price
$145
Updated
2021/12/16
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a-Hydroxy Tamoxifen Chemical Properties,Usage,Production

Description

Tamoxifen is a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer. Although it is an antagonist of ER action in breast tissue, it acts as an ER agonist in bone and blood vessels and a partial ER agonist in uterine tissues. α-hydroxy Tamoxifen is a reactive metabolite of tamoxifen that is formed by the action of cytochrome P450 3A4 in human liver. It can be further converted into genotoxic DNA adducts though a mechanism involving reversible O-sulfonation of the hydroxyl moiety, which in rats has been linked with hepatocarcinoma.

Chemical Properties

Pale Yellow Solid

Uses

A metabolite of the chemotherapeutic drug Tamoxifen (T006000). Exhibits a more potent estrogen agonist/antagonist activity than the parent drug. Also active as an intramembranous inhibitor of lipid peroxidation.

Uses

A metabolite of the chemotherapeutic drug tamoxifen. Exhibits a more potent estrogen agonist/antagonist activity than the parent drug. Also active as an intramembranous inhibitor of lipid peroxidation.

Definition

ChEBI: Alpha-Hydroxytamoxifen is a stilbenoid.

a-Hydroxy Tamoxifen Preparation Products And Raw materials

Raw materials

Preparation Products

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a-Hydroxy Tamoxifen Suppliers

BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
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United States
ProdList
14055
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65
BOC Sciences
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16314854226
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info@bocsci.com
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United States
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9923
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TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
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United States
ProdList
32165
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58
Aladdin Scientific
Tel
+1-+1(833)-552-7181
Email
sales@aladdinsci.com
Country
United States
ProdList
52925
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Cayman Chemical Company
Tel
--
Fax
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Email
cayman@caymanchem.com
Country
United States
ProdList
6213
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MedChemExpress
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Email
sales@medchemexpress.com
Country
United States
ProdList
6398
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Medical Isotopes
Tel
--
Fax
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Email
stohler@medicalisotopes.com
Country
United States
ProdList
6181
Advantage
68

97151-02-5, a-Hydroxy TamoxifenRelated Search:


  • (E)-α-Hydroxy Tamoxifen
  • (E)-(+/-)-alpha-Hydroxytamoxifen
  • α-OHTAM
  • Benzeneethanol, β-[[4-[2-(dimethylamino)ethoxy]phenyl]phenylmethylene]-α-methyl-, (βE)-
  • α-hydroxy Tamoxifen
  • (E)-α-Hydroxy tamoxifen
  • α-OHTAM
  • Benzeneethanol,b-[[4-[2-(dimethylamino)ethoxy]phenyl]phenylmethylene]-a-methyl-,(bE)-
  • 97151-02-5
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • Amines
  • Aromatics