CGS 15943
- Product Name
- CGS 15943
- CAS No.
- 104615-18-1
- Chemical Name
- CGS 15943
- Synonyms
- CGS 15943;CGS-15943A;CGS-15943 solid;CGS-15943 ADENOSINE A1 RECEPTOR;9-CHLORO-2-(2-FURYL)(1,2,4)TRIAZOLO(1,5-C)QUINAZOLIN-5-AMINE;9-chloro-2-(2-furyl)-(1,2,4)triazolo(1,5-c)quinazolin-5-imine;9-Chloro-2-(furan-2-yl)[1,2,4]triazolo[1,5-c]quinazolin-5-amine;9-CHLORO-2-(2-FURANYL)-[1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINE;[1,2,4]Triazolo[1,5-c]quinazolin-5-amine,9-chloro-2-(2-furanyl)-;9-Chloro-5,6-dihydro-2-(furan-2-yl)[1,2,4]triazolo[1,5-c]quinazolin-5-imine
- CBNumber
- CB3351424
- Molecular Formula
- C13H8ClN5O
- Formula Weight
- 285.69
- MOL File
- 104615-18-1.mol
CGS 15943 Property
- Melting point:
- 278-279 °C
- Density
- 1.72±0.1 g/cm3(Predicted)
- storage temp.
- room temp
- solubility
- DMSO: >16 mg/mL
- form
- solid
- pka
- 1.23±0.30(Predicted)
- color
- white
Safety
- WGK Germany
- 3
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
H315Causes skin irritation
H319Causes serious eye irritation
H335May cause respiratory irritation
- Precautionary statements
-
P261Avoid breathing dust/fume/gas/mist/vapours/spray.
P280Wear protective gloves/protective clothing/eye protection/face protection.
P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.
P302+P352IF ON SKIN: wash with plenty of soap and water.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
N-Bromosuccinimide Price
- Product number
- C199
- Product name
- CGS-15943
- Purity
- solid
- Packaging
- 25mg
- Price
- $160
- Updated
- 2024/03/01
- Product number
- J61313
- Product name
- CGS 15943, 99+%
- Packaging
- 10mg
- Price
- $94.8
- Updated
- 2021/12/16
- Product number
- J61313
- Product name
- CGS 15943, 99+%
- Packaging
- 50mg
- Price
- $327
- Updated
- 2021/12/16
- Product number
- 22073
- Product name
- CGS 15943
- Purity
- ≥95%
- Packaging
- 5mg
- Price
- $33
- Updated
- 2024/03/01
- Product number
- 22073
- Product name
- CGS 15943
- Purity
- ≥95%
- Packaging
- 10mg
- Price
- $62
- Updated
- 2024/03/01
CGS 15943 Chemical Properties,Usage,Production
Uses
Potent adenosine receptor antagonist
Definition
ChEBI: A member of the class of triazoloquinazolines that is [1,2,4]triazolo[1,5-c]quinazoline substited at positions 2, 5 and 9 by furan-2-yl, amino and chloro groups respectively. A potent antagonist at adenosine A1 and adenosi e A2A receptors.
Synthesis Reference(s)
Journal of Heterocyclic Chemistry, 27, p. 1549, 1990 DOI: 10.1002/jhet.5570270605
Biological Activity
Potent adenosine receptor antagonist (K i values are 3.5, 4.2, 16 and 51 nM for human A 1 , A 2A , A 2B and A 3 receptors respectively). Orally active in vivo .
Biochem/physiol Actions
CGS-15943 is a potent and non-selective adenosine receptor antagonist. It exhibits anti-carcinogenic and anti-apoptotic activity.
storage
Store at RT
CGS 15943 Preparation Products And Raw materials
Raw materials
Preparation Products
CGS 15943 Suppliers
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