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Diloxanide furoate

Product Name
Diloxanide furoate
CAS No.
3736-81-0
Chemical Name
Diloxanide furoate
Synonyms
8073cb;Furoate;furamide;amebiazol;furentomin;histomibal;diclofurazol;dichlofurazol;entamidefuroate;diloxanidfuroate
CBNumber
CB4723149
Molecular Formula
C14H11Cl2NO4
Formula Weight
328.15
MOL File
3736-81-0.mol
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Diloxanide furoate Property

Melting point:
111-114 °C
Boiling point:
438.4±45.0 °C(Predicted)
Density 
1.424±0.06 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
Chloroform (Slightly), Methanol (Slightly)
form 
Solid
pka
-0?+-.0.50(Predicted)
color 
Off-White to Light Beige
BCS Class
4
CAS DataBase Reference
3736-81-0(CAS DataBase Reference)
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Safety

Hazard Codes 
Xn
Risk Statements 
22
Safety Statements 
36
WGK Germany 
3
RTECS 
LV1821800
HS Code 
2924296000
Toxicity
mouse,LDLo,oral,710mg/kg (710mg/kg),Archives of Environmental Contamination and Toxicology. Vol. 14, Pg. 111, 1985.
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
1204805
Product name
Diloxanide furoate
Purity
United States Pharmacopeia (USP) Reference Standard
Packaging
200mg
Price
$381
Updated
2024/03/01
TRC
Product number
F861000
Product name
Furamide
Packaging
500mg
Price
$430
Updated
2021/12/16
Biosynth Carbosynth
Product number
FD63298
Product name
Diloxanide furoate
Packaging
250mg
Price
$450
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0002378
Product name
DILOXANIDE FUROATE
Purity
95.00%
Packaging
1G
Price
$1428
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0002378
Product name
DILOXANIDE FUROATE
Purity
95.00%
Packaging
1KG
Price
$6706.51
Updated
2021/12/16
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Diloxanide furoate Chemical Properties,Usage,Production

Uses

selective agonist for delta-opioid receptor

Uses

Antidiarrhoeals / Antiprotozoles

Uses

Furamide is an ambecide, an anti-protozoal drug used in the treatment of amoebozoa infections.

Definition

ChEBI: Diloxanide furoate is a carboxylic ester resulting from the formal condensation of the carboxy group of furan-2-carboxylic acid with the hydroxy group of 2,2-dichloro-N-(4-hydroxyphenyl)-N-methylacetamide. It is a drug used for the treatment of asymptomatic amebiasis. It has a role as an antiamoebic agent and a prodrug. It is a member of furans, a carboxylic ester, a tertiary carboxamide and an organochlorine compound.

Indications

Diloxanide furoate (Furamide) is an amebicide that is effective against trophozoites in the intestinal tract. In mild or asymptomatic infections, cures of 83 to 95% have been achieved; in patients with dysentery, cure rates may be less impressive. The drug is administered only orally and is rapidly absorbed from the gastrointestinal tract following hydrolysis of the ester group. It is remarkably free of side effects, but occasionally flatulence, abdominal distention, anorexia, nausea, vomiting, diarrhea, pruritus, and urticaria occur. Diloxanide is excreted in the urine, largely as the glucuronide. It is not available in the United States.

Clinical Use

Diloxanide furoate (available from the Centers for Disease Control and Prevention [CDC]) is prescribed for the treatment of asymptomatic amebiasis but is ineffective as a single agent for the extraintestinal form of the disease. The drug is administered orally and is hydrolyzed in the gut to give diloxanide, which is considered to be the active drug. Diloxanide is the only form identified in the bloodstream. The drug is found in the urine as the glucuronide.

Diloxanide furoate Preparation Products And Raw materials

Raw materials

Preparation Products

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Diloxanide furoate Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
Sinopharm Chemical Reagent Co,Ltd.
Tel
86-21-63210123
Fax
86-21-63290778 86-21-63218885
Email
sj_scrc@sinopharm.com
Country
China
ProdList
9815
Advantage
79
GIHI CHEMICALS CO.,LTD
Tel
0086-571-86217390
Fax
0086-571-86217391
Email
Sales@gihichem.com
Country
China
ProdList
860
Advantage
58
Jai Radhe Sales
Tel
+(91)-(79)-26431096/65255722
Fax
+(91)-(79)-26569884
Email
info@jairadhesales.com
Country
India
ProdList
397
Advantage
60
Zhengzhou Alfachem Co., Ltd.
Tel
0371-53765687 18937137882
Fax
QQ:2885373884
Email
2853979813@qq.com
Country
China
ProdList
7980
Advantage
55
Shanghai Qiao Chemical Science Co., Ltd
Tel
021-58892003
Email
info@qiaochem.com
Country
China
ProdList
5902
Advantage
65
Shanghai Chaolan Chemical Technology Center
Tel
QQ:65489617 15618227136
Fax
21-5161 9052
Email
Sales@ATKchemical.com
Country
China
ProdList
7266
Advantage
58
Beijing Solarbio Science & Tecnology Co., Ltd.
Tel
010-50973186 4009686088
Email
3193328036@qq.com
Country
China
ProdList
18338
Advantage
68
Beijing Jin Ming Biotechnology Co., Ltd.
Tel
010-60605840 18892239720
Fax
010-60605840
Email
psaitong@jm-bio.com
Country
China
ProdList
12306
Advantage
58
Musechem
Tel
+1-800-259-7612
Fax
+1-800-259-7612
Email
info@musechem.com
Country
United States
ProdList
4660
Advantage
60
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View Lastest Price from Diloxanide furoate manufacturers

Shaanxi Dideu Medichem Co. Ltd
Product
Diloxanide furoate 3736-81-0
Price
US $1.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
20t
Release date
2024-07-14
Shaanxi Dideu Medichem Co. Ltd
Product
Diloxanide furoate 3736-81-0
Price
US $0.00-0.00/Kg
Min. Order
1KG
Purity
99.0%
Supply Ability
500 tons
Release date
2020-04-27

3736-81-0, Diloxanide furoateRelated Search:


  • 2,2-DICHLORO-N-(4-HYDROXYPHENYL)-N-METHYLACETAMIDE 2-FUROIC ACID ESTER
  • DILOXANIDE FUROATE
  • 2-furancarboxylicacid,4-((dichloroacetyl)methylamino)phenylester
  • 2-furoicacid,esterwith2,2-dichloro-4’-hydroxy-n-methylacetanilide
  • 8073cb
  • amebiazol
  • dichlofurazol
  • diclofurazol
  • diloxanidfuroate
  • entamide2-furoate
  • entamidefuroate
  • furamide
  • furamide(amebicide)
  • furentomin
  • histomibal
  • 4-[(dichloroacetyl)methylamino]phenyl 2-furoate
  • Diloxanide 2-furoic acid ester
  • [4-[(2,2-dichloroacetyl)-methylamino]phenyl] furan-2-carboxylate
  • [4-[2,2-dichloroethanoyl(methyl)amino]phenyl] furan-2-carboxylate
  • furan-2-carboxylic acid [4-[(2,2-dichloroacetyl)-methyl-amino]phenyl] ester
  • Diloxanide Furoate (200 mg)
  • 4-(2,2-Dichloro-N-MethylacetaMido)phenyl furan-2-carboxylate
  • Furoate
  • 2-Furancarboxylic acid, 4-[(2,2-dichloroacetyl)methylamino]phenyl ester
  • Diloxanide Furoate (1204805)
  • 3736-81-0
  • 376-81-0
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