ChemicalBook > CAS DataBase List > sorivudine

sorivudine

Product Name
sorivudine
CAS No.
77181-69-2
Chemical Name
sorivudine
Synonyms
YN-72;BvAraU;D01734;BV-araU;Bravavir;Brovavir;Sorivudin;sorivudine;Bravavir (tn);Sorivudine (jan/usan/inn)
CBNumber
CB51074625
Molecular Formula
C11H13BrN2O6
Formula Weight
349.13
MOL File
77181-69-2.mol
More
Less

sorivudine Property

Melting point:
182° (Sakata, 1980); mp 195-200° (dec) (Machida, Sakata, 1983)
alpha 
D25 +0.5° (1N NaOH)
Density 
1.979±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: 250 mg/mL (716.07 mM)
form 
Solid
pka
8.37±0.10(Predicted)
color 
White to off-white
More
Less

Safety

Toxicity
LD50 in mice (mg/kg): ~3300 i.p.; >5000 s.c.; >10000 orally (Machida, Sakata, 1984)
More
Less

Hazard and Precautionary Statements (GHS)

More
Less

N-Bromosuccinimide Price

TRC
Product number
S677200
Product name
Sorivudine
Packaging
100mg
Price
$605
Updated
2021/12/16
ChemScene
Product number
CS-0080932
Product name
Sorivudine
Purity
95.03%
Packaging
50mg
Price
$700
Updated
2021/12/16
ChemScene
Product number
CS-0080932
Product name
Sorivudine
Purity
95.03%
Packaging
5mg
Price
$145
Updated
2021/12/16
ChemScene
Product number
CS-0080932
Product name
Sorivudine
Purity
95.03%
Packaging
10mg
Price
$230
Updated
2021/12/16
ChemScene
Product number
CS-0080932
Product name
Sorivudine
Purity
95.03%
Packaging
25mg
Price
$420
Updated
2021/12/16
More
Less

sorivudine Chemical Properties,Usage,Production

Description

Sorivudine is an orally-active antiviral nucleoside analog. It has potent and selective activity against herpes simplex virus type-1 (HSV-1) and varicella-zoster virus (VZV). In a cutaneous model infection of mice with HSV-1, oral administration of sorivudine at dose of 20 mg/kg resulted in a significant increase in the survival rate. Five percent sorivudine cream is also useful in the topical treatment of cutaneous HSV-1 infection, including immunocompromised patients. It has been suggested that its antiviral activity may be mediated by inhibition of DNA synthesis in virus infected cells.
Since the metabolite of sorivudine inhibits the enzyme for pyrimidine catabolism, caution should be taken not to use sorivudine in combination with fluorouracil drugs in order to avoid hematological disorders.

Originator

Yamasa Shoyu (Japan)

Uses

Sorivudine is an antimetabolite drug and can be used to synthesize antiviral compounds as well as compounds that can treat diseases of viral etiol.

Uses

Antiviral.

Definition

ChEBI: Sorivudine is an organic molecular entity.

brand name

Bravavir (Bristol-Myers Squibb);Usevir.

sorivudine Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

sorivudine Suppliers

LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9806
Advantage
58
Changzhou PBpharmaceutical R&D Co.,Ltd
Tel
0519-83990708
Fax
0519-83990708
Email
lxy2046@yeah.net
Country
China
ProdList
476
Advantage
55
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32165
Advantage
58
Changzhou PBpharmaceutical R&D Co.,Ltd
Tel
0519-83990708
Email
info@pbpharm.com
Country
CHINA
ProdList
498
Advantage
58
Shanghai Kaiwei Chemical Technology Co., Ltd.
Tel
021-58461859 15821823057
Email
service@aiviche.com
Country
China
ProdList
49312
Advantage
58
Hangzhou Jinghao Biotechnology Co., LTD
Tel
17513242016 17513242016
Fax
QQ:1576861551
Email
1576861551@qq.com
Country
China
ProdList
2800
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing@energy-chemical.com
Country
China
ProdList
44918
Advantage
58
Bide Pharmatech Ltd.
Tel
400-1647117 13681763483
Email
product02@bidepharm.com
Country
China
ProdList
62075
Advantage
58
InvivoChem
Tel
13549236410
Email
sales@invivochem.cn
Country
China
ProdList
6753
Advantage
58

77181-69-2, sorivudineRelated Search:


  • sorivudine
  • 1-(β-D-Arabinofuranosyl)-5-[(E)-2-bromoethenyl]uracil
  • 1-β-D-Arabinofuranosyl-5-[(E)-2-bromovinyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
  • Brovavir
  • BvAraU
  • BV-araU
  • YN-72
  • Bravavir
  • Bravavir (tn)
  • D01734
  • Sorivudine (jan/usan/inn)
  • 1-β-D-Arabinofuranosyl-5-[(1E)-2-bromoethenyl]-2,4(1H,3H)-pyrimidinedione
  • Sorivudin
  • 2,4(1H,3H)-Pyrimidinedione, 1-β-D-arabinofuranosyl-5-[(1E)-2-bromoethenyl]-
  • nucleoside,antiviral,inhibit,antimetabolite,Epstein-Barr,pyrimidine,virus,zoster,oral,varicella,Sorivudine,Inhibitor,herpes,DNA/RNA Synthesis,simplex,type
  • 1-β-D-Arabinofuranosyl-5-[(1E)-2-bromoethenyl]-2,4(1H,3H)-pyrimidinedione
  • 5-((E)-2-Bromovinyl)-1-((2R,3S,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione
  • 5-(E)-Bromovinyl-ara-uridine
  • 77181-69-2
  • C11H13BrN2O6