ChemicalBook > CAS DataBase List > (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Product Name
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
CAS No.
208706-12-1
Chemical Name
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Synonyms
264;3'R/1R;3'S)-L-054;S)-DuanPhos;(1R,1’S)-L-054,264;-iodo-1’(1R,1S,3R/1R,1R,3'S);S)-Octahydro-1-(2’-Hydroxy pravastatin sodium salt
CBNumber
CB52453421
Molecular Formula
C33H41N5O2
Formula Weight
539.71
MOL File
208706-12-1.mol
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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Property

Boiling point:
865.2±65.0 °C(Predicted)
Density 
1.25±0.1 g/cm3(Predicted)
storage temp. 
Store at +4°C
solubility 
Soluble to 50 mM in DMSO and to 100 mM in ethanol
form 
Powder
pka
12.79±0.20(Predicted)
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
2444
Product name
(1R,1S,3R/1R,1R,3'S)-L-054,264
Purity
≥96%(HPLC)
Packaging
10
Price
$289
Updated
2021/12/16
Tocris
Product number
2444
Product name
(1R,1S,3R/1R,1R,3'S)-L-054,264
Purity
≥96%(HPLC)
Packaging
1
Price
$134
Updated
2021/12/16
TRC
Product number
A633290
Product name
N-​[(1R)​-​2-​[[[3-​(Aminomethyl)​cyclohexyl]​methyl]​amino]​-​1-​(1H-​indol-​3-​ylmethyl)​-​2-​oxoethyl]​-spiro[1H-​indene-​1,​4''-​piperidine]​-​1''-​carboxamide
Packaging
2.5mg
Price
$315
Updated
2021/12/16
ApexBio Technology
Product number
B7057
Product name
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Packaging
10mg
Price
$423
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0009813
Product name
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Purity
95.00%
Packaging
5MG
Price
$504.41
Updated
2021/12/16
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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Chemical Properties,Usage,Production

Uses

Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor.N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4''-?piperidine]?-?1''-?carboxamide is a selective somatostatin sst2 receptor agonist.

Biological Activity

Potent and selective somatostatin sst 2 receptor agonist (K i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst 2 , sst 1 , sst 4 , sst 3 and sst 5 receptors respectively).

storage

Store at +4°C

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Preparation Products And Raw materials

Raw materials

Preparation Products

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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Suppliers

3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15839
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69
Shanghai T&W Pharmaceutical Co., Ltd.
Tel
+86 21 61551611
Fax
+86 21 50676805
Country
China
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9891
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58
EMMX Biotechnology LLC
Tel
888-539-0666
Fax
888-539-0666
Email
info@emmx.com
Country
United States
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8447
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TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32161
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Shanghai Universal Biotech Co.,Ltd
Tel
13774214275
Email
zhouzz@univ-bio.com
Country
China
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24994
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TargetMol Chemicals Inc.
Tel
4008200310
Email
marketing@tsbiochem.com
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China
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24644
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Henan Alpha Chemical Co., Ltd.
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0371-55013243 15324716602
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2853979810@qq.com
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China
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10034
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Nantong QuanYi Biotechnology Co., Ltd
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0513-66337626 18051384581
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sales@chemhifuture.com
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China
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TargetMol Chemicals Inc.
Tel
+8613564774135
Email
zijue.cai@tsbiochem.com
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United States
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19885
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Aladdin Scientific
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+1-+1(833)-552-7181
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sales@aladdinsci.com
Country
United States
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52924
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208706-12-1, (1R,1'S,3'R/1R,1'R,3'S)-L-054,264Related Search:


  • -methylethyl)-7a-methyl-inden-4-one
  • S)-DuanPhos
  • -Hydroxy pravastatin sodium salt
  • (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
  • N-[(1R)-2-[[[(1S*,3R*)-3-(AMINOMETHYL)CYCLOHEXYL]METHYL]AMINO]-1-(1H-INDOL-3-YLMETHYL)-2-OXOETHYL]SPIRO[1H-INDENE-1,4'-PIPERIDINE]-1'-CARBOXAMIDE
  • S)-L-054,264
  • (1R,1&rsquo
  • -iodo-1&rsquo
  • S)-Octahydro-1-(2&rsquo
  • -methylethyl)-7a-methyl-inden-4-ol
  • -(((2-Aminopropane-1,3-diyl)bis(oxy))bis(methylene))bis(phenylcyclopropanecarboxamide)
  • Spiro[1H-indene-1,4'-piperidine]-1'-carboxamide, N-[(1R)-2-[[[3-(aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]-
  • N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4'-?piperidine]?-?1'-?carboxamide
  • (1R,1S,3R/1R,1R,3'S)
  • 264
  • 3'R/1R
  • 3'S)-L-054
  • (1R,1'S,3'R/1R,1'R,3'S)L054,264,(1R,1'S,3'R/1R,1'R,3'S) L 054,264
  • N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide
  • (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
  • N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide
  • 208706-12-1
  • C33H41N5O2