(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Product Name: (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
CAS No.: 208706-12-1
Chemical Name: (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Synonyms: 264;3'R/1R;3'S)-L-054;S)-DuanPhos;(1R,1’S)-L-054,264;-iodo-1’(1R,1S,3R/1R,1R,3'S);S)-Octahydro-1-(2’-Hydroxy pravastatin sodium salt
CBNumber: CB52453421
Molecular Formula: C33H41N5O2
Formula Weight: 539.71
MOL File: 208706-12-1.mol

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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Property

Boiling point:: 865.2±65.0 °C(Predicted)
Density: 1.25±0.1 g/cm3(Predicted)
storage temp.: Store at +4°C
solubility: Soluble to 50 mM in DMSO and to 100 mM in ethanol
form: Powder
pka: 12.79±0.20(Predicted)

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris

Product number: 2444
Product name: (1R,1S,3R/1R,1R,3'S)-L-054,264
Purity: ≥96%(HPLC)
Packaging: 10
Price: $289
Updated: 2021/12/16

Tocris

Product number: 2444
Product name: (1R,1S,3R/1R,1R,3'S)-L-054,264
Purity: ≥96%(HPLC)
Packaging: 1
Price: $134
Updated: 2021/12/16

TRC

Product number: A633290
Product name: N-[(1R)-2-[[[3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]-spiro[1H-indene-1,4''-piperidine]-1''-carboxamide
Packaging: 2.5mg
Price: $315
Updated: 2021/12/16

ApexBio Technology

Product number: B7057
Product name: (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Packaging: 10mg
Price: $423
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: API0009813
Product name: (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Purity: 95.00%
Packaging: 5MG
Price: $504.41
Updated: 2021/12/16

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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Chemical Properties,Usage,Production

Uses

Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor.N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4''-?piperidine]?-?1''-?carboxamide is a selective somatostatin sst2 receptor agonist.

Biological Activity

Potent and selective somatostatin sst 2 receptor agonist (K i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst 2 , sst 1 , sst 4 , sst 3 and sst 5 receptors respectively).

storage

Store at +4°C

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Preparation Products And Raw materials

Raw materials

Preparation Products

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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Suppliers

China 7 United Kingdom 1 United States 7 USA 1 Global 16

3B Pharmachem (Wuhan) International Co.,Ltd.

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TargetMol Chemicals Inc.

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Henan Alpha Chemical Co., Ltd.

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Hangzhou MolCore BioPharmatech Co.,Ltd.

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208706-12-1, (1R,1'S,3'R/1R,1'R,3'S)-L-054,264Related Search:

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 SPIRO[INDENE-1,4'-PIPERIDINE] 1,3-Cyclohexanebis(methylamine)

-methylethyl)-7a-methyl-inden-4-one

S)-DuanPhos

-Hydroxy pravastatin sodium salt

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

N-[(1R)-2-[[[(1S*,3R*)-3-(AMINOMETHYL)CYCLOHEXYL]METHYL]AMINO]-1-(1H-INDOL-3-YLMETHYL)-2-OXOETHYL]SPIRO[1H-INDENE-1,4'-PIPERIDINE]-1'-CARBOXAMIDE

S)-L-054,264

(1R,1&rsquo

-iodo-1&rsquo

S)-Octahydro-1-(2&rsquo

-methylethyl)-7a-methyl-inden-4-ol

-(((2-Aminopropane-1,3-diyl)bis(oxy))bis(methylene))bis(phenylcyclopropanecarboxamide)

Spiro[1H-indene-1,4'-piperidine]-1'-carboxamide, N-[(1R)-2-[[[3-(aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]-

N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4'-?piperidine]?-?1'-?carboxamide

(1R,1S,3R/1R,1R,3'S)

264

3'R/1R

3'S)-L-054

(1R,1'S,3'R/1R,1'R,3'S)L054,264,(1R,1'S,3'R/1R,1'R,3'S) L 054,264

N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide

208706-12-1

C33H41N5O2