ChemicalBook > CAS DataBase List > (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
- Product Name
- (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
- CAS No.
- 208706-12-1
- Chemical Name
- (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
- Synonyms
- 264;3'R/1R;3'S)-L-054;S)-DuanPhos;(1R,1’S)-L-054,264;-iodo-1’(1R,1S,3R/1R,1R,3'S);S)-Octahydro-1-(2’-Hydroxy pravastatin sodium salt
- CBNumber
- CB52453421
- Molecular Formula
- C33H41N5O2
- Formula Weight
- 539.71
- MOL File
- 208706-12-1.mol
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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Property
- Boiling point:
- 865.2±65.0 °C(Predicted)
- Density
- 1.25±0.1 g/cm3(Predicted)
- storage temp.
- Store at +4°C
- solubility
- Soluble to 50 mM in DMSO and to 100 mM in ethanol
- form
- Powder
- pka
- 12.79±0.20(Predicted)
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N-Bromosuccinimide Price
Tocris
- Product number
- 2444
- Product name
- (1R,1S,3R/1R,1R,3'S)-L-054,264
- Purity
- ≥96%(HPLC)
- Packaging
- 10
- Price
- $289
- Updated
- 2021/12/16
Tocris
- Product number
- 2444
- Product name
- (1R,1S,3R/1R,1R,3'S)-L-054,264
- Purity
- ≥96%(HPLC)
- Packaging
- 1
- Price
- $134
- Updated
- 2021/12/16
TRC
- Product number
- A633290
- Product name
- N-[(1R)-2-[[[3-(Aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]-spiro[1H-indene-1,4''-piperidine]-1''-carboxamide
- Packaging
- 2.5mg
- Price
- $315
- Updated
- 2021/12/16
ApexBio Technology
- Product number
- B7057
- Product name
- (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
- Packaging
- 10mg
- Price
- $423
- Updated
- 2021/12/16
American Custom Chemicals Corporation
- Product number
- API0009813
- Product name
- (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
- Purity
- 95.00%
- Packaging
- 5MG
- Price
- $504.41
- Updated
- 2021/12/16
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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Chemical Properties,Usage,Production
Uses
Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor.N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4''-?piperidine]?-?1''-?carboxamide is a selective somatostatin sst2 receptor agonist.
Biological Activity
Potent and selective somatostatin sst 2 receptor agonist (K i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst 2 , sst 1 , sst 4 , sst 3 and sst 5 receptors respectively).
storage
Store at +4°C
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Preparation Products And Raw materials
Raw materials
Preparation Products
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