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THIOPERAMIDE MALEATE

Product Name
THIOPERAMIDE MALEATE
CAS No.
106243-16-7
Chemical Name
THIOPERAMIDE MALEATE
Synonyms
Thiop;MR 12842;thioperamide;THIOPERAMIDE MALEATE;THIOPERAMIDE MALEATE SALT;THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE;N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide;N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide;N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE;N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
CBNumber
CB5245732
Molecular Formula
C15H24N4S
Formula Weight
292.44
MOL File
106243-16-7.mol
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THIOPERAMIDE MALEATE Property

storage temp. 
Store at -20°C
solubility 
H2O: 10 mg/mL
form 
solid
color 
white
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Safety

Hazard Codes 
Xi
Risk Statements 
36/37/38
Safety Statements 
26-36
WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
0644
Product name
Thioperamide
Purity
≥99%(HPLC)
Packaging
10
Price
$123
Updated
2021/12/16
Tocris
Product number
0644
Product name
Thioperamide
Purity
≥99%(HPLC)
Packaging
50
Price
$515
Updated
2021/12/16
TRC
Product number
T344808
Product name
Thioperamide
Packaging
10mg
Price
$110
Updated
2021/12/16
Usbiological
Product number
256923
Product name
Thioperamide
Packaging
10mg
Price
$389
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0007635
Product name
THIOPERAMIDE
Purity
95.00%
Packaging
100MG
Price
$2116.25
Updated
2021/12/16
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THIOPERAMIDE MALEATE Chemical Properties,Usage,Production

Uses

Thioperamide is a highly potent and selective ligand for histamine H3-receptors.

Definition

ChEBI: Thioperamide is a primary aliphatic amine.

Biological Activity

Potent histamine H 3 and H 4 antagonist/inverse agonist. K i values are 25 and 27 nM for human recombinant H 3 and H 4 receptors respectively. Blocks eosinophil shape change (IC 50 = 1.4 μ M) and chemotaxis (IC 50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H 3 Receptor Tocriset™ .

storage

Store at -20°C

THIOPERAMIDE MALEATE Preparation Products And Raw materials

Raw materials

Preparation Products

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THIOPERAMIDE MALEATE Suppliers

3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15839
Advantage
69
Ascent Scientific
Tel
4401179829988
Fax
4402030 700 369
Email
customerservice@ascentscientific.co.uk
Country
United Kingdom
ProdList
279
Advantage
60
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd.
Tel
025-66099280 17798518460
Fax
(1)02557626880
Email
cfzhang@aikonchem.com
Country
China
ProdList
19915
Advantage
55
Beijin Yangguang Furui Chemical co.,Ltd.
Tel
010-57495520 13521095525
Email
zhw512@foxmail.com
Country
China
ProdList
488
Advantage
55
EMMX Biotechnology LLC
Tel
888-539-0666
Fax
888-539-0666
Email
info@emmx.com
Country
United States
ProdList
8447
Advantage
60
Amadis Chemical Company Limited
Tel
571-89925085
Fax
0086-571-89925065
Email
sales@amadischem.com
Country
China
ProdList
131957
Advantage
58
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32161
Advantage
58
MedBioPharmaceutical Technology Inc
Tel
021-69568360 18916172912
Email
order@med-bio.cn
Country
China
ProdList
8140
Advantage
58
Beijing Jin Ming Biotechnology Co., Ltd.
Tel
010-60605840 15801484223;
Email
psaitong@jm-bio.com
Country
China
ProdList
29774
Advantage
58
Shanghai Universal Biotech Co.,Ltd
Tel
13774214275
Email
zhouzz@univ-bio.com
Country
China
ProdList
24994
Advantage
58

106243-16-7, THIOPERAMIDE MALEATERelated Search:


  • N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
  • MR 12842
  • THIOPERAMIDE MALEATE
  • THIOPERAMIDE MALEATE SALT
  • THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE
  • N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide
  • Thiop
  • N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide
  • thioperamide
  • N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
  • N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE
  • N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
  • 1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-5-yl)-
  • 106243-16-7
  • C15H24N4SC4H4O4
  • Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier.
  • Histamine receptor
  • Histamine