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THIOPERAMIDE MALEATE

Product Name
THIOPERAMIDE MALEATE
CAS No.
106243-16-7
Chemical Name
THIOPERAMIDE MALEATE
Synonyms
Thiop;MR 12842;thioperamide;THIOPERAMIDE MALEATE;THIOPERAMIDE MALEATE SALT;THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE;N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide;N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide;N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE;N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
CBNumber
CB5245732
Molecular Formula
C15H24N4S
Formula Weight
292.44
MOL File
106243-16-7.mol
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THIOPERAMIDE MALEATE Property

storage temp. 
Store at -20°C
solubility 
H2O: 10 mg/mL
form 
solid
color 
white
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Safety

Hazard Codes 
Xi
Risk Statements 
36/37/38
Safety Statements 
26-36
WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
0644
Product name
Thioperamide
Purity
≥99%(HPLC)
Packaging
10
Price
$123
Updated
2021/12/16
Tocris
Product number
0644
Product name
Thioperamide
Purity
≥99%(HPLC)
Packaging
50
Price
$515
Updated
2021/12/16
TRC
Product number
T344808
Product name
Thioperamide
Packaging
10mg
Price
$110
Updated
2021/12/16
Usbiological
Product number
256923
Product name
Thioperamide
Packaging
10mg
Price
$389
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0007635
Product name
THIOPERAMIDE
Purity
95.00%
Packaging
100MG
Price
$2116.25
Updated
2021/12/16
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THIOPERAMIDE MALEATE Chemical Properties,Usage,Production

Uses

Thioperamide is a highly potent and selective ligand for histamine H3-receptors.

Definition

ChEBI: Thioperamide is a primary aliphatic amine.

Biological Activity

Potent histamine H 3 and H 4 antagonist/inverse agonist. K i values are 25 and 27 nM for human recombinant H 3 and H 4 receptors respectively. Blocks eosinophil shape change (IC 50 = 1.4 μ M) and chemotaxis (IC 50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H 3 Receptor Tocriset™ .

storage

Store at -20°C

THIOPERAMIDE MALEATE Preparation Products And Raw materials

Raw materials

Preparation Products

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THIOPERAMIDE MALEATE Suppliers

China 12 Europe 1 Germany 2 Japan 1 Switzerland 1 United Kingdom 6 United States 9 USA 1 Global 33
BIOTREND Chemicals AG
Tel
--
Fax
--
Email
info@biotrend.ch
Country
Germany
ProdList
1250
Advantage
62
Service Chemical Inc.
Tel
--
Fax
--
Email
sales@chemos-group.com
Country
Germany
ProdList
6350
Advantage
71

106243-16-7, THIOPERAMIDE MALEATERelated Search:

1,3-Dibutyl-2-thiourea 1-CYCLOHEXYL-2-THIOUREA 4-(1H-IMIDAZOL-4-YL)-1-METHYL-PIPERIDINE 4-(1H-IMIDAZOLE-4(5)-YL) PIPERIDINE N,N-DIETHYLTHIOUREA 1-PIPERIDINETHIOCARBOXAMIDE THIOPERAMIDE MALEATE N,N'-DI-N-PROPYLTHIOUREA

  • N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
  • MR 12842
  • THIOPERAMIDE MALEATE
  • THIOPERAMIDE MALEATE SALT
  • THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE
  • N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide
  • Thiop
  • N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide
  • thioperamide
  • N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
  • N-CYCLOHEXYL-4-(1H-IMIDAZOL-5-YL)-1-PIPERIDINECARBOTHIOAMIDE
  • N-Cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
  • 1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-5-yl)-
  • 106243-16-7
  • C15H24N4SC4H4O4
  • Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier.
  • Histamine receptor
  • Histamine