ChemicalBook > CAS DataBase List > carbutamide

carbutamide

Product Name
carbutamide
CAS No.
339-43-5
Chemical Name
carbutamide
Synonyms
Emedan;U-6987;Oranil;Bucrol;Burcol;Nadisan;Invenol;Alentin;Bucarban;Bukarban
CBNumber
CB5883608
Molecular Formula
C11H17N3O3S
Formula Weight
271.34
MOL File
339-43-5.mol
More
Less

carbutamide Property

Melting point:
144-145°
Density 
1.2840 (rough estimate)
refractive index 
1.6630 (estimate)
storage temp. 
Refrigerator
solubility 
DMSO (Slightly), Methanol (Slightly)
form 
Solid
pka
pKa 5.75(H2O t=25±0.02 I=0.2) (Uncertain)
color 
Off-White to Pale Beige
Water Solubility 
535.2mg/L(37 ºC)
EPA Substance Registry System
Benzenesulfonamide, 4-amino-N-[(butylamino)carbonyl]- (339-43-5)
More
Less

Safety

Hazardous Substances Data
339-43-5(Hazardous Substances Data)
Toxicity
LD50 s.c. in mice: 3 g/kg (Haack, Hagedorn)
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P362Take off contaminated clothing and wash before reuse.

P403+P233Store in a well-ventilated place. Keep container tightly closed.

P501Dispose of contents/container to..…

More
Less

N-Bromosuccinimide Price

Sigma-Aldrich
Product number
S385433
Product name
N1-(BUTYLCARBAMOYL)-SULFANILAMIDE
Purity
Aldrich
Packaging
50mg
Price
$209
Updated
2024/03/01
TRC
Product number
C183300
Product name
Carbutamide
Packaging
5mg
Price
$80
Updated
2021/12/16
TRC
Product number
C183300
Product name
Carbutamide
Packaging
25mg
Price
$120
Updated
2021/12/16
Biosynth Carbosynth
Product number
FC19809
Product name
Carbutamide
Packaging
25mg
Price
$160
Updated
2021/12/16
Biosynth Carbosynth
Product number
FC19809
Product name
Carbutamide
Packaging
10mg
Price
$86
Updated
2021/12/16
More
Less

carbutamide Chemical Properties,Usage,Production

Chemical Properties

Off-White to Pale Peach Solid

Originator

Carbutamide,Servier

Uses

Antidiabetic.

Definition

ChEBI: Carbutamide is a sulfonamide and a member of benzenes.

Manufacturing Process

223 g of the sodium salt of acetylsulfaniamide are stirred with 223 ml of triethylene glycol. 118 g of n-butyl isothiocyanate are added to the resulting homogeneous mixture. The resulting syrup is heated to 85°C for 4 hours. The mixture is then stirred with 1000 ml of chloroform and 1000 ml of water. The chloroform layer is twice shaken with water, each time with 250 ml. The aqueous extracts are combined and rendered weakly alkaline to phenolphthalein by addition of hydrochloric acid. Unreacted acetyl sulfanilamide precipitates and filtered off. The filtrate is acidified to a pH of 6.5 by the addition of HCl. An oily precipitate settles from the reaction solution and is separated therefrom. N-Butyl acetyl sulfanilylthiourea is precipitated from mother liquors obtained thereby by addition of HCl until Congo paper changes its color to blue. 210 g N-butyl acetyl sulfanilylthiourea are dissolved in 1400 ml of acetone while heating. The solution is mixed with 500 ml of water. A solution of 63 g of sodium nitrite in 120 ml of water is added thereto within about 45 minutes while stirring and cooling to 15°-20°C.
A suspension of crystals is obtained. 240 ml of 25% glacial acid are added thereto within 30 minutes. Stirring of the mixture is continued for 6 hours. N-Butyl acetyl sulfanilylurea mixed with sulfur is precipitated and filtered off. The crude reaction product is suspended in 1000 ml of water and is rendered weakly alkaline to phenolphthalein. Undissolved sulfur is filtered off. The filtrate is acidified by the addition of HCl. 250 g of N-butyl acetyl sulfanilylthiourea having a melting point of 186°-189°C are obtained. It is heated with 500 ml of 5 N potassium hydroxide solution to a temperature of 92°C for 2 hours while stirring. The solid reaction product is dissolved by heating with 750 ml of water and is purified by means of activated charcoal. The resulting solution is heated to 60°C and acidified by addition of HCl. 187 g of N-butyl acetyl sulfanilylthiourea melting at 139°-141°C obtained thereby.

Therapeutic Function

Oral hypoglycemic

Safety Profile

A poison by intraperitoneal route. Moderately toxic by ingestion and subcutaneous routes. An experimental teratogen. Other experimental reproductive effects. When heated to decomposition it emits very toxic fumes of NO, and SOx.

carbutamide Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

carbutamide Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
94657
Advantage
76
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky(shanghai)International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
Advantage
50
Shanghai Aladdin Bio-Chem Technology Co.,LTD
Tel
400-400-6206333 18521732826
Fax
021-50323701
Email
market@aladdin-e.com
Country
China
ProdList
25003
Advantage
65
ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Fax
0755-28363542
Email
sales@chem-strong.com
Country
China
ProdList
18070
Advantage
56
Shanghai CanSpecsci Instrument Co., Ltd.
Tel
400-6087598 15021221957
Fax
4006087598-8012
Email
order@canspecsci.com
Country
China
ProdList
2045
Advantage
56
ShangHai KenEn Chemical Technology Co., Ltd.
Tel
13120367189
Fax
021-50315529
Email
mychess007@163.com
Country
China
ProdList
1994
Advantage
55
Shanghai Xingui Biotechnology Co., Ltd.
Tel
17501653715
Email
xingui2022@126.com
Country
China
ProdList
10015
Advantage
58
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9806
Advantage
58
Shandong Xiya Chemical Co., Ltd.
Tel
4009903999 13395398332
Fax
0539-6365991
Email
sales@xiyashiji.com
Country
China
ProdList
20806
Advantage
60
More
Less

View Lastest Price from carbutamide manufacturers

Career Henan Chemical Co
Product
carbutamide 339-43-5
Price
US $1.00/KG
Min. Order
1KG
Purity
98%
Supply Ability
1lg; 2kg; 5kg; 10kg; 100kg
Release date
2019-08-31

339-43-5, carbutamideRelated Search:


  • carbutamide
  • UREA,1-BUTYL-3-SULFANILYL-
  • UREA,1-BUTYL-3-SULPHANILYL
  • 1-(4-aminophenyl)sulfonyl-3-butyl-urea
  • Emedan
  • Invenol
  • Nadisan
  • Oranil
  • U-6987
  • 1-(4-azanylphenyl)sulfonyl-3-butyl-urea
  • 1-Butyl-3-sulfanilylurea
  • Alentin
  • AMinophenurobutane
  • Bucarban
  • Bucrol
  • Bukarban
  • Burcol
  • Butisulfina
  • CarbutaMid
  • Diaboral
  • Glucidoral
  • N1-(ButylcarbaMoyl) sulfanilaMide
  • 4-Amino-N-(butylcarbamoyl)benzenesulfonamide
  • Benzenesulfonamide, 4-amino-N-[(butylamino)carbonyl]-
  • carbutamide USP/EP/BP
  • Benzenesulfonamide,4-amino-N-[(butylamino)carbony
  • Inhibitor,BZ-55,first-generation,orally,Anti-diabetic,inhibit,Carbutamide,BZ 55,hypoglycemic,BZ55,sulfonylurea
  • 339-43-5
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • Sulfur & Selenium Compounds
  • Amines
  • Aromatics