AZD2461

Product Name: AZD2461
CAS No.: 1174043-16-3
Chemical Name: AZD2461
Synonyms: CS-739;AZD2461;AZD 2461, >=98%;AZD2461 AZD-2461;AZD2461 USP/EP/BP;4-(4-Fluoro-3-(4-methoxypiperidine-1-carbonyl)benzyl)phthalazin-1(2H)-one;4-[4-Fluoro-3-[(4-methoxypiperidin-1-yl)carbonyl]benzyl]phthalazin-1(2H)-one;4-[[4-fluoro-3-(4-methoxypiperidine-1-carbonyl)phenyl]methyl]-2H-phthalazin-1-one;4-[[4-Fluoro-3-[(4-methoxy-1-piperidinyl)carbonyl]phenyl]methyl]-1(2H)-phthalazinone;1(2H)-Phthalazinone, 4-[[4-fluoro-3-[(4-methoxy-1-piperidinyl)carbonyl]phenyl]methyl]-
CBNumber: CB62655394
Molecular Formula: C22H22FN3O3
Formula Weight: 395.43
MOL File: 1174043-16-3.mol

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AZD2461 Property

Density: 1.33±0.1 g/cm3(Predicted)
storage temp.: 2-8°C
solubility: insoluble in H2O; ≥16.35 mg/mL in DMSO; ≥45.2 mg/mL in EtOH with ultrasonic
form: powder
pka: 12.07±0.40(Predicted)
color: white to beige

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

H373May cause damage to organs through prolonged or repeated exposure

Precautionary statements

P260Do not breathe dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P314Get medical advice/attention if you feel unwell.

P330Rinse mouth.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Sigma-Aldrich

Product number: SML1858
Product name: AZD2461
Purity: ≥98% (HPLC)
Packaging: 5MG
Price: $102
Updated: 2023/06/20

Sigma-Aldrich

Product number: SML1858
Product name: AZD2461
Purity: ≥98% (HPLC)
Packaging: 25MG
Price: $413
Updated: 2023/06/20

Cayman Chemical

Product number: 16876
Product name: AZD 2461
Purity: ≥95%
Packaging: 1mg
Price: $44
Updated: 2024/03/01

Cayman Chemical

Product number: 16876
Product name: AZD 2461
Purity: ≥95%
Packaging: 5mg
Price: $183
Updated: 2024/03/01

Cayman Chemical

Product number: 16876
Product name: AZD 2461
Purity: ≥95%
Packaging: 10mg
Price: $341
Updated: 2024/03/01

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AZD2461 Chemical Properties,Usage,Production

Uses

4-[4-Fluoro-3-[(4-methoxypiperidin-1-yl)carbonyl]benzyl]phthalazin-1(2H)-one is a phthalazinone derivative and potential PARP inhibitor.

Biochem/physiol Actions

AZD2461, an olaparib analog, is an orally available, potent and selective PARP1 and PARP2 inhibitor that is a poor substrate for drug transporters. AZD2461 exhibits a high efficacy in olaparib-resistant tumors that overexpress P-glycoprotein.

storage

Store at -20°C

AZD2461 Preparation Products And Raw materials

Raw materials

Preparation Products

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AZD2461 Suppliers

Canada 1 China 92 India 2 United Kingdom 1 United States 15 Global 111

Tocris Bioscience

Tel: --
Fax: --
Email: customerservice@tocris.co.uk
Country: United Kingdom
ProdList: 5726
Advantage: 77

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View Lastest Price from AZD2461 manufacturers

Henan Aochuang Chemical Co.,Ltd.

Product: AZD2461 1174043-16-3
Price: US $0.00-0.00/KG
Min. Order: 1KG
Purity: 98%
Supply Ability: 1Ton
Release date: 2022-10-13

Career Henan Chemical Co

Product: AZD2461 1174043-16-3
Price: US $3.00/KG
Min. Order: 1KG
Purity: 98%
Supply Ability: 100KG
Release date: 2020-01-29

1174043-16-3, AZD2461Related Search:

FLURBIPROFEN AXETIL Nintedanib SB525334 Veliparib Rapamycin PLX4032 Olaparib

4-[[4-fluoro-3-(4-methoxypiperidine-1-carbonyl)phenyl]methyl]-2H-phthalazin-1-one

4-[[4-Fluoro-3-[(4-methoxy-1-piperidinyl)carbonyl]phenyl]methyl]-1(2H)-phthalazinone

CS-739

AZD2461

4-[4-Fluoro-3-[(4-methoxypiperidin-1-yl)carbonyl]benzyl]phthalazin-1(2H)-one

1(2H)-Phthalazinone, 4-[[4-fluoro-3-[(4-methoxy-1-piperidinyl)carbonyl]phenyl]methyl]-

AZD 2461, >=98%

AZD2461 USP/EP/BP

4-(4-Fluoro-3-(4-methoxypiperidine-1-carbonyl)benzyl)phthalazin-1(2H)-one

AZD2461 AZD-2461

1174043-16-3

Inhibitors

Inhibitor