ChemicalBook > CAS DataBase List > SB 218795
SB 218795
- Product Name
- SB 218795
- CAS No.
- 174635-53-1
- Chemical Name
- SB 218795
- Synonyms
- SB 218795;Sb 218795r;Methyl (R)-2-phenyl-2-(2-phenylquinoline-4-carboxamido)acetate;methyl (2R)-2-phenyl-2-[(2-phenylquinoline-4-carbonyl)amino]acetate;(-)-(R)-N-(α-Methoxycarbonylbenzyl)-2-phenylquinoline-4-carboxamide;(-)-(R)-N-(ALPHA-METHOXYCARBONYLBENZYL)-2-PHENYLQUINOLINE-4-CARBOXAMIDE;(R)-[[(2-PHENYL-4-QUINOLINYL)CARBONYL]AMINO]-METHYL ESTER BENZENEACETIC ACID;Benzeneacetic acid, α-[[(2-phenyl-4-quinolinyl)carbonyl]amino]-, methyl ester, (αR)-;Benzeneacetic acid, alpha-(((2-phenyl-4-quinolinyl)carbonyl)amino)-, methyl ester, (alphar)-;constriction,SB-218795,Neurokinin Receptor,Inhibitor,neurokinin-3,NK receptor,pupillary,inhibit,Tachykinin receptor,SB218795,SB 218795,NK-3
- CBNumber
- CB7376630
- Molecular Formula
- C25H20N2O3
- Formula Weight
- 396.44
- MOL File
- 174635-53-1.mol
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SB 218795 Property
- Boiling point:
- 623.7±55.0 °C(Predicted)
- Density
- 1.237±0.06 g/cm3(Predicted)
- storage temp.
- 2-8°C
- solubility
- DMSO: 40 mg/mL, soluble
- form
- solid
- pka
- 11.41±0.46(Predicted)
- color
- white
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Safety
- WGK Germany
- 3
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N-Bromosuccinimide Price
Tocris
- Product number
- 1376
- Product name
- SB218795
- Purity
- ≥99%(HPLC)
- Packaging
- 10
- Price
- $174
- Updated
- 2021/12/16
Tocris
- Product number
- 1376
- Product name
- SB218795
- Purity
- ≥99%(HPLC)
- Packaging
- 50
- Price
- $713
- Updated
- 2021/12/16
TRC
- Product number
- S155070
- Product name
- SB218795
- Packaging
- 50mg
- Price
- $865
- Updated
- 2021/12/16
American Custom Chemicals Corporation
- Product number
- API0007579
- Product name
- SB 218795
- Purity
- 95.00%
- Packaging
- 50MG
- Price
- $1327.97
- Updated
- 2021/12/16
ApexBio Technology
- Product number
- B6710
- Product name
- SB218795
- Packaging
- 50mg
- Price
- $1362
- Updated
- 2021/12/16
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SB 218795 Chemical Properties,Usage,Production
Uses
SB 218795 is an NK3 receptor antagonist.
Definition
ChEBI: (2R)-2-[[oxo-(2-phenyl-4-quinolinyl)methyl]amino]-2-phenylacetic acid methyl ester is a member of quinolines.
Biological Activity
Potent, selective and competitive non-peptide NK 3 receptor antagonist (K i = 13 nM at hNK 3 ). Displays 90-fold and 7000-fold selectivity over hNK 2 and hNK 1 receptors respectively. Active in vivo , inhibiting agonist-induced pupillary constriction.
SB 218795 Preparation Products And Raw materials
Raw materials
Preparation Products
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SB 218795 Suppliers
174635-53-1, SB 218795Related Search:
CHEMBRDG-BB 9071014
SB 218795
N-(2-HYDROXYETHYL)ISONICOTINAMIDE, 99
FOR-D-PHG-OH
N-METHYL-1-QUINOLIN-4-YLMETHANAMINE
N-ME-D-PHG-OH
2-methylquinoline-4-carboxamide
D(-)-AC-ALPHA-PHENYLGLYCINOL