BQ-788
- Product Name
- BQ-788
- CAS No.
- 156161-89-6
- Chemical Name
- BQ-788
- Synonyms
- CS-1494;BQ-788 SODIUM;BQ789 Sodium Salt;1-ELAIDYLPHOSPHOCHOLINE, >97%;BQ788 SODIUM SALT; BQ 788 SODIUM SALT;BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-;N-cis-2,6-dimethylpiperidinocarbonyl-L-γMeLeu-D-Trp(COOMe)-D-Nle-ONa;2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle;DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl)
- CBNumber
- CB7710904
- Molecular Formula
- C34H52N5NaO7
- Formula Weight
- 665.81
- MOL File
- 156161-89-6.mol
BQ-788 Property
- storage temp.
- -20°C
- solubility
- acetonitrile: 0.3 mg/mL
- form
- solid
- color
- white
Safety
- WGK Germany
- 3
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
H315Causes skin irritation
H319Causes serious eye irritation
H335May cause respiratory irritation
- Precautionary statements
-
P261Avoid breathing dust/fume/gas/mist/vapours/spray.
P280Wear protective gloves/protective clothing/eye protection/face protection.
P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.
P302+P352IF ON SKIN: wash with plenty of soap and water.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
N-Bromosuccinimide Price
- Product number
- B157
- Product name
- BQ-788
- Purity
- ≥95%,solid
- Packaging
- 200μg
- Price
- $231
- Updated
- 2024/03/01
- Product number
- 17403
- Product name
- BQ-788 (sodium salt)
- Purity
- ≥95%
- Packaging
- 500μg
- Price
- $175
- Updated
- 2024/03/01
- Product number
- 17403
- Product name
- BQ-788 (sodium salt)
- Purity
- ≥95%
- Packaging
- 1mg
- Price
- $242
- Updated
- 2024/03/01
- Product number
- B676670
- Product name
- BQ788
- Packaging
- 5mg
- Price
- $595
- Updated
- 2021/12/16
- Product number
- CS-2685
- Product name
- BQ-788(sodiumsalt)
- Purity
- 98.03%
- Packaging
- 10mg
- Price
- $600
- Updated
- 2021/12/16
BQ-788 Chemical Properties,Usage,Production
Uses
BQ-788 has been used as a selective endothelin-B (ETRB) blocker in human airway smooth muscle cells (HASMCs), uterine mesothelial cells (UtMCs)-derived vascular smooth muscle cells (VSMCs), and human umbilical vein endothelial cells (HUVECs)
Biological Activity
Potent, selective ET B receptor antagonist (IC 50 = 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells).
Biochem/physiol Actions
Selective ETB endothelin receptor antagonist.
storage
+4°C