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PIRENPERONE

Product Name
PIRENPERONE
CAS No.
75444-65-4
Chemical Name
PIRENPERONE
Synonyms
PIRENPERONE;PIRENPERONE (R-47,465) >97% SEROTONIN 5- HT2 ANTAG;3-[2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one;3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one;3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one;4H-Pyrido[1,2-a]pyrimidin-4-one,3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-;R-47,465, 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido-[1,2-a] pyrimidin-4-one;R 47465,anxiolytic activity,Pirenperone,5-HT Receptor,Inhibitor,R47465,inhibit,5-hydroxytryptamine Receptor,Serotonin Receptor,R-47465
CBNumber
CB8504115
Molecular Formula
C23H24FN3O2
Formula Weight
393.45
MOL File
75444-65-4.mol
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PIRENPERONE Property

Boiling point:
556.3±60.0 °C(Predicted)
Density 
1.26±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
0.1 M HCl: 11 mg/mL
form 
solid
pka
7.91±0.10(Predicted)
color 
light yellow
Water Solubility 
Water: Insoluble
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Safety

WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

TRC
Product number
P508505
Product name
Pirenperone
Packaging
500mg
Price
$910
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
BRS0000667
Product name
PIRENPERONE
Purity
95.00%
Packaging
10MG
Price
$280.35
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
BRS0000667
Product name
PIRENPERONE
Purity
95.00%
Packaging
25MG
Price
$628.93
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
BRS0000667
Product name
PIRENPERONE
Purity
95.00%
Packaging
100MG
Price
$797.99
Updated
2021/12/16
Ambeed
Product number
A108159
Product name
3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
Purity
98%
Packaging
100mg
Price
$971
Updated
2021/12/16
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PIRENPERONE Chemical Properties,Usage,Production

Uses

5-HT2 antagonist

Uses

antianginal, antihypertensive

Uses

Pirenperone is a 5-HT2 serotonin receptor antagonist. Pirenperone also increases phosphorylation in human glioma cells by inhibiting cellular gap junctions.

Definition

ChEBI: 3-[2-[4-[(4-fluorophenyl)-oxomethyl]-1-piperidinyl]ethyl]-2-methyl-4-pyrido[1,2-a]pyrimidinone is an aromatic ketone.

PIRENPERONE Preparation Products And Raw materials

Raw materials

Preparation Products

75444-65-4, PIRENPERONERelated Search:


  • PIRENPERONE (R-47,465) >97% SEROTONIN 5- HT2 ANTAG
  • R-47,465, 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido-[1,2-a] pyrimidin-4-one
  • 3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
  • 3-[2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
  • 3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
  • 4H-Pyrido[1,2-a]pyrimidin-4-one,3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-
  • R 47465,anxiolytic activity,Pirenperone,5-HT Receptor,Inhibitor,R47465,inhibit,5-hydroxytryptamine Receptor,Serotonin Receptor,R-47465
  • PIRENPERONE
  • 75444-65-4
  • C23H24FN3O2
  • ADALAT