ChemicalBook > CAS DataBase List > Antazoline

Antazoline

Product Name
Antazoline
CAS No.
91-75-8
Chemical Name
Antazoline
Synonyms
5512-M;Avissul;Azalone;Antastan;Antasten;Antistin;Antazolin;Antistine;Chemiopen;Histostab
CBNumber
CB8667315
Molecular Formula
C17H19N3
Formula Weight
265.35
MOL File
91-75-8.mol
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Antazoline Property

Melting point:
120-122°
Boiling point:
398.57°C (rough estimate)
Density 
0.9786 (rough estimate)
refractive index 
1.6080 (estimate)
pka
pKa 6.65(H2O t = 25 I = 0.05) (Uncertain)
form 
A solid
color 
White to off-white
Water Solubility 
663.4mg/L(30 ºC)
CAS DataBase Reference
91-75-8(CAS DataBase Reference)
NIST Chemistry Reference
Antazoline(91-75-8)
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Safety

Hazardous Substances Data
91-75-8(Hazardous Substances Data)
Toxicity
LD50 oral in mouse: 398mg/kg
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H312Harmful in contact with skin

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P321Specific treatment (see … on this label).

P322Specific measures (see …on this label).

P330Rinse mouth.

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

P363Wash contaminated clothing before reuse.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Biosynth Carbosynth
Product number
FA30098
Product name
Antazoline
Packaging
100mg
Price
$70
Updated
2021/12/16
AK Scientific
Product number
G399
Product name
Antazoline
Packaging
100mg
Price
$98
Updated
2021/12/16
Biosynth Carbosynth
Product number
FA30098
Product name
Antazoline
Packaging
250mg
Price
$100
Updated
2021/12/16
Biosynth Carbosynth
Product number
FA30098
Product name
Antazoline
Packaging
500mg
Price
$160
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0007303
Product name
ANTAZOLINE
Purity
95.00%
Packaging
100MG
Price
$225.75
Updated
2021/12/16
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Antazoline Chemical Properties,Usage,Production

Chemical Properties

White, odorless crystalline powder with bitter taste. Sparingly soluble in alcohol and water; practically insoluble in benzene and ether.

Originator

Antistine HCl,Ciba,US,1948

Uses

Antihistaminic.

Definition

ChEBI: A member of the class of imidazolines that is 2-aminomethyl-2-imidazoline in which the exocyclic amino hydrogens are replaced by benzyl and phenyl groups. Antazoline is only found in individuals that have taken the drug.

Manufacturing Process

15.4 parts of 2-chloromethylimidazoline hydrochloride, 45.8 parts of Nbenzylaniline and 150 parts of alcohol are heated in an oil bath at 100° to 110°C. After distilling off the alcohol, the reaction mass is maintained at this temperature for a further 3 hours and then triturated with water and 10 parts of sodium bicarbonate. The unconsumed benzylaniline is extracted with ether and the aqueous solution neutralized with dilute hydrochloric acid. By evaporating this solution and extracting the residue with alcohol there is obtained 2-(N-phenyl-N-benzylaminomethyl)imidazoline hydrochloride in the form of colorless crystals of melting point 227° to 229°C.

Therapeutic Function

Antihistaminic

Clinical Use

Antazoline is used for local application to the eye in allergic conjunctivitis.

Safety Profile

Poison by ingestion, subcutaneous, and intraperitoneal routes. An eye irritant. When heated to decomposition it emits toxic fumes of NOx.

Antazoline Preparation Products And Raw materials

Raw materials

Preparation Products

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Antazoline Suppliers

LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky (shanghai) International Co.,Ltd
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
15402
Advantage
60
HBCChem, Inc.
Tel
+1-510-219-6317
Fax
+1-650-486-1361
Email
sales@hbcchem.com
Country
United States
ProdList
10648
Advantage
60
ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Fax
0755-28363542
Email
sales@chem-strong.com
Country
China
ProdList
18070
Advantage
56
Wuhan Dahua Pharmaceutical Co., Ltd.
Tel
027-59262863 13277907145 3091977954
Fax
027-59420980
Country
China
ProdList
4943
Advantage
58
Creative Peptides
Tel
Email
info@creative-peptides.com
Country
United States
ProdList
6083
Advantage
56
Amadis Chemical Company Limited
Tel
571-89925085
Fax
0086-571-89925065
Email
sales@amadischem.com
Country
China
ProdList
131957
Advantage
58
Jiangsu United-value International Trading Co., Ltd.
Tel
0519-89885611 89885616 15312500313
Fax
+86(519)89885615
Email
luke.li@uvcs.cn.com
Country
China
ProdList
469
Advantage
58
Aikon International Limited
Tel
025-58851090 13611564524
Fax
(6)02557626880
Email
lwan@aikonchem.com
Country
China
ProdList
15951
Advantage
58
Wuhan FengyaoTonghui Chemical Products Co., Ltd.
Tel
027-87466105 15377573527
Email
2678564200@qq.com
Country
China
ProdList
17987
Advantage
58
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View Lastest Price from Antazoline manufacturers

Shaanxi Dideu Medichem Co. Ltd
Product
Antazoline 91-75-8
Price
US $1.00-1.00/KG
Min. Order
1g
Purity
99%
Supply Ability
50tons
Release date
2020-05-11
Hebei Ganmiao New material Technology Co., LTD
Product
Antazoline 91-75-8
Price
US $13.00-7.00/kg
Min. Order
1kg
Purity
99.9%
Supply Ability
200ton
Release date
2024-06-19
Hebei Mojin Biotechnology Co.,Ltd
Product
Antazoline 91-75-8
Price
US $0.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
50000KG/month
Release date
2024-07-22

91-75-8, AntazolineRelated Search:


  • 1H-Imidazole-2-methanamine, 4,5-dihydro-N-phenyl-N-(phenylmethyl)-
  • 2-(N-Phenyl-N-benzylaminomethyl)imidazoline
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  • 2-[(N-Benzylanilino)methyl]-2-imidazoline
  • 2-Imidazoline, 2-[(N-benzylanilino)methyl]-
  • 2-Phenyl-benzyl-amino-methylimidazolin
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  • Imidazoline agonist; more potent than efaroxan in inducing insulin release from beta cells; H1 histamine receptor antagonist.