ANTAZOLINE PHOSPHATE

Product Name: ANTAZOLINE PHOSPHATE
CAS No.: 154-68-7
Chemical Name: ANTAZOLINE PHOSPHATE
Synonyms: ANTAZOLINE H3PO4;2-(N-Benzylanili;ANTISTIN PHOSPHATE;HISTOSAB PHOSPHATE;Antistine phosphate;ANTAZOLINE PHOSPHATE;ANTAZOLINE PHOSPHATE SALT;Antazoline Phosphate (200 mg);Antazoline Phosphate (1038003);ANTAZOLINE PHOSPHATE CRYSTALLINE
CBNumber: CB8771906
Molecular Formula: C17H22N3O4P
Formula Weight: 363.35
MOL File: 154-68-7.mol

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ANTAZOLINE PHOSPHATE Property

Melting point:: 194-198°
storage temp.: Refrigerator
solubility: DMSO, Methanol
color: White
CAS DataBase Reference: 154-68-7(CAS DataBase Reference)

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Safety

Hazard Codes: Xn
Risk Statements: 20/21/22-36/37/38
Safety Statements: 26-36
WGK Germany: 3
HS Code: 2933290000

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich

Product number: PHR3455
Product name: Antazoline Phosphate
Purity: certified reference material, pharmaceutical secondary standard
Packaging: 500MG
Price: $223.25
Updated: 2025/07/31

Sigma-Aldrich

Product number: 1038003
Product name: Antazoline phosphate
Purity: United States Pharmacopeia (USP) Reference Standard
Packaging: 200mg
Price: $406
Updated: 2025/07/31

Sigma-Aldrich

Product number: A3766
Product name: Antazoline phosphate salt
Purity: analytical standard, for drug analysis
Packaging: 1g
Price: $37.8
Updated: 2022/05/15

TRC

Product number: A678410
Product name: Antazoline phosphate
Packaging: 1g
Price: $90
Updated: 2021/12/16

TRC

Product number: A678410
Product name: Antazoline phosphate
Packaging: 10g
Price: $140
Updated: 2021/12/16

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ANTAZOLINE PHOSPHATE Chemical Properties,Usage,Production

Uses

Antazoline Phosphate acts as a histamine H1 receptor blocker, functioning as an antihistamine pharmaceutical.

General Description

Antazoline phosphate, 2-[(Nbenzylanilino)methyl]-2-imidazoline dihydrogen phosphate,is a bitter, white to off-white crystalline powder thatis soluble in water. It has a pKa of 10.0, and a 2% solutionhas a pH of about 4.5. Antazoline, like the ethylenediamines,contains an N-benzylanilino group linked to a basicnitrogen through a two-carbon chain.
Antazoline is less active than most of the other antihistaminicdrugs, but it is characterized by the lack of local irritation.The more soluble phosphate salt is applied topicallyto the eye in a 0.5% solution. The less soluble hydrochlorideis given orally. In addition to its use as an antihistamine, antazolinehas more than twice the local anesthetic potency ofprocaine and also exhibits anticholinergic actions.

Biological Activity

Imidazoline agonist; more potent than efaroxan in inducing insulin release from β cells; H1 histamine receptor antagonist.

in vivo

Antazoline phosphate (IP; 0.01 ml/g; 30min) as H1 receptor antagonists diminishes the anticonvulsant activity of carbamazepine and diphenylhydantoin^[3].

Animal Model:	Swiss mice^[3]
Dosage:	0.01 mL/g
Administration:	IP; 0.01 ml/g; 30min
Result:	Showed some proconvulsive activity.

ANTAZOLINE PHOSPHATE Preparation Products And Raw materials

Raw materials

Preparation Products

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ANTAZOLINE PHOSPHATE Suppliers

Canada 1 China 75 Germany 3 India 4 Japan 1 South Korea 1 Switzerland 2 United Kingdom 6 United States 22 Global 115

J & K SCIENTIFIC LTD.

Tel: 18210857532; 18210857532
Fax: 86-10-82849933
Email: jkinfo@jkchemical.com
Country: China
ProdList: 96815
Advantage: 76

Chemsky（shanghai）International Co.,Ltd.

Tel: 021-50135380
Email: shchemsky@sina.com
Country: China
ProdList: 32321
Advantage: 50

Sinopharm Chemical Reagent Co,Ltd.

Tel: 86-21-63210123
Fax: 86-21-63290778 86-21-63218885
Email: sj_scrc@sinopharm.com
Country: China
ProdList: 9815
Advantage: 79

BOC Sciences

Tel: 1-631-485-4226; 16314854226
Email: info@bocsci.com
Country: United States
ProdList: 12952
Advantage: 65

S.Z. PhyStandard Bio-Tech. Co., Ltd.

Tel: 0755-83725681-603
Fax: +86 755 28094224
Country: China
ProdList: 4496
Advantage: 50

3B Scientific (Wuhan) Corporation Limited

Tel: 027-88063677 18971314022;
Fax: 027-88063656
Email: sales@3bsc.com
Country: China
ProdList: 294
Advantage: 58

Creative Peptides

Tel
Email: info@creative-peptides.com
Country: United States
ProdList: 6083
Advantage: 56

Beijing Solarbio Science & Tecnology Co., Ltd.

Tel: 17801761073
Email: 3193328036@qq.com
Country: China
ProdList: 6338
Advantage: 68

Guangzhou Kafen Biotech Co.,Ltd

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Country: China
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Wuhai Shuou Technology Co., Ltd.

Tel: 17792809151
Fax: 18872220797
Email: 2355916837@ycphar.com
Country: China
ProdList: 6133
Advantage: 55

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View Lastest Price from ANTAZOLINE PHOSPHATE manufacturers

Hebei Chuanghai Biotechnology Co., Ltd

Product: ANTAZOLINE PHOSPHATE 154-68-7
Price: US $10.00/KG
Min. Order: 100KG
Purity: 99%
Supply Ability: 100 mt
Release date: 2024-11-20

Shaanxi Dideu Medichem Co. Ltd

Product: Antazoline phosphate 154-68-7
Price: US $0.00-0.00/KG
Min. Order: 1KG
Purity: 99.0%
Supply Ability: 1000KG
Release date: 2024-07-16

Career Henan Chemical Co

Product: ANTAZOLINE PHOSPHATE 154-68-7
Price: US $1.00/KG
Min. Order: 1KG
Purity: 98%
Supply Ability: 200kg
Release date: 2019-08-30

154-68-7, ANTAZOLINE PHOSPHATERelated Search:

Antazoline Phenamazoline 2-METHYL-2-IMIDAZOLINE DIETHYLAMINE PHOSPHATE Antazoline hydrochloride ANTAZOLINE PHOSPHATE

N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline

N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline hydrochloride

N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline hydrochloride

HISTOSAB PHOSPHATE

ANTISTIN PHOSPHATE

ANTAZOLINE H3PO4

ANTAZOLINE PHOSPHATE

ANTAZOLINE PHOSPHATE SALT

BENZYL-(4,5-DIHYDRO-1H-IMIDAZOL-2-YLMETHYL)-PHENYL-AMINE H3PO4

2-[(N-BENZYLANILINO)METHYL]-2-IMIDAZOLINE PHOSPHATE

2-(N-BENZYLANILINOMETHYL) IMIDAZOLINE PHOSPHATE

2-(N-PHENYL-N-BENZYL-AMINOMETHYL)-IMIDAZOLINE H3PO4

N-benzyl-4,5-dihydro-N-phenyl-1H-imidazole-2-methylamine monophosphate

ANTAZOLINE PHOSPHATE CRYSTALLINE

Antistine phosphate

Antazoline Phosphate (200 mg)

2-(N-Benzylanili

benzyl-(4,5-dihydro-1H-imidazol-2-ylmethyl)-phenyl-amine

benzyl-(4,5-dihydro-1H-imidazol-2-ylmethyl)-phenyl-amine hydrochloride

N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline,phosphoric acid

Antazoline Phosphate (1038003)

N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline,phosphoricaci

Antazoline phosphate salt analytical standard, for drug analysis

154-68-7

C17H22N3O4P

C17H19N3H3PO4

Imidazoline agonist; more potent than efaroxan in inducing insulin release from beta cells; H1 histamine receptor antagonist.

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