ChemicalBook > CAS DataBase List > ANTAZOLINE PHOSPHATE

ANTAZOLINE PHOSPHATE

Product Name
ANTAZOLINE PHOSPHATE
CAS No.
154-68-7
Chemical Name
ANTAZOLINE PHOSPHATE
Synonyms
ANTAZOLINE H3PO4;2-(N-Benzylanili;ANTISTIN PHOSPHATE;HISTOSAB PHOSPHATE;Antistine phosphate;ANTAZOLINE PHOSPHATE;ANTAZOLINE PHOSPHATE SALT;Antazoline Phosphate (200 mg);Antazoline Phosphate (1038003);ANTAZOLINE PHOSPHATE CRYSTALLINE
CBNumber
CB8771906
Molecular Formula
C17H22N3O4P
Formula Weight
363.35
MOL File
154-68-7.mol
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ANTAZOLINE PHOSPHATE Property

Melting point:
194-198°
storage temp. 
Refrigerator
solubility 
DMSO, Methanol
color 
White
CAS DataBase Reference
154-68-7(CAS DataBase Reference)
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Safety

Hazard Codes 
Xn
Risk Statements 
20/21/22-36/37/38
Safety Statements 
26-36
WGK Germany 
3
HS Code 
2933290000
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
PHR3455
Product name
Antazoline Phosphate
Purity
certified reference material, pharmaceutical secondary standard
Packaging
500MG
Price
$223.25
Updated
2025/07/31
Sigma-Aldrich
Product number
1038003
Product name
Antazoline phosphate
Purity
United States Pharmacopeia (USP) Reference Standard
Packaging
200mg
Price
$406
Updated
2025/07/31
Sigma-Aldrich
Product number
A3766
Product name
Antazoline phosphate salt
Purity
analytical standard, for drug analysis
Packaging
1g
Price
$37.8
Updated
2022/05/15
TRC
Product number
A678410
Product name
Antazoline phosphate
Packaging
1g
Price
$90
Updated
2021/12/16
TRC
Product number
A678410
Product name
Antazoline phosphate
Packaging
10g
Price
$140
Updated
2021/12/16
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ANTAZOLINE PHOSPHATE Chemical Properties,Usage,Production

Uses

Antazoline Phosphate acts as a histamine H1 receptor blocker, functioning as an antihistamine pharmaceutical.

General Description

Antazoline phosphate, 2-[(Nbenzylanilino)methyl]-2-imidazoline dihydrogen phosphate,is a bitter, white to off-white crystalline powder thatis soluble in water. It has a pKa of 10.0, and a 2% solutionhas a pH of about 4.5. Antazoline, like the ethylenediamines,contains an N-benzylanilino group linked to a basicnitrogen through a two-carbon chain.
Antazoline is less active than most of the other antihistaminicdrugs, but it is characterized by the lack of local irritation.The more soluble phosphate salt is applied topicallyto the eye in a 0.5% solution. The less soluble hydrochlorideis given orally. In addition to its use as an antihistamine, antazolinehas more than twice the local anesthetic potency ofprocaine and also exhibits anticholinergic actions.

Biological Activity

Imidazoline agonist; more potent than efaroxan in inducing insulin release from β cells; H1 histamine receptor antagonist.

in vivo

Antazoline phosphate (IP; 0.01 ml/g; 30min) as H1 receptor antagonists diminishes the anticonvulsant activity of carbamazepine and diphenylhydantoin[3].

Animal Model:Swiss mice[3]
Dosage:0.01 mL/g
Administration:IP; 0.01 ml/g; 30min
Result:Showed some proconvulsive activity.

ANTAZOLINE PHOSPHATE Preparation Products And Raw materials

Raw materials

Preparation Products

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View Lastest Price from ANTAZOLINE PHOSPHATE manufacturers

Hebei Chuanghai Biotechnology Co., Ltd
Product
ANTAZOLINE PHOSPHATE 154-68-7
Price
US $10.00/KG
Min. Order
100KG
Purity
99%
Supply Ability
100 mt
Release date
2024-11-20
Shaanxi Dideu Medichem Co. Ltd
Product
Antazoline phosphate 154-68-7
Price
US $0.00-0.00/KG
Min. Order
1KG
Purity
99.0%
Supply Ability
1000KG
Release date
2024-07-16
Career Henan Chemical Co
Product
ANTAZOLINE PHOSPHATE 154-68-7
Price
US $1.00/KG
Min. Order
1KG
Purity
98%
Supply Ability
200kg
Release date
2019-08-30

154-68-7, ANTAZOLINE PHOSPHATERelated Search:

Antazoline Phenamazoline 2-METHYL-2-IMIDAZOLINE DIETHYLAMINE PHOSPHATE Antazoline hydrochloride ANTAZOLINE PHOSPHATE

  • N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline
  • N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-N-(phenylmethyl)aniline hydrochloride
  • N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline hydrochloride
  • HISTOSAB PHOSPHATE
  • ANTISTIN PHOSPHATE
  • ANTAZOLINE H3PO4
  • ANTAZOLINE PHOSPHATE
  • ANTAZOLINE PHOSPHATE SALT
  • BENZYL-(4,5-DIHYDRO-1H-IMIDAZOL-2-YLMETHYL)-PHENYL-AMINE H3PO4
  • 2-[(N-BENZYLANILINO)METHYL]-2-IMIDAZOLINE PHOSPHATE
  • 2-(N-BENZYLANILINOMETHYL) IMIDAZOLINE PHOSPHATE
  • 2-(N-PHENYL-N-BENZYL-AMINOMETHYL)-IMIDAZOLINE H3PO4
  • N-benzyl-4,5-dihydro-N-phenyl-1H-imidazole-2-methylamine monophosphate
  • ANTAZOLINE PHOSPHATE CRYSTALLINE
  • Antistine phosphate
  • Antazoline Phosphate (200 mg)
  • 2-(N-Benzylanili
  • benzyl-(4,5-dihydro-1H-imidazol-2-ylmethyl)-phenyl-amine
  • benzyl-(4,5-dihydro-1H-imidazol-2-ylmethyl)-phenyl-amine hydrochloride
  • N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline,phosphoric acid
  • Antazoline Phosphate (1038003)
  • N-benzyl-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)aniline,phosphoricaci
  • Antazoline phosphate salt analytical standard, for drug analysis
  • 154-68-7
  • C17H22N3O4P
  • C17H19N3H3PO4
  • Imidazoline agonist; more potent than efaroxan in inducing insulin release from beta cells; H1 histamine receptor antagonist.
  • Analytical Standards
  • AM to AQ
  • Analytical Chromatography Product Catalog
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