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Tubulysin A,TubA

Product Name
Tubulysin A,TubA
CAS No.
205304-86-5
Chemical Name
Tubulysin A,TubA
Synonyms
TubA;CS-1324;Tubulysin A;Tubulysins A;Tubulysin A,TubA;(2S,4R)-4-[[2-[(1R,3R)-1-acetyloxy-4-methyl-3-[3-methylbutanoyloxymethyl-[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidine-2-carbonyl]amino]pentanoyl]amino]pentyl]-1,3-thiazole-4-carbonyl]amino]-5-(4-hydroxyphenyl)-2-methylpentanoicaci;Benzenepentanoic acid, γ-[[[2-[(1R,3R)-1-(acetyloxy)-4-methyl-3-[[(2S,3S)-3-methyl-2-[[[(2R)-1-methyl-2-piperidinyl]carbonyl]amino]-1-oxopentyl][(3-methyl-1-oxobutoxy)methyl]amino]pentyl]-4-thiazolyl]carbonyl]amino]-4-hydroxy-α-methyl-, (αS,γR)-
CBNumber
CB92518395
Molecular Formula
C43H65N5O10S
Formula Weight
844.07
MOL File
205304-86-5.mol
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Tubulysin A,TubA Property

Melting point:
106-108 °C(Solv: methanol (67-56-1); water (7732-18-5))
Boiling point:
979.9±65.0 °C(Predicted)
Density 
1.195±0.06 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
organic solvents: soluble
form 
film
pka
4.52±0.23(Predicted)
color 
colorless or white
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Safety

Hazard Codes 
T
Risk Statements 
23/24/25-36/37/38
Safety Statements 
36/37-45
RIDADR 
UN 2811 6.1 / PGIII
WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H301Toxic if swalloed

H311Toxic in contact with skin

H315Causes skin irritation

H319Causes serious eye irritation

H331Toxic if inhaled

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P311Call a POISON CENTER or doctor/physician.

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N-Bromosuccinimide Price

TRC
Product number
T897135
Product name
TubulysinA
Packaging
0.25mg
Price
$385
Updated
2021/12/16
TRC
Product number
T897135
Product name
TubulysinA
Packaging
1mg
Price
$1405
Updated
2021/12/16
TRC
Product number
T897135
Product name
TubulysinA
Packaging
2.5mg
Price
$2805
Updated
2021/12/16
TRC
Product number
T897135
Product name
TubulysinA
Packaging
5mg
Price
$4235
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
PEP0004574
Product name
TUBULYSIN A
Purity
95.00%
Packaging
1MG
Price
$2684.85
Updated
2021/12/16
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Tubulysin A,TubA Chemical Properties,Usage,Production

Uses

Tubulysin A is a novel antibiotic, which is anti-microtubule, anti-mitotic, an apoptosis inducer, anticancer, anti-angiogenic, and antiproliferative.

Definition

ChEBI: Tubulysin A is a diester and a carboxylic acid.

Biochem/physiol Actions

Tubulysin A is a novel antibiotic, which is anti-microtubule, anti-mitotic, apoptosis inducer, anticancer, anti-angiogenic, and antiproliferative. Tubulysins are cytotoxic peptides, which include 9 members (A-I). Tubulysin A has potential application as an anticancer agent. It arrests cells in the G2/M phase. Tubulysin A inhibits polymerization more efficiently than vinblastine and induces depolymerization of isolated microtubules. Tubulysin A has potent cytostatic effects on various tumor cell lines with IC50 in the picomolar range.

Tubulysin A,TubA Preparation Products And Raw materials

Raw materials

Preparation Products

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Tubulysin A,TubA Suppliers

Climax Product
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India
ProdList
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Music Valley Instruments Private Limited
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Oswal Band
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View Lastest Price from Tubulysin A,TubA manufacturers

Career Henan Chemical Co
Product
Tubulysin A,TubA 205304-86-5
Price
US $1.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
g/kg/Ton
Release date
2019-12-25

205304-86-5, Tubulysin A,TubARelated Search:


  • TubA
  • Tubulysin A
  • Tubulysin A,TubA
  • Tubulysins A
  • CS-1324
  • Benzenepentanoic acid, γ-[[[2-[(1R,3R)-1-(acetyloxy)-4-methyl-3-[[(2S,3S)-3-methyl-2-[[[(2R)-1-methyl-2-piperidinyl]carbonyl]amino]-1-oxopentyl][(3-methyl-1-oxobutoxy)methyl]amino]pentyl]-4-thiazolyl]carbonyl]amino]-4-hydroxy-α-methyl-, (αS,γR)-
  • (2S,4R)-4-[[2-[(1R,3R)-1-acetyloxy-4-methyl-3-[3-methylbutanoyloxymethyl-[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidine-2-carbonyl]amino]pentanoyl]amino]pentyl]-1,3-thiazole-4-carbonyl]amino]-5-(4-hydroxyphenyl)-2-methylpentanoicaci
  • 205304-86-5
  • C43H65N5O10S