ChemicalBook > CAS DataBase List > Val-cit-PAB-OH

Val-cit-PAB-OH

Product Name
Val-cit-PAB-OH
CAS No.
159857-79-1
Chemical Name
Val-cit-PAB-OH
Synonyms
H-Val-Cit-PAB-OH;(S)-2-((S)-2-amino-3-methylbutanamido)-N-(4-(hydroxymethyl)phenyl)-5-ureidopentanamide;EOS-61316;al-Cit-PAB-OH;H-Val-Cit-PAB;Val-cit-PAB-OH;(D)-VAL-CIT-PAB;NH2-Val-Cit-PAB;2-(4-(((2,6-dimethylbenzoyl)oxy)methyl)phenyl)aceticacid;L-Valyl-N5-(aminocarbonyl)-N-[4-(hydroxymethyl)phenyl]-L-ornithinamide
CBNumber
CB92715206
Molecular Formula
C18H29N5O4
Formula Weight
379.45
MOL File
159857-79-1.mol
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Val-cit-PAB-OH Property

Melting point:
168 °C(dec.)
Boiling point:
715.0±60.0 °C(Predicted)
Density 
1.243±0.06 g/cm3(Predicted)
storage temp. 
2-8°C(protect from light)
solubility 
DMF: 10 mg/ml; DMSO: 10 mg/ml; PBS (pH 7.2): 1 mg/ml
form 
powder to crystal
pka
13.75±0.46(Predicted)
color 
White to Almost white
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Safety

HS Code 
2924.29.7790
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

TCI Chemical
Product number
V0155
Product name
Val-Cit-PAB-OH
Packaging
25MG
Price
$160
Updated
2024/03/01
TCI Chemical
Product number
V0155
Product name
Val-Cit-PAB-OH
Packaging
100MG
Price
$482
Updated
2024/03/01
TRC
Product number
V091545
Product name
Val-cit-PAB-OH
Packaging
100mg
Price
$580
Updated
2021/12/16
ChemScene
Product number
CS-5171
Product name
Val-cit-PAB-OH
Purity
99.35%
Packaging
100mg
Price
$87
Updated
2021/12/16
AK Scientific
Product number
7337DL
Product name
Val-cit-PAB-OH
Packaging
5mg
Price
$103
Updated
2021/12/16
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Val-cit-PAB-OH Chemical Properties,Usage,Production

Description

Val-Cit-PAB-OH is a peptide cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs). The Val-Cit will specifically be cleaved by Cathepsin B.

Uses

Val-cit-PAB-OH acts as a reagent in the preparation of cell-penetrating peptidic GRP78 ligand for tumor cell-specific prodrug therapy, preparation of monomethylvaline derivative conjugates with ligands and antibodies for cancer treatment.

Val-cit-PAB-OH Preparation Products And Raw materials

Raw materials

Preparation Products

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Val-cit-PAB-OH Suppliers

TOKYO CHEMICAL INDUSTRY CO., LTD.
Tel
03-36680489
Fax
03-3668-0520
Email
Sales-JP@TCIchemicals.com
Country
Japan
ProdList
28387
Advantage
80
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View Lastest Price from Val-cit-PAB-OH manufacturers

Xian confluore Biological Technology Co., Ltd.
Product
Val-Cit-PAB-OH 159857-79-1
Price
US $0.00/g
Min. Order
5g
Purity
>95.00%
Supply Ability
5g
Release date
2024-03-29
Henan Aochuang Chemical Co.,Ltd.
Product
Val-cit-PAB-OH 159857-79-1
Price
US $0.00-0.00/KG
Min. Order
1KG
Purity
98%
Supply Ability
1Ton
Release date
2022-10-13
Career Henan Chemical Co
Product
Val-cit-PAB-OH 159857-79-1
Price
US $1.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
g/kg/Ton
Release date
2020-03-05

159857-79-1, Val-cit-PAB-OHRelated Search:


  • (S)-2-((R)-2-amino-3-methylbutanamido)-N-(4-(hydroxymethyl)phenyl)-5-ureidopentanamide
  • EOS-61316
  • (S)-2-((S)-2-amino-3-methylbutanamido)-N-(4-(hydroxymethyl)phenyl)-5-ureidopentanamide
  • L-Ornithinamide, L-valyl-N5-(aminocarbonyl)-N-[4-(hydroxymethyl)phenyl]-
  • Val-cit-PAB-OH
  • L-Valyl-N5-(aminocarbonyl)-N-[4-(hydroxymethyl)phenyl]-L-ornithinamide
  • NH2-Val-Cit-PAB
  • (D)-VAL-CIT-PAB
  • al-Cit-PAB-OH
  • H-Val-Cit-PAB-OH
  • 2-(4-(((2,6-dimethylbenzoyl)oxy)methyl)phenyl)aceticacid
  • H-Val-Cit-PAB
  • (2S)-2-[[(2S)-2-amino-3-methyl-butanoyl]amino]-N-[4-(hydroxymethyl)phenyl]-5-ureido-pentanamide
  • 159857-79-1
  • Linker
  • ADC LINKER
  • ADCs
  • ADC-Linkers