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Inhibitor Activator

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Chemical Name:
WH-4-023 (SRC inhibitor)
Chemical Name:
TG101348 (JAK inhibitor)
Chemical Name:
PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
Chemical Name:
PD184352 (MEK inhibitor)
Chemical Name:
ML324 (HISTONE DEMETHYLASE inhibitor)
Chemical Name:
KU0063794 (MTOR inhibitor)
Chemical Name:
JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
Chemical Name:
GSK1292263 (GPR agonist)
Chemical Name:
BYL719 (PI3K inhibitor)
Chemical Name:
BML-210 (HDAC inhibitor)
Structure:
Chemical Name:
2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)-
CAS:
745051-61-0
MF:
C20H23FN2O4S2
Chemical Name:
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
Chemical Name:
U-104 (CARBONIC ANHYDRASE INHIBITOR)
Chemical Name:
SALUBRINAL (PERK inhibitor)
Chemical Name:
FLAVOPIRIDOL HCL (CDK inhibitor)
Chemical Name:
DEFACTINIB (FAK inhibitor)
Chemical Name:
CEDIRANIB (VEGFR inhibitor)
Chemical Name:
BAY11-7082 (IΚB/IKK inhibitor)
Chemical Name:
(-)-BLEBBISTATIN (ATPASE inhibitor)
Chemical Name:
AG14361 (PARP1 inhibitor)
Chemical Name:
ACP-196 (BTK inhibitor)
Chemical Name:
ABT-737 (BCL-2 inhibitor)
Structure:
Chemical Name:
CK-2127107
CAS:
1345410-31-2
MF:
C19H18F2N6O
Chemical Name:
VILAZODONE (SSRI inhibitor)
Chemical Name:
TBA-354 (anti-tuberculosis)
Chemical Name:
SAG (HEDGEHOG/SMOOTHENED agonist)
Chemical Name:
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
Chemical Name:
OSU-03012 (PDK-1 inhibitor)
Chemical Name:
MONOMETHYL AURISTATIN E (microtubule-associated inhibitor)
Chemical Name:
ML141 (RHO inhibitor)
Chemical Name:
KN-93 PHOSPHATE (CAMK Inhibitor)
Chemical Name:
GSK126 (EZH2 inhibitor)
Chemical Name:
GELDANAMYCIN (HSP90 inhibitor)
Chemical Name:
GANT61 (HEDGEHOG/SMOOTHENED Inhibitor)
Chemical Name:
EPZ-6438 (E7438) (EZH2 inhibitor)
Chemical Name:
EMPAGLIFLOZIN (SGLT inhibitor)
Chemical Name:
DOXORUBICIN (TOPOISOMERASE inhibitor)
Chemical Name:
DAPT (Γ-SECRETASE inhibitor)
Chemical Name:
DACLATASVIR (HCV NS5A inhibitor)
Chemical Name:
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
Chemical Name:
CABOZANTINIB (VEGFR inhibitor)
Chemical Name:
BREFELDIN A (protein transport inhibitor)
Chemical Name:
BKM120 (PI3K inhibitor)
Chemical Name:
AKT INHIBITOR VIII (AKT inhibitor)
Chemical Name:
ABT-199 (BCL-2 inhibitor)
Structure:
Chemical Name:
Porfiromycin
CAS:
801-52-5
MF:
C16H20N4O5
Chemical Name:
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
Chemical Name:
TETRABENAZINE (VMAT-2 Inhibitor)
Chemical Name:
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
Chemical Name:
PLX4032 (RAF inhibitor)
Chemical Name:
PD123319 (RAAS inhibitor)
Chemical Name:
NS-2028 (SGC inhibitor)
Chemical Name:
NECROSTATIN-1 (TNF-ALPHA inhibitor)
Chemical Name:
ML323 (DUB inhibitor)
Chemical Name:
KU-55933 (ATM inhibitor)
Chemical Name:
(+)-JQ1 (BRD4 inhibitor)
Chemical Name:
GSK2141795 (AKT inhibitor)
Chemical Name:
GANETESPIB (HSP inhibitor)
Chemical Name:
ENZALUTAMIDE (MDV3100) (AR inhibitor)
Chemical Name:
BRIVANIB (VEGFR inhibitor)
Chemical Name:
BARDOXOLONE METHYL (IΚB/IKK inhibitor)
Chemical Name:
AZ20 (ATM/ATR inhibitor)
Chemical Name:
ARN-509 (ANDROGEN RECEPTOR Inhibitor)
Structure:
Chemical Name:
5-PREGNEN-3BETA-OL-20-ONE-16ALPHA-CARBONITRILE
CAS:
1434-54-4
MF:
C22H31NO2
Chemical Name:
TWS119 (GSK-3 inhibitor)
Chemical Name:
SC-514 (IΚB/IKK inhibitor)
Chemical Name:
ROMIDEPSIN (HDAC inhibitor)
Chemical Name:
REGADENOSON (ADENOSINE RECEPTOR agonist)
Chemical Name:
PYRIDONE 6 (JAK inhibitor)
Chemical Name:
PRT062607 HCL (SYK inhibitor)
Chemical Name:
PAZOPANIB (VEGFR inhibitor)
Chemical Name:
MLN9708 (20S PROTEASOME Inhibitor)
Chemical Name:
INDIPLON (GABA RECEPTOR Conditioner)
Chemical Name:
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
Chemical Name:
EVEROLIMUS (MTOR inhibitor)
Chemical Name:
ENTOSPLETINIB (SYK inhibitor)
Chemical Name:
DABRAFENIB (RAF inhibitor)
Chemical Name:
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
Chemical Name:
BMS-5 (LIMK inhibitor)
Chemical Name:
AZD7762 (CHK inhibitor)
Chemical Name:
AG1024 (IGF-1R inhibitor)
Chemical Name:
VISMODEGIB (HEDGEHOG/SMOOTHENED INHIBITOR)
Chemical Name:
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
Chemical Name:
PAC-1 (CASPASE Activator)
Chemical Name:
OSELTAMIVIR PHOSPHATE (NEURAMINIDASE Inhibitor)
Chemical Name:
MONENSIN (protein transport inhibitor)
Chemical Name:
LINIFANIB (VEGFR inhibitor)
Chemical Name:
LCZ696 (RAAS inhibitor)
Chemical Name:
IONOMYCIN (calcium ionophore)
Chemical Name:
HYDROXYUREA (DNA SYNTHESIS inhibitor)
Chemical Name:
GZD824 DIMESYLATE (BCR-ABL inhibitor)
Chemical Name:
FORETINIB (C-MET inhibitor)
Chemical Name:
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
Chemical Name:
CNX-774 (BTK inhibitor)
Chemical Name:
BIRB 796 (P38 MAPK Inhibitor)
Chemical Name:
BAY87-2243 (HIF inhibitor)
Chemical Name:
B-AP15 (DUB inhibitor)
Chemical Name:
APIXABAN (FACTOR XA Inhibitor)
Chemical Name:
TPA Deficient Plasma
Structure:
Chemical Name:
TUFTSIN
CAS:
9063-57-4
MF:
C21H40N8O6