Basic information Safety Supplier Related

Oosponol

Basic information Safety Supplier Related

Oosponol Basic information

Product Name:
Oosponol
Synonyms:
  • Oosponol
  • 4-(1-Oxo-2-hydroxyethyl)-8-hydroxyisocoumarin
  • 4-Glycolyl-8-hydroxyisocoumarin
  • 8-Hydroxy-4-(hydroxyacetyl)-1H-2-benzopyran-1-one
  • Lenzitin
  • Brn 1287762
  • Isocoumarin, 4-glycolyl-8-hydroxy-
CAS:
146-04-3
MW:
0
Mol File:
146-04-3.mol
More
Less

Oosponol Chemical Properties

LogP
0.789 (est)
More
Less

Safety Information

Toxicity
LD50 oral in rat: 250mg/kg
More
Less

Oosponol Usage And Synthesis

Uses

Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.Oospongol has strong antifungal activity against many antagonistic fungi[1][2].

in vivo

Oosponol (6.25 mg/kg, 3.1 mg/kg, ip, Once) can lower blood pressure in spontaneously hypertensive rats model[1].

Animal Model:Spontaneously hypertensive rats[1]
Dosage:6.25 mg/kg, 3.1 mg/kg
Administration:Intraperitoneal injection, once.
Result:The intraperitoneal injection of 6.25 mg/kg lowered the pressure from 186 mm to 138~112 mm, the intraperitoneal injection of 3.1 mg/kg lowered the pressure from 185 mm to 164~131 mm[1].
Animal Model:Spontaneously hypertensive rats[1]
Dosage:6.25 mg/kg, 3.1 mg/kg
Administration:Intraperitoneal injection, once.
Result:The intraperitoneal injection of 6.25 mg/kg lowered the pressure from 186 mm to 138~112 mm, the intraperitoneal injection of 3.1 mg/kg lowered the pressure from 185 mm to 164~131 mm.

References

[1] Umezawa H, et al.. Dopamine -hydroxylase inhibitor produced by Gloeophyllum striatum and its identity with oosponol. J Antibiot (Tokyo). 1972 Apr;25(4):239-42. DOI:10.7164/antibiotics.25.239
[2] Sonnenbichler J,et al. Influence of the Gloeophyllum metabolite oosponol and some synthetic analogues on protein and RNA synthesis in target cells. Eur J Biochem. 1997 May 15;246(1):45-9. DOI:10.1111/j.1432-1033.1997.t01-2-00045.x

OosponolSupplier

Shanghai Haozhixiang Biotechnology Co., Ltd
Tel
526763801 13301653310
Email
526763801@qq.com
TargetMol Chemicals Inc.
Tel
+1-781-999-5354; +17819995354
Email
marketing@targetmol.com
BOC Sciences
Tel
+1-631-485-4226
Email
inquiry@bocsci.com
Chengdu Jiuding Chemical Technology Co., Ltd. - Song Bo
Tel
18584079237
Email
312074905@qq.com
Zhejiang Huida Biotech Co., LTD
Tel
0571-89903882 18679456698
Email
mingxinzhu@huidabiotech.com