5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE
5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE Basic information
- Product Name:
- 5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE
- Synonyms:
-
- 3,5-DIHYDRO-5-METHYL-N-3-PYRIDINYLBENZO[1,2-B:4,5-B']DIPYRROLE-1(2H)-CARBOXAMIDE HYDROCHLORIDE
- 5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE
- SB 206553
- SB 206553 HYDROCHLORIDE
- N-3-PYRIDINYL-3,5-DIHYDRO-5-METHYL-BENZO[1,2-B:4,5-B']DIPYRROLE-1(2H)-CARBOXAMIDE HYDROCHLORIDE
- SB 206553 HCL
- 5-METHYL-3,5-DIHYDRO-2H-PYRROLO[2,3-F]INDOLE-1-CARBOXYLIC ACID PYRIDIN-3-YLAMIDE
- 5-methyl-1-(3-pyridylcarbamoyl)-1,2,3,5-tetrahydropyrrolo[2,3-f]indole hydrochloride
- CAS:
- 158942-04-2
- MF:
- C17H16N4O
- MW:
- 292.34
- Product Categories:
-
- Serotonin receptor
- pharmacetical
- Mol File:
- 158942-04-2.mol
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5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE Chemical Properties
- Boiling point:
- 575.4±50.0 °C(Predicted)
- Density
- 1.33±0.1 g/cm3(Predicted)
- storage temp.
- Desiccate at RT
- solubility
- H2O: 30 mg/mL
- form
- solid
- pka
- 13.50±0.20(Predicted)
- color
- brown
MSDS
- Language:English Provider:SigmaAldrich
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5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLE Usage And Synthesis
Uses
SB 206553 Hydrochloride is a 5-HT2 antagonist.
Definition
ChEBI: SB 206553 is a pyrroloindole.
Biological Activity
Potent and selective 5-HT 2B /5-HT 2C receptor antagonist (rat 5-HT 2B pA 2 = 8.89, human 5-HT 2C pK i = 7.92). Displays > 80-fold selectivity over all other 5-HT receptor subtypes and a variety of other receptors (pK i < 6). Centrally active following oral administration in vivo .
5-METHYL-1-(3-PYRIDYLCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO [2,3-F]INDOLESupplier
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