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(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride

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(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride Basic information

Product Name:
(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride
Synonyms:
  • (S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride
  • (S)-Dolaphenine hydrochloride
  • (R)-2-phenyl-1-(thiazol-2-yl)ethan-1-amine hydrochloride
  • (1S)-2-phenyl-1-(1,3-thiazol-2-yl)ethanamine, hydrochloride salt
  • (S)-alpha-(Phenylmethyl)-2-thiazolemethanamine monohydrochloride
  • (S)-2-phenyl-1-(thiazol-2-yl)ethan-1-amine hydrochloride
  • (S) Dolaphenine hydrochloride,(S)Dolaphenine hydrochloride
CAS:
135383-60-7
MF:
C11H13ClN2S
MW:
240.75
Mol File:
135383-60-7.mol
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(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride Chemical Properties

storage temp. 
Inert atmosphere,Room Temperature
solubility 
DMSO : ≥ 50 mg/mL (207.68 mM);Water : ≥ 50 mg/mL (207.68 mM)
form 
Solid
color 
Light yellow to yellow
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(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride Usage And Synthesis

Uses

(S)-Dolaphenine hydrochloride is a component of Dolastatin 10 (HY-15580). Dolastatin 10, an antineoplastic agent, inhibits tubulin polymerization[1].

References

[1] Zhou W , et al. A practical approach to asymmetric synthesis of dolastatin 10. Org Biomol Chem. 2017;15(29):6119-6131. DOI:10.1039/c7ob01395g

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