Basic information Definition Uses Reaction Preparation Suzuki reaction Safety Supplier Related
ChemicalBook >  Product Catalog >  Chemical Reagents >  Organic reagents >  Boric acid >  Bis(pinacolato)diboron

Bis(pinacolato)diboron

Basic information Definition Uses Reaction Preparation Suzuki reaction Safety Supplier Related

Bis(pinacolato)diboron Basic information

Product Name:
Bis(pinacolato)diboron
Synonyms:
  • 4,4,4',4',5,5,5',5'-OCTAMETHYL-2,2'-BL-1,3,2-DIOXABOROLANE
  • 4,4,4',4',5,5,5',5'-OCTAMETHYL-2,2'-BIS(1,3,2-DIOXABOROLANE)
  • 4,4,4',4',5,5,5',5'-OCTAMETHYL-2,2'-BI-1,3,2-DIOXABOROLANE
  • 4,4,4',4',5,5,5',5'-OCTAMETHYL-2,2-BI-1,3,2-DIOXABOROLANE
  • 4,4,5,5,4',4',5',5'-OCTAMETHYL-[2,2']BI[[1,3,2]DIOXABOROLANYL]
  • BIS(2,2,3,3-TETRAMETHYL-2,3-BUTANEDIONATO)DIBORON
  • BIS(PINACOLATO)DIBORANE
  • DIBORON PINACOL ESTER
CAS:
73183-34-3
MF:
C12H24B2O4
MW:
253.94
EINECS:
615-925-0
Product Categories:
  • Reagent
  • Organoborons
  • Miscellaneous
  • Diboron Esters
  • B (Classes of Boron Compounds)
  • CHIRAL CHEMICALS
  • blocks
  • BoronicAcids
  • Small molecule
  • Aliphatics
  • Boronic Acids & Esters
  • DIBORON SERIES
  • Boronic Acids & Esters
  • OLED materials,pharm chemical,electronic
  • Pharmaceutical Intermediates
  • Boron Compounds
  • 73183-34-3
  • OLED
Mol File:
73183-34-3.mol
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Bis(pinacolato)diboron Chemical Properties

Melting point:
137-140 °C(lit.)
Boiling point:
222.6±7.0 °C(Predicted)
Density 
0.98
storage temp. 
Keep in dark place,Sealed in dry,Room Temperature
solubility 
Chloroform (Slightly), Methanol (Slightly)
form 
Powder or Platelets
color 
White
Water Solubility 
Soluble in tetrahydrofuran, dichloromethane, toluene, hexane and heptane. Insoluble in water.
Sensitive 
moisture sensitive
Merck 
14,1300
BRN 
7703552
InChIKey
IPWKHHSGDUIRAH-UHFFFAOYSA-N
CAS DataBase Reference
73183-34-3(CAS DataBase Reference)
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Safety Information

Hazard Codes 
Xi,Xn
Risk Statements 
36/37/38-20/21/22
Safety Statements 
26-37/39-36-24/25
WGK Germany 
3
Hazard Note 
Irritant
TSCA 
No
HazardClass 
IRRITANT, IRRITANT-HARMFUL, KEEP COLD
HS Code 
29349990

MSDS

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Bis(pinacolato)diboron Usage And Synthesis

Definition

Bis(pinacolato)diboron is a covalent compound containing two boron atoms and two pinacolato ligands. It has the formula [(CH3)4C2O2B]2; the pinacol groups are sometimes abbreviated as "pin", so the structure is sometimes represented as B2pin2.

Uses

It is a colourless solid that is soluble in organic solvents. It is a commercially available reagent for making pinacol boronic esters for organic synthesis. Unlike some other diboron compounds, B2pin2 is not moisture-sensitive and can be handled in air.

Reaction

  1. Reagent used for the synthesis of aryl, alkenyl, allyl and alkylboronic esters.
  2. Reagent used for the borylation of an α,β-unsaturated ketones.
  3. Reagent used for the synthesis of precursors for conducting polymers.
  4. Reagent used for the synthesis of in vivo fluorescent probes.
  5. Reagent used for the diborylation of alkynes. 


Preparation

Bis(pinacolato)diboron may be prepared by reacting tetrakis(dimethylamino)diboron with pinacol in acidic conditions. The B-B bond length is 1.711(6) Å.
The B-B bond adds across alkenes and alkynes to give the 1,2-diborylated alkanes and alkenes. Using various organorhodium or organoiridium catalysts, it can also be installed onto saturated hydrocarbons: CH3(CH2)6CH3 + [pinB]2 → pinBH + CH3(CH2)7Bpin These reactions proceed via boryl complexes.

Suzuki reaction

In the Suzuki reaction, Bis (pinacolato) diboron has the advantages of high reaction selectivity, mild conditions, and high yield. For some compounds that are unstable or need to improve the selectivity of the reaction, Bis (pinacolato) diboron and aryl halide are used. React is a good choice.

Chemical Properties

Bis(pinacolato)diboron is a white crystal powder, It is commonly used coupling reagent.

Uses

As a boron source in Pt-mediated diborations, coupling reactions; in Rh-or Ir-mediated borylations of alkanes and arenes, and in carbenoid chemistry.

Uses

suzuki reaction

Uses

Bis(pinacolato)diboron is used as a condensation agent in the preparation poly(arylene)s. Bis(pinacolato)diboron is an organoboranate with potential use as matrix metallo-proteinase (MMP-2) inhibitor.

Definition

ChEBI: Bis(pinacolato)diboron is a 1,3,2-dioxaborolane that is 4,4,5,5-tetramethyl-1,3,2-dioxaborolane in which the boron hydrogen at position 2 is replaced by a 4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl group. It is a reagent used in organic synthesis to synthesise pinacol boronic esters. It has a role as an EC 3.4.24.24 (gelatinase A) inhibitor.

General Description

Bis(pinacolato)diboron or (B2pin2) is the most commonly used diborane reagent in organic synthesis due to its high stability in air and moisture. It can be synthesized by treating tetrakis(dimethylamino)diboron with pinacol in acidic conditions.

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