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Etamsylate

Basic information Safety Supplier Related

Etamsylate Basic information

Product Name:
Etamsylate
Synonyms:
  • altodor
  • e141
  • eselin
  • md141
  • 2,5-dihydroxy-benzenesulfonicacicompd.withdiethylamine
  • 2,5-dihydroxy-benzenesulfonicacicompd.withn-ethylethanamine(1:1)
  • 2,5-dihydroxybenzenesulfonicacidcompd.withn-ethylethanamine
  • 2,5-DihydroxybenzenesulfonicacidcompdwithN-ethylethanamine
CAS:
2624-44-4
MF:
C10H17NO5S
MW:
263.31
EINECS:
220-090-7
Product Categories:
  • Other APIs
  • For the prevention and treatment of bleeding before surgery, but for intestinal bleeding, bleeding and urinary tract bleeding, etc
  • Amines
  • Aromatics
  • Intermediates & Fine Chemicals
  • API
  • Pharmaceuticals
  • Sulfur & Selenium Compounds
  • 2624-44-4
Mol File:
2624-44-4.mol
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Etamsylate Chemical Properties

Melting point:
125°
Density 
1.3441 (rough estimate)
refractive index 
1.5060 (estimate)
storage temp. 
Keep in dark place,Inert atmosphere,Room temperature
solubility 
Very soluble in water, freely soluble in methanol, soluble in anhydrous ethanol, practically insoluble in methylene chloride.
form 
Solid
color 
White to Pale Red
Merck 
14,3722
Stability:
Hygroscopic
InChI
InChI=1S/C6H6O5S.C4H11N/c7-4-1-2-5(8)6(3-4)12(9,10)11;1-3-5-4-2/h1-3,7-8H,(H,9,10,11);5H,3-4H2,1-2H3
InChIKey
HBGOLJKPSFNJSD-UHFFFAOYSA-N
SMILES
C1(S(=O)(=O)O)=CC(=CC=C1O)O.N(CC)CC
CAS DataBase Reference
2624-44-4(CAS DataBase Reference)
EPA Substance Registry System
Ethamsylate (2624-44-4)
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Safety Information

RTECS 
DB6145000
HS Code 
2921.19.6190
HazardClass 
IRRITANT
Toxicity
LD50 i.v. in mice, rats: 800, 1350 mg/kg (Esteve)

MSDS

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Etamsylate Usage And Synthesis

Chemical Properties

White Solid

Uses

Haemostatic / Anti Coagulant

Uses

Hemostatic;prostaglandin synthesis inhibitor

Definition

ChEBI: Etamsylate is a sulfonic acid derivative and an organosulfur compound.

Mechanism of action

Etamsylate is an antihaemorrhagic and vasoprotective agent. It increases platelet adhesiveness and capillary vascular wall resistance, thereby reducing capillary exudation and blood loss.

Clinical Use

Short-term treatment of blood loss in menorrhagia
Prophylaxis of surgical bleeding (unlicensed)

Side effects

Significant: Hypotension (parenteral). Rarely, severe hypersensitivity reaction, including anaphylaxis.
Blood and lymphatic system disorders: Parenteral: Rarely, neutropenia, agranulocytosis, thrombocytopenia.
Gastrointestinal disorders: Nausea, vomiting, diarrhoea, abdominal pain or discomfort.
General disorders and administration site conditions: Asthenia (parenteral). Rarely, fever.
Musculoskeletal and connective tissue disorders: Rarely, arthralgia.
Nervous system disorders: Headache.
Skin and subcutaneous tissue disorders: Rash.
Vascular disorders: Rarely, thromboembolism (parenteral).

Metabolism

Etamsylate is excreted unchanged, mainly in the urine.

Etamsylate Preparation Products And Raw materials

Raw materials

EtamsylateSupplier

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