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K145 (hydrochloride)

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K145 (hydrochloride) Basic information

Product Name:
K145 (hydrochloride)
Synonyms:
  • SphK2 inhibitor
  • SPHK2 INHIBITOR;K 145 HYDROCHLORIDE;K-145 HYDROCHLORIDE
  • K145 (hydrochloride)
  • K145(HCl)
  • 3-(2-Aminoethyl)-5-[3-(4-butoxyphenyl)propylidene]-2,4-thiazolidinedione hydrochloride (1:1)
  • 3-(2-Amino-ethyl)-5-[3-(4-butoxyl-phenyl)-propylidene]-thiazolidine-2,4-dione hydrochloride
  • K14 (hydrochloride)
  • K145 hydrochloride >=98% (HPLC)
CAS:
1449240-68-9
MF:
C18H25ClN2O3S
MW:
384.9207
Product Categories:
  • API
Mol File:
1449240-68-9.mol
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K145 (hydrochloride) Chemical Properties

storage temp. 
2-8°C
solubility 
DMSO: soluble20mg/mL, clear
form 
powder
color 
white to beige
InChI
1S/C18H24N2O3S.ClH/c1-2-3-13-23-15-9-7-14(8-10-15)5-4-6-16-17(21)20(12-11-19)18(22)24-16;/h6-10H,2-5,11-13,19H2,1H3;1H/b16-6-;
InChIKey
HADFDMGQKBGVAV-NKBLJONXSA-N
SMILES
S1\C(=C/CCc2ccc(cc2)OCCCC)\C(=O)N(C1=O)CCN.Cl
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Safety Information

WGK Germany 
3
Storage Class
11 - Combustible Solids
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K145 (hydrochloride) Usage And Synthesis

Uses

K145 hydrochloride has been used in the analysis of apoptosis.

General Description

K145 hydrochloride (3-(2-Amino-ethyl)-5-[3-(4-butoxyl-phenyl)-propylidene]-thiazolidine-2,4-dione) is an analog of sphingosine.

Biochem/physiol Actions

It has the ability to prevent leukemia cell growth in vitro.

in vivo

K145 (50 mg/kg; oral gavage; daily; for 15 days; BALB/c-nu mice) treatment significantly inhibits the growth of U937 tumors in nude mice[1].

Animal Model:BALB/c-nu mice injected with U937 cells[1]
Dosage:50 mg/kg
Administration:Oral gavage; daily; for 15 days
Result:Inhibited the growth of U937 tumors at 50 mg/kg dose and no apparent toxicity was observed.

IC 50

SphK2

K145 (hydrochloride)Supplier

Shanghai Boyle Chemical Co., Ltd.
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sales@boylechem.com
Haoyuan Chemexpress Co., Ltd.
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021-58950125
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info@chemexpress.com
MedChemexpress LLC
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021-58955995
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Bide Pharmatech Ltd.
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400-400-164-7117 18317119277
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product02@bidepharm.com
LETOPHARM LIMITED
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+86-21-5821 5861
Email
sales@letopharm.com
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K145 (hydrochloride)(1449240-68-9)Related Product Information