TELENZEPINE DIHYDROCHLORIDE
TELENZEPINE DIHYDROCHLORIDE Basic information
- Product Name:
- TELENZEPINE DIHYDROCHLORIDE
- Synonyms:
-
- 4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE
- TELENZEPINE DIHYDROCHLORIDE
- TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN
- 4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride
- Telenzepine dihydrochloide
- Telenzepine hydrate dihydrochloride
- 4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)
- JTQJFSQQHGPLOX-UHFFFAOYSA-N
- CAS:
- 147416-96-4
- MF:
- C19H22N4O2S
- MW:
- 370.47
- Product Categories:
-
- Acetylcholine receptor
- Mol File:
- 147416-96-4.mol
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TELENZEPINE DIHYDROCHLORIDE Chemical Properties
- storage temp.
- Store at RT
- solubility
- H2O: >10 mg/mL
- form
- solid
- color
- white
- Water Solubility
- Soluble to 100 mM in water
MSDS
- Language:English Provider:SigmaAldrich
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TELENZEPINE DIHYDROCHLORIDE Usage And Synthesis
Uses
Antiulcerative;M1 muscarinic antagonist
Uses
Telenzepine dihydrochloride is a potent and selective muscarnic receptor antagonist.
Uses
Telenzepine dihydrochloride hydrate was used to study M1 muscarinic receptor-mediated signaling in juvenile rat hippocampus and rat urinary bladder.
Biological Activity
Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion.
Biochem/physiol Actions
Telenzepine is an analog of pirenzepine and inhibits the secretion of gastric acid. It is an antagonist to M1-receptor and targets the oxyntic gastric glands and the salivary glands.
storage
Desiccate at RT
TELENZEPINE DIHYDROCHLORIDESupplier
3B Pharmachem (Wuhan) International Co.,Ltd.
- Tel
- 821-50328103-801 18930552037
- 3bsc@sina.com
BOC Sciences
- Tel
- 1-631-485-4226; 16314854226
- info@bocsci.com
Shanghai TaoSu Biochemical Technology Co., Ltd.
- Tel
- 021-33632979
- info@tsbiochem.com
Sigma-Aldrich
- Tel
- 021-61415566 800-8193336
- orderCN@merckgroup.com
EMMX Biotechnology LLC
- Tel
- 888-539-0666
- info@emmx.com
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TELENZEPINE DIHYDROCHLORIDE(147416-96-4)Related Product Information
- Pirenzepine hydrochloride
- N1-(2-AMINOPHENYL)-N2,N2-DIMETHYLGLYCINAMIDE
- N-(2-aminophenyl)-2-(4-methylpiperazin-1-yl)acetamide
- telenzepine dihydrochloride hydrate
- PIPERAZINE ACETIC ACID ANILIDE DIHYDROCHLORIDE
- N-(2-aminophenyl)-2-(diethylamino)acetamide
- TELENZEPINE DIHYDROCHLORIDE
- 2-PIPERAZINE-1-YL-ACETAMIDE
- (PIPERAZIN-1-YL)-ACETAMIDE X 2 HCL X 1/2 H2O