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PDK1 inhibitor

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PDK1 inhibitor Basic information

Product Name:
PDK1 inhibitor
Synonyms:
  • PDK1 inhibitor
  • PDK1 inhibitor 7
  • 1-[(3,4-Difluorophenyl)methyl]-N-[(1R)-2-[(2,3-dihydro-2-oxo-1H-benzimidazol-5-yl)oxy]-1-phenylethyl]-1,2-dihydro-2-oxo-3-pyridinecarboxamide
  • 3-PyridinecarboxaMide, 1-[(3,4-difluorophenyl)Methyl]-N-[(1R)-2-[(2,3-dihydro-2-oxo-1H-benziMidazol-5-yl)oxy]-1-phenylethyl]-1,2-dihydro-2-oxo-
  • MP7
  • 2-dihydro-2-oxo-
  • 3-dihydro-2-oxo-1H-benzimidazol-5-yl)oxy]-1-phenylethyl]-1
  • 4-difluorophenyl)methyl]-N-[(1R)-2-[(2
CAS:
1001409-50-2
MF:
C28H22F2N4O4
MW:
516.5
Mol File:
1001409-50-2.mol
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PDK1 inhibitor Chemical Properties

Boiling point:
724.4±60.0 °C(Predicted)
Density 
1.398
storage temp. 
Store at -20°C
solubility 
Soluble in DMSO
form 
Powder
pka
11.48±0.20(Predicted)
color 
Light yellow to yellow
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PDK1 inhibitor Usage And Synthesis

Uses

MP7 (PDK1 inhibitor) is a phosphoinositide-dependent kinase-1 (PDK1) inhibitor.

Definition

ChEBI: 1-[(3,4-difluorophenyl)methyl]-2-oxo-N-[(1R)-2-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)oxy]-1-phenylethyl]-3-pyridinecarboxamide is a member of benzimidazoles.

target

PDK1

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