Basic information Safety Supplier Related

LENAMPICILLIN HYDROCHLORIDE

Basic information Safety Supplier Related

LENAMPICILLIN HYDROCHLORIDE Basic information

Product Name:
LENAMPICILLIN HYDROCHLORIDE
Synonyms:
  • (5-methyl-2-oxo-1,3-dioxolen-4-yl)methyl-d-alpha-aminobenzylpenicillinatehyd
  • -2-carboxylicacid,hydrochloride
  • -amino-2-phenylacetamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane
  • ampicillin,(5-methyl-2-oxo-1,3-dioxolen-4-yl)methylester,hydrochloride
  • carbonicacid,cyclic1-(hydroxymethyl)-2-methylethyleneester,esterwith6-(2
  • kb1585
  • kbt1585
  • kbt-1585
CAS:
80734-02-7
MF:
C21H23N3O7S
MW:
461.49
Product Categories:
  • Amines
  • Drug Analogues
  • Heterocycles
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • Sulfur & Selenium Compounds
Mol File:
80734-02-7.mol
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LENAMPICILLIN HYDROCHLORIDE Chemical Properties

Melting point:
145° (dec)
storage temp. 
Store at -20°C, sealed storage, away from moisture and light
solubility 
DMSO:100.0(Max Conc. mg/mL);200.82(Max Conc. mM)
form 
Solid
color 
White to off-white
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Safety Information

Toxicity
LD50 in male, female rats, male, female mice (mg/kg): approx 10000, approx 10000, 8294, 8492 orally; 4362, 4471, 3576, 4284 s.c.; 876, 838, 711, 775 i.v.; in dogs (mg/kg): >300 orally (Ogino)
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LENAMPICILLIN HYDROCHLORIDE Usage And Synthesis

Uses

Lenampicillin is an oral ampicillin prodrug. Antibiotic used in the treatment of respiratory tract infections and urinary tract infections.

Definition

ChEBI: Valacillin (TN) is a peptide.

in vivo

Lenampicillin hydrochloride (KBT-1585) (oral adminstration; 0-1000 mg/kg) does not lead to death in dogs, and maximum dose of in this acute toxicity study is recorded because of causing emesis[2].Lenampicillin hydrochloride (LAPC) are identified for it main metabolites in rat and dogs. The main metabolite in peripheral plasma is 2,3-butanediol in rats and dog, On the other hand, high levels of acetoin is found in portal plasma for early period after dosing of LAPC. These results shows that the biotransformation of promoiety in LAPC to acetoin carried out mainly in intestinal tissues, but acetoin is converted to 2,3-butanediol in liver[3].

LENAMPICILLIN HYDROCHLORIDESupplier

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