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PHENPROCOUMON

Product Name
PHENPROCOUMON
CAS No.
435-97-2
Chemical Name
PHENPROCOUMON
Synonyms
MARCUMA;Fencumar;Liquamar;Marcumar;Falithrom;Falithiom;Marcoumar;RO 1-4849;Phenprocumon;PHENPROCOUMON
CBNumber
CB1295890
Molecular Formula
C18H16O3
Formula Weight
280.32
MOL File
435-97-2.mol
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PHENPROCOUMON Property

Melting point:
179-180°
Boiling point:
463.2±45.0 °C(Predicted)
Density 
1.261±0.06 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
Chloroform (Slightly), Methanol (Slightly)
form 
Solid
pka
4.50±1.00(Predicted)
color 
White to Off-White
EPA Substance Registry System
Phenprocoumon (435-97-2)
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Safety

RIDADR 
2811
HazardClass 
6.1(b)
PackingGroup 
III
Hazardous Substances Data
435-97-2(Hazardous Substances Data)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H301Toxic if swalloed

H311Toxic in contact with skin

H331Toxic if inhaled

H370Causes damage to organs

Precautionary statements

P260Do not breathe dust/fume/gas/mist/vapours/spray.

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P307+P311IF exposed: call a POISON CENTER or doctor/physician.

P311Call a POISON CENTER or doctor/physician.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P321Specific treatment (see … on this label).

P322Specific measures (see …on this label).

P330Rinse mouth.

P361Remove/Take off immediately all contaminated clothing.

P363Wash contaminated clothing before reuse.

P403+P233Store in a well-ventilated place. Keep container tightly closed.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

TRC
Product number
P318820
Product name
Phenprocoumon
Packaging
100mg
Price
$95
Updated
2021/12/16
Usbiological
Product number
165912
Product name
Phenprocoumon
Packaging
1g
Price
$460
Updated
2021/12/16
TRC
Product number
P318820
Product name
Phenprocoumon
Packaging
1g
Price
$775
Updated
2021/12/16
TRC
Product number
P318820
Product name
Phenprocoumon
Packaging
500mg
Price
$425
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0003816
Product name
PHENPROCOUMON
Purity
95.00%
Packaging
1G
Price
$450
Updated
2021/12/16
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PHENPROCOUMON Chemical Properties,Usage,Production

Chemical Properties

White Solid

Originator

Liquamar ,Organon ,US,1958

Uses

Phenprocoumon is known for being an oral anti-coagulant.

Definition

ChEBI: A hydroxycoumarin that is 4-hydroxycoumarin which is substituted at position 3 by a 1-phenylpropyl group.

Manufacturing Process

8.3 parts by weight of powdered sodium in 300 parts by volume of benzene, 100 parts by weight of diethyl (1'-phenylpropyl)-malonate and 72 parts by weight of acetylsalicylic acid chloride are reacted together to form diethyl 1(o-acetoxybenzoy1)-1-(1'-phenylpropyl)malonate, which boils at 195°198°C/0.03 mm Hg.
10.3 parts of weight of diethyl 1-(o-acetoxybenzoyl)-1-(1'-phenylpropyl)malonate are dissolved in 60 parts by volume of absolute ether and to this solution are added portion. wise at 10°C, while stirring, 2.6 parts by weight of sodium methylate. The reaction mixture is stirred for 4 hours, whereupon it is poured into ice water. The ether solution is washed neutral with ice water. After having distilled off the ether, a thick oil consisting of 3-carbethoxy-3-(1'phenylpropyl)-4-oxo-dihydrocoumarinis obtained. This compound crystallized in butyl oxide and has a MP of 108°-109°C.
The 3-carbethoxy-3-(1'-phenylpropyl)-4-oxo-dihydrocoumarinmay be hydrolyzed and decarboxylated as follows. The crude product is heated to 85°C for 1/2 hour with 100 parts by volume of 5% aqueous sodium hydroxide, while agitating or stirring. To remove traces of undissolved oil, the cooled solution is treated with 1 part by weight of charcoal, whereupon it is filtrated and acidified to Congo reaction with dilute sulfuric acid. The 3-(1'phenylpropyl)-4-hydroxycoumarin formed is separated off and recrystallized in 80% ethanol, whereupon it melts at 178°-179°C according to US Patent 2,701,804.

brand name

Liquamar (Organon).

Therapeutic Function

Anticoagulant

Synthesis

Phenprocoumon, 3-(|á-ethylbenzyl)-4-hydroxycoumarin (24.1.14), is synthesized by acylating sodium salts of diethyl ester (1-phenylpropyl)butyric acid with acetylsalicylic acid chloride, which forms the compound 24.1.12, which upon reaction with sodium ethoxide cyclizes to 3-(|á-ethylbenzyl)-2-carboethoxy-4-hydroxycoumarin (24.1.13). Alkaline hydrolysis of this product and further decarboxylation gives phenprocoumon(24.1.14).

PHENPROCOUMON Preparation Products And Raw materials

Raw materials

Preparation Products

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PHENPROCOUMON Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky(shanghai)International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
Advantage
50
Shanghai Sunway Pharmaceutical Technology Co., Ltd
Tel
021-51613915-820 13611835272
Fax
021 51613951
Email
mmwang@sunwaypharm.cn
Country
China
ProdList
9734
Advantage
57
BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
ProdList
14055
Advantage
65
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Wuhan Kaymke Chemical Co., Ltd.,
Tel
027-027-87342388 18086026008
Fax
027-87342388
Email
sales@kaymke.com
Country
China
ProdList
3881
Advantage
55
AdooQ BioScience, LLC
Tel
+1 (866) 930-6790
Fax
+1 (866) 333-9607
Email
info@adooq.com
Country
United States
ProdList
2782
Advantage
58
Bide Pharmatech Ltd.
Tel
400-164-7117 13681763483
Fax
+86-21-61629029
Email
product02@bidepharm.com
Country
China
ProdList
41462
Advantage
60
ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Fax
0755-28363542
Email
sales@chem-strong.com
Country
China
ProdList
18042
Advantage
56
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View Lastest Price from PHENPROCOUMON manufacturers

Honest Joy Holdings Limited
Product
4-Hydroxy-3-(1-phenylpropyl)-2H-chromen-2-on 435-97-2
Price
US $0.00/KG
Min. Order
1KG
Purity
97.4%
Supply Ability
100 tons
Release date
2022-02-20

435-97-2, PHENPROCOUMONRelated Search:


  • PHENPROCOUMON
  • 2H-1-Benzopyran-2-one, 4-hydroxy-3-(1-phenylpropyl)-
  • 3-(1-Phenylpropyl)-4-hydroxycoumarin
  • 3-(1'-Phenyl-propyl)-4-oxycoumarin
  • 3-(alpha-Ethylbenzyl)-4-hydroxycoumarin
  • 4-Hydroxy-3-(1-phenylpropyl)-2H-1-benzopyran-2-one
  • 4-Hydroxy-3-(1-phenylpropyl)-2H-chromen-2-one
  • Coumarin, 3-(alpha-ethylbenzyl)-4-hydroxy-
  • Falithiom
  • Falithrom
  • Fencumar
  • Liquamar
  • Marcoumar
  • Marcumar
  • Phenprocoumarol
  • Phenprocoumarole
  • Phenprocumone
  • RO 1-4849
  • 4-hydroxy-3-(1-phenylpropyl)coumarin
  • PHENYLPROPYL-4-HYDROXYCOUMARIN
  • Phenprocumon
  • 3-(α-Ethylbenzyl)-4-hydroxycoumarin
  • 4-Hydroxy-2-oxo-3-(1-phenylpropyl)-2H-chromene
  • 2-hydroxy-3-[(1S)-1-phenylpropyl]-4H-chroMen-4-one
  • 4-Hydroxy-3-(1-phenylpropyl)-2H-chromen-2-on
  • Phenprocoumon (Marcumar)
  • MARCUMA
  • inhibit,Phenprocoumon,Inhibitor
  • 4-Hydroxy-3-(1-phenyl propyl)-2H-1-Benzopyran Custom
  • 435-97-2