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Taurolithocholic Acid-d5

Product Name
Taurolithocholic Acid-d5
CAS No.
2410279-97-7
Chemical Name
Taurolithocholic Acid-d5
Synonyms
Taurolithocholic acid-d4 sodium;D4-Taurolithocholic Acid Sodium Salt;Taurolithocholic acid, sodium salt (2,2,4,4-D?, 98%);TAUROLITHOCHOLICACID,SODIUMSALT(2,2,4,4-D4) IN METHANOL;Taurolithocholic acid, sodium salt (2,2,4,4-D?, 98%) 100 μg/mL in methanol;2-[[(3α,5β)-3-hydroxy-24-oxocholan-24-yl-2,2,4,4-d4]amino]-ethanesulfonic acid, monosodium salt
CBNumber
CB18570997
Molecular Formula
C26H46NNaO5S
Formula Weight
507.71
MOL File
2410279-97-7.mol
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Taurolithocholic Acid-d5 Property

storage temp. 
-20°C
solubility 
DMF: 25 mg/ml; DMSO: 20 mg/ml; Ethanol: 1 mg/ml; PBS (pH 7.2): 1 mg/ml
form 
A crystalline solid
CAS Number Unlabeled
6042-32-6
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Safety

WGK Germany 
WGK 2
Storage Class
3 - Flammable liquids
Hazard Classifications
Acute Tox. 3 Dermal
Acute Tox. 3 Inhalation
Acute Tox. 3 Oral
Flam. Liq. 2
STOT SE 1
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H225Highly Flammable liquid and vapour

H370Causes damage to organs

Precautionary statements

P210Keep away from heat/sparks/open flames/hot surfaces. — No smoking.

P233Keep container tightly closed.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P303+P361+P353IF ON SKIN (or hair): Remove/Take off Immediately all contaminated clothing. Rinse SKIN with water/shower.

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Taurolithocholic Acid-d5 Chemical Properties,Usage,Production

Description

Taurolithocholic acid-d4 (TLCA-d4) is intended for use as an internal standard for the quantification of TLCA by GC- or LC-MS. TLCA is a taurine-conjugated form of the secondary bile acid lithocholic acid .1 TLCA (75 μM) increases caspase-3 and -7 activity in Hep3B cells transfected with sodium taurocholate cotransporting peptide (NTCP), but not nontransfected Hep3B cells.2 It has been used to induce cholestasis in ex vivo and in vivo animal models of hepatocellular cholestasis.3,4 Serum levels of TLCA increase approximately 5-fold within two hours during an oral lipid tolerance test in humans.1

Uses

Taurolithocholic acid-d4 (sodium) is the deuterium labeled Taurolithocholic acid (sodium salt). Taurolithocholic acid sodium salt, a potent cholestatic agent, is a potent Ca2+ agonist[1].

References

1. Schmid, A., Neumann, H., Karrasch, T., et al. Bile acid metabolome after an oral lipid tolerance test by liquid chromatography-tandem mass spectrometry (LC-MS/MS) PLoS One 11(2),e0148869(2016).
2. Rust, C., Wild, N., Bernt, C., et al. Bile acid-induced apoptosis in hepatocytes is caspase-6-dependent J. Biol. Chem. 284(5),2908-2916(2009).
3. Denk, G.U., Maitz, S., Wimmer, R., et al. Conjugation is essential for the anticholestatic effect of NorUrsodeoxycholic acid in taurolithocholic acid-induced cholestasis in rat liver Hepatology 52(5),1758-1768(2010).
4. Javitt, N.B. Cholestasis in rats induced by taurolithocholate Nature 210(5042),1262-1263(1966).

Taurolithocholic Acid-d5 Preparation Products And Raw materials

Raw materials

Preparation Products

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Taurolithocholic Acid-d5 Suppliers

Shanghai EFE Biological Technology Co., Ltd.
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021-65675885 18964387627
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info@efebio.com
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China
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Reer Technology (Shanghai) Co., LTD
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CHINA ISOTOPE CO., LIMITED
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Merck KGaA
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Biosynth Biological Technology (Suzhou) Co Ltd
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2410279-97-7, Taurolithocholic Acid-d5Related Search:


  • 2-[[(3α,5β)-3-hydroxy-24-oxocholan-24-yl-2,2,4,4-d4]amino]-ethanesulfonic acid, monosodium salt
  • TAUROLITHOCHOLICACID,SODIUMSALT(2,2,4,4-D4) IN METHANOL
  • Taurolithocholic acid-d4 sodium
  • D4-Taurolithocholic Acid Sodium Salt
  • Taurolithocholic acid, sodium salt (2,2,4,4-D?, 98%)
  • Taurolithocholic acid, sodium salt (2,2,4,4-D?, 98%) 100 μg/mL in methanol
  • 2410279-97-7