ChemicalBook > CAS DataBase List > Gemifioxacin mesylate

Gemifioxacin mesylate

Product Name
Gemifioxacin mesylate
CAS No.
210353-53-0
Chemical Name
Gemifioxacin mesylate
Synonyms
CS-775;LB-20304a;SB-265805S;LB-20304 Mesilate;GEMIFIOXACIN MESYLATE;(Z)-Gemifloxacin Mesilate;Gemifioxacin mesylate, 98.5%;Gemifloxacin Mesylate (300 mg);Gemifioxacin mesylate USP/EP/BP;Gemifloxacin,Inhibitor,inhibit,Gemifloxacin mesylate,Bacterial
CBNumber
CB5245303
Molecular Formula
C19H24FN5O7S
Formula Weight
485.49
MOL File
210353-53-0.mol
More
Less

Gemifioxacin mesylate Property

Melting point:
235-2370C
storage temp. 
room temp
solubility 
DMSO (Slightly), Methanol (Slightly, Heated), Water (Slightly)
form 
powder
color 
white to light brown
Stability:
Hygroscopic
CAS DataBase Reference
210353-53-0(CAS DataBase Reference)
More
Less

Safety

Safety Statements 
24/25
HS Code 
29339900
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H341Suspected of causing genetic defects

H373May cause damage to organs through prolonged or repeated exposure

Precautionary statements

P202Do not handle until all safety precautions have been read and understood.

P260Do not breathe dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P308+P313IF exposed or concerned: Get medical advice/attention.

P405Store locked up.

P501Dispose of contents/container to..…

More
Less

N-Bromosuccinimide Price

Sigma-Aldrich
Product number
SML1625
Product name
Gemifloxacin mesylate
Purity
≥98% (HPLC)
Packaging
5MG
Price
$105
Updated
2023/06/20
Sigma-Aldrich
Product number
SML1625
Product name
Gemifloxacin mesylate
Purity
≥98% (HPLC)
Packaging
25MG
Price
$424
Updated
2023/06/20
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
5mg
Price
$37
Updated
2024/03/01
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
10mg
Price
$62
Updated
2024/03/01
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
25mg
Price
$119
Updated
2024/03/01
More
Less

Gemifioxacin mesylate Chemical Properties,Usage,Production

Description

Gemifloxacin is a new fluoroquinolone derivative that is active against both Grampositive and Gram-negative bacteria, and it was launched as an oral treatment for bacterial respiratory infections. Compared with other fluoroquinolones currently on the market, gemifloxacin possesses enhanced in vitro activity against Streptococcus pneumoniae, including isolates resistant to b-lactams, macrolides, and ciprofloxacin. Gemifloxacin is specifically indicated for treating community- acquired pneumonia (CAP) caused by multi-drug resistant S. pneumoniae and for treating acute bacterial exacerbations of chronic bronchitis (AECB). The recommended dose of gemifloxacin is 320 mg daily for 5 days for AECB and 320 mg daily for 7 days for CAP.

Chemical Properties

gemifloxacin mesylate is a synthetic broad-spectrum antibacterial agent for oral administration. Gemifloxacin, a compound related to the fluoroquinolone class of antibiotics, is available as the mesylate salt in the sesquihydrate form. The mesylate salt is a white to light brown solid with a molecular weight of 485.49. Gemifloxacin is considered freely soluble at neutral pH (350 μg/mL at 37oC, pH 7.0).

Originator

LG Life Sciences (S. Korea)

Uses

Third generation fluorinated quinolone antibacterial.

Definition

ChEBI: Gemifloxacin mesylate is the mesylate salt of gemifloxacin. It has a role as an antimicrobial agent and a topoisomerase IV inhibitor. It contains a gemifloxacin.

brand name

Factive

Biochem/physiol Actions

Gemifloxacin is a broad-spectrum quinolone antibacterial. Fluoroquinolones stabilize DNA strand breaks created by DNA gyrase and topoisomerase IV by binding to the enzyme-DNA complex generating persistent, covalent enzyme–DNA adducts, inhibiting DNA synthesis. Gemifloxacin is used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. Gemifloxacin has also been found to inhibit migration and invasion of human colon cancer cells.

Gemifioxacin mesylate Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

Gemifioxacin mesylate Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky(shanghai)International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
Advantage
50
Jinan Trio PharmaTech Co., Ltd.
Tel
+86 (531) 88811783
Fax
+86 (531) 55696010 QQ 1762738062
Email
sales@trio-pharmatech.com (International market)
Country
China
ProdList
1856
Advantage
62
Shanghai Ennopharm Co., Ltd.
Tel
+86 (21) 6435-5022
Country
China
ProdList
4267
Advantage
65
BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
ProdList
14055
Advantage
65
Dalian Meilun Biotech Co., Ltd.
Tel
0411-62910999 13889544652
Email
meilunui@163.com
Country
China
ProdList
4727
Advantage
58
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Shanghai T&W Pharmaceutical Co., Ltd.
Tel
+86 21 61551611
Fax
+86 21 50676805
Country
China
ProdList
9891
Advantage
58
Haoyuan Chemexpress Co., Ltd.
Tel
021-58950125
Fax
(86) 21-58955996
Email
info@chemexpress.com
Country
China
ProdList
7552
Advantage
61
More
Less

View Lastest Price from Gemifioxacin mesylate manufacturers

Hebei Weibang Biotechnology Co., Ltd
Product
Gemifioxacin mesylate 210353-53-0
Price
US $10.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
10 mt
Release date
2021-11-01
Hebei Mojin Biotechnology Co., Ltd
Product
Gemifioxacin mesylate 210353-53-0
Price
US $0.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
50000KG/month
Release date
2023-08-18
Dideu Industries Group Limited
Product
Gemifioxacin mesylate 210353-53-0
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-07-19

210353-53-0, Gemifioxacin mesylateRelated Search:


  • GEMIFIOXACIN MESYLATE
  • 7-(3-aminomethyl)-4-methoxyimino-pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid mesylate
  • LB-20304 Mesilate
  • Gemifioxacin mesylate, 98.5%
  • CS-775
  • (Z)-Gemifloxacin Mesilate
  • LB-20304a
  • SB-265805S
  • Gemifioxacin mesylate USP/EP/BP
  • (Z)-7-(3-(Aminomethyl)-4-(methoxyimino)pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid methanesulfonic acid salt
  • Gemifloxacin,Inhibitor,inhibit,Gemifloxacin mesylate,Bacterial
  • Gemifloxacin Mesylate (300 mg)
  • 210353-53-0
  • C18H20FN5O4CH4SO3
  • C19H24FN5O7S
  • Intermediates & Fine Chemicals
  • Pharmaceuticals