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Gemifioxacin mesylate

Product Name
Gemifioxacin mesylate
CAS No.
210353-53-0
Chemical Name
Gemifioxacin mesylate
Synonyms
CS-775;LB-20304a;SB-265805S;LB-20304 Mesilate;GEMIFIOXACIN MESYLATE;(Z)-Gemifloxacin Mesilate;Gemifioxacin mesylate, 98.5%;Gemifloxacin Mesylate (300 mg);Gemifioxacin mesylate USP/EP/BP;Gemifloxacin,Inhibitor,inhibit,Gemifloxacin mesylate,Bacterial
CBNumber
CB5245303
Molecular Formula
C19H24FN5O7S
Formula Weight
485.49
MOL File
210353-53-0.mol
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Gemifioxacin mesylate Property

Melting point:
235-2370C
storage temp. 
room temp
solubility 
DMSO (Slightly), Methanol (Slightly, Heated), Water (Slightly)
form 
powder
color 
white to light brown
Stability:
Hygroscopic
CAS DataBase Reference
210353-53-0(CAS DataBase Reference)
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Safety

Safety Statements 
24/25
HS Code 
29339900
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H341Suspected of causing genetic defects

H373May cause damage to organs through prolonged or repeated exposure

Precautionary statements

P202Do not handle until all safety precautions have been read and understood.

P260Do not breathe dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P308+P313IF exposed or concerned: Get medical advice/attention.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
SML1625
Product name
Gemifloxacin mesylate
Purity
≥98% (HPLC)
Packaging
5MG
Price
$105
Updated
2023/06/20
Sigma-Aldrich
Product number
SML1625
Product name
Gemifloxacin mesylate
Purity
≥98% (HPLC)
Packaging
25MG
Price
$424
Updated
2023/06/20
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
5mg
Price
$37
Updated
2024/03/01
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
10mg
Price
$62
Updated
2024/03/01
Cayman Chemical
Product number
21047
Product name
Gemifloxacin (mesylate)
Purity
≥98%
Packaging
25mg
Price
$119
Updated
2024/03/01
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Gemifioxacin mesylate Chemical Properties,Usage,Production

Description

Gemifloxacin is a new fluoroquinolone derivative that is active against both Grampositive and Gram-negative bacteria, and it was launched as an oral treatment for bacterial respiratory infections. Compared with other fluoroquinolones currently on the market, gemifloxacin possesses enhanced in vitro activity against Streptococcus pneumoniae, including isolates resistant to b-lactams, macrolides, and ciprofloxacin. Gemifloxacin is specifically indicated for treating community- acquired pneumonia (CAP) caused by multi-drug resistant S. pneumoniae and for treating acute bacterial exacerbations of chronic bronchitis (AECB). The recommended dose of gemifloxacin is 320 mg daily for 5 days for AECB and 320 mg daily for 7 days for CAP.

Chemical Properties

gemifloxacin mesylate is a synthetic broad-spectrum antibacterial agent for oral administration. Gemifloxacin, a compound related to the fluoroquinolone class of antibiotics, is available as the mesylate salt in the sesquihydrate form. The mesylate salt is a white to light brown solid with a molecular weight of 485.49. Gemifloxacin is considered freely soluble at neutral pH (350 μg/mL at 37oC, pH 7.0).

Originator

LG Life Sciences (S. Korea)

Uses

Third generation fluorinated quinolone antibacterial.

Definition

ChEBI: Gemifloxacin mesylate is the mesylate salt of gemifloxacin. It has a role as an antimicrobial agent and a topoisomerase IV inhibitor. It contains a gemifloxacin.

brand name

Factive

Biochem/physiol Actions

Gemifloxacin is a broad-spectrum quinolone antibacterial. Fluoroquinolones stabilize DNA strand breaks created by DNA gyrase and topoisomerase IV by binding to the enzyme-DNA complex generating persistent, covalent enzyme–DNA adducts, inhibiting DNA synthesis. Gemifloxacin is used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. Gemifloxacin has also been found to inhibit migration and invasion of human colon cancer cells.

Gemifioxacin mesylate Preparation Products And Raw materials

Raw materials

Preparation Products

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Gemifioxacin mesylate Suppliers

Novachem Aromatici S.R.L.
Tel
--
Fax
--
Email
umberto.grigoli@novachemaromatici.com
Country
Italy
ProdList
193
Advantage
58
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View Lastest Price from Gemifioxacin mesylate manufacturers

Hebei Weibang Biotechnology Co., Ltd
Product
Gemifioxacin mesylate 210353-53-0
Price
US $10.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
10 mt
Release date
2021-11-01
Hebei Mojin Biotechnology Co., Ltd
Product
Gemifioxacin mesylate 210353-53-0
Price
US $0.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
50000KG/month
Release date
2023-08-18
Dideu Industries Group Limited
Product
Gemifioxacin mesylate 210353-53-0
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-07-19

210353-53-0, Gemifioxacin mesylateRelated Search:


  • GEMIFIOXACIN MESYLATE
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  • SB-265805S
  • Gemifioxacin mesylate USP/EP/BP
  • (Z)-7-(3-(Aminomethyl)-4-(methoxyimino)pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid methanesulfonic acid salt
  • Gemifloxacin,Inhibitor,inhibit,Gemifloxacin mesylate,Bacterial
  • Gemifloxacin Mesylate (300 mg)
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