ChemicalBook > CAS DataBase List > Triprolidine hydrochloride

Triprolidine hydrochloride

Product Name
Triprolidine hydrochloride
CAS No.
6138-79-0
Chemical Name
Triprolidine hydrochloride
Synonyms
rate,stereoisomer;TRIPROLIDINE HCL USP;trans-TriprolidineHCl;Tripolidine Hydrochloride;Triprolidine hydrochloride;Triprolidine Hydrochlorise;TRIPROLIDINE HCL MONOHYDRATE;TRIPROLIDINEHYDROCHLORIDE,USP;Triprolidine hydrochloride (347);triprolidinesigmareferencestandard
CBNumber
CB6232533
Molecular Formula
C19H23ClN2
Formula Weight
314.85
MOL File
6138-79-0.mol
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Triprolidine hydrochloride Property

Melting point:
115-120°C
storage temp. 
2-8°C
solubility 
alcohol: soluble1 in 1.5 of solvent
form 
Solid
color 
White to Off-White
Water Solubility 
>=10 g/100 mL at 20 ºC
Merck 
13,9817
Stability:
Stable, but discolours in light. Incompatible with strong oxidizing agents.
LogP
4.223 (est)
CAS DataBase Reference
6138-79-0(CAS DataBase Reference)
EPA Substance Registry System
Pyridine, 2-[1-(4-methylphenyl)-3-(1-pyrrolidinyl)-1-propenyl]-, monohydrochloride, monohydrate, (E)- (6138-79-0)
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Safety

Hazard Codes 
Xn
Risk Statements 
22-36/37/38
Safety Statements 
26-36
WGK Germany 
3
RTECS 
UT7658000
HS Code 
2933399090
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
T6764
Product name
Triprolidine hydrochloride
Purity
≥99%
Packaging
1g
Price
$45.5
Updated
2024/03/01
Sigma-Aldrich
Product number
PHR2662
Product name
Triprolidine
Purity
PharmaceuticalSecondaryStandard;CertifiedReferenceMaterial
Packaging
500MG
Price
$200
Updated
2024/03/01
Sigma-Aldrich
Product number
1696007
Product name
Triprolidine hydrochloride
Purity
United States Pharmacopeia (USP) Reference Standard
Packaging
300mg
Price
$436
Updated
2024/03/01
Sigma-Aldrich
Product number
BP347
Product name
Triprolidine hydrochloride
Purity
British Pharmacopoeia (BP) Reference Standard
Packaging
100MG
Price
$263
Updated
2023/01/07
Sigma-Aldrich
Product number
T-140
Product name
Triprolidine hydrochloride solution
Purity
1?mg/mL in methanol ((as free base)), certified reference material, ampule of 1?mL, Cerilliant?
Packaging
1ML
Price
$88.7
Updated
2022/05/15
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Triprolidine hydrochloride Chemical Properties,Usage,Production

Chemical Properties

TRIPROLIDINE HYDROCHLORIDE is a white, crystalline powder.

Uses

anticholinergic (opthalmic)

Uses

trans-Triprolidine Hydrochloride is a potent H1 receptor antagonist. Anti-histamines.

Uses

TRIPROLIDINE HYDROCHLORIDE is used as bulk pharmaceutical (antihistaminic). Product Data Sheet

Definition

TRIPROLIDINE HYDROCHLORIDE is a hydrate that is the monohydrate form of triprolidine hydrochloride. A sedating antihistamine, it is used for the symptomatic relief of uticaria, rhinitis, and various pruritic skin disorders.

brand name

Actidil (GlaxoSmithKline); Myidyl (USl).

General Description

Triprolidine hydrochloride,(E)-2-[3-(1-pyrrolidinyl)-1-p-tolylpropenyl]pyridine monohydrochloridemonohydrate (Actidil), is a white crystalline powder with a slight, but unpleasant, odor. It is soluble inwater and in alcohol, and its solutions are alkaline to litmus.
The antihistaminic activity is confined mainly to the geometricisomer in which the pyrrolidinomethyl group is transto the 2-pyridyl group. Pharmacological studies confirm thehigh activity of triprolidine and the superiority of (E) overcorresponding (Z) isomers as H1-antihistamines. At guineapig ileum sites, the affinity of triprolidine for H-receptorswas more than 1,000 times the affinity of its (Z) diasteromer.The relative potency of triprolidine is of the same orderas that of dexchlorpheniramine. The peak effect occursabout 3.5 hours after oral administration, and the duration ofeffect is about 12 hours.

General Description

Odorless white crystalline powder. Bitter taste.

Air & Water Reactions

Water soluble.

Reactivity Profile

Triprolidine hydrochloride discolors on exposure to light.

Health Hazard

SYMPTOMS: Symptoms of exposure to Triprolidine hydrochloride may include depression to stimulation of the central nervous system, dry mouth, fixed dilated pupils, flushing, hallucinations, convulsions, urinary retention, cardiac arrhythmias and coma. Other symptoms may include excitability, drowsiness, nervousness, dizziness, high fever and sleeplessness. It can also cause sedation. It may also cause local anesthesia, dryness of the throat and nose and abdominal pain with vomiting or diarrhea.

Fire Hazard

Flash point data for Triprolidine hydrochloride are not available; however, Triprolidine hydrochloride is probably combustible.

Biological Activity

Potent H 1 receptor antagonist.

Triprolidine hydrochloride Preparation Products And Raw materials

Raw materials

Preparation Products

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Triprolidine hydrochloride Suppliers

Hubei wei shi reagent group ltd., company
Tel
027-59105166 13125137732
Email
2853863890@qq.com
Country
China
ProdList
2981
Advantage
58
Wuhan Dingxintong Pharmaceutical Co. , Ltd.
Tel
027-027-52344656 15871722230
Fax
2796190295
Email
15871722230@163.com
Country
China
ProdList
4854
Advantage
58
3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15839
Advantage
69
XiaoGan ShenYuan ChemPharm co,ltd
Tel
15527768850
Email
1791901229@qq.com
Country
China
ProdList
8843
Advantage
52
China Langchem Inc.
Tel
0086-21-58956006
Fax
0086-21-58956100
Country
China
ProdList
7811
Advantage
57
Sinopharm Chemical Reagent Co,Ltd.
Tel
86-21-63210123
Fax
86-21-63290778 86-21-63218885
Email
sj_scrc@sinopharm.com
Country
China
ProdList
9815
Advantage
79
Hangzhou Yuhao Chemical Technology Co., Ltd
Tel
0571-82693216
Fax
+86-571-82880190
Email
info@yuhaochemical.com
Country
China
ProdList
9387
Advantage
52
Spectrum Chemical Manufacturing Corp.
Tel
021-021-021-67601398-809-809-809 15221380277
Fax
021-57711696
Email
marketing_china@spectrumchemical.com
Country
China
ProdList
9658
Advantage
60
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Shanghai T&W Pharmaceutical Co., Ltd.
Tel
+86 21 61551611
Fax
+86 21 50676805
Country
China
ProdList
9891
Advantage
58
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View Lastest Price from Triprolidine hydrochloride manufacturers

WUHAN FORTUNA CHEMICAL CO., LTD
Product
Triprolidine hydrochloride 6138-79-0
Price
US $0.00-0.00/Kg/Drum
Min. Order
1KG
Purity
98%-101%
Supply Ability
100KG
Release date
2021-05-28
Zhuhai Hairuide Bioscience and Technology Co., Ltd
Product
Triprolidine hydrochloride 6138-79-0
Price
US $0.00/KG Ton
Min. Order
1KG Ton
Purity
USP4398%+
Supply Ability
2 tons/month
Release date
2022-10-09
Zhuozhou Wenxi import and Export Co., Ltd
Product
Triprolidine hydrochloride 6138-79-0
Price
US $15.00-10.00/KG
Min. Order
1KG
Purity
99%+ HPLC
Supply Ability
Monthly supply of 1 ton
Release date
2021-07-09

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