ChemicalBook > CAS DataBase List > BQ-788

BQ-788

Product Name
BQ-788
CAS No.
156161-89-6
Chemical Name
BQ-788
Synonyms
CS-1494;BQ-788 SODIUM;BQ789 Sodium Salt;1-ELAIDYLPHOSPHOCHOLINE, >97%;BQ788 SODIUM SALT; BQ 788 SODIUM SALT;BQ 788 sodium salt, ETB receptor antagonist;BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-;N-cis-2,6-dimethylpiperidinocarbonyl-L-γMeLeu-D-Trp(COOMe)-D-Nle-ONa;2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
CBNumber
CB7710904
Molecular Formula
C34H52N5NaO7
Formula Weight
665.81
MOL File
156161-89-6.mol
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BQ-788 Property

storage temp. 
-20°C
solubility 
acetonitrile: 0.3 mg/mL
form 
solid
color 
white
Water Solubility 
acetonitrile: 0.3mg/mL
DMSO: 1.2mg/mL
ethanol: 1.2mg/mL
H2O: slightly soluble
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Safety

WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
B157
Product name
BQ-788
Purity
≥95%,solid
Packaging
200μg
Price
$231
Updated
2024/03/01
Cayman Chemical
Product number
17403
Product name
BQ-788 (sodium salt)
Purity
≥95%
Packaging
500μg
Price
$175
Updated
2024/03/01
Cayman Chemical
Product number
17403
Product name
BQ-788 (sodium salt)
Purity
≥95%
Packaging
1mg
Price
$242
Updated
2024/03/01
TRC
Product number
B676670
Product name
BQ788
Packaging
5mg
Price
$595
Updated
2021/12/16
ChemScene
Product number
CS-2685
Product name
BQ-788(sodiumsalt)
Purity
98.03%
Packaging
10mg
Price
$600
Updated
2021/12/16
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BQ-788 Chemical Properties,Usage,Production

Uses

BQ-788 has been used as a selective endothelin-B (ETRB) blocker in human airway smooth muscle cells (HASMCs), uterine mesothelial cells (UtMCs)-derived vascular smooth muscle cells (VSMCs), and human umbilical vein endothelial cells (HUVECs)

Biological Activity

Potent, selective ET B receptor antagonist (IC 50 = 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells).

Biochem/physiol Actions

Selective ETB endothelin receptor antagonist.

storage

+4°C

BQ-788 Preparation Products And Raw materials

Raw materials

Preparation Products

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BQ-788 Suppliers

Tocris Bioscience
Tel
--
Fax
--
Email
customerservice@tocris.co.uk
Country
United Kingdom
ProdList
5726
Advantage
77
MOLEKULA Ltd.
Tel
--
Fax
--
Email
kevinbanks@molekula.com
Country
United Kingdom
ProdList
6140
Advantage
66
Fluorochem Ltd
Tel
--
Fax
--
Email
vernam@fluorochem.co.uk
Country
United Kingdom
ProdList
6375
Advantage
65

156161-89-6, BQ-788Related Search:


  • BQ-788 SODIUM
  • BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT
  • N-[(cis-2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucinesodiumsalt
  • 1-ELAIDYLPHOSPHOCHOLINE, >97%
  • N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt, 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
  • N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-
  • DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl)
  • 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
  • N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt
  • BQ789 Sodium Salt
  • N-cis-2,6-dimethylpiperidinocarbonyl-L-γMeLeu-D-Trp(COOMe)-D-Nle-ONa
  • BQ788 SODIUM SALT; BQ 788 SODIUM SALT
  • CS-1494
  • sodium,(2R)-2-[[(2R)-2-amino-3-(1-methoxycarbonylindol-3-yl)propanoyl]-[(2S)-2-[[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]amino]-4,4-dimethylpentanoyl]amino]hexanoate
  • D-Norleucine, N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-, sodium salt (1:1)
  • Sodium (R)-2-((R)-2-((S)-2-((2R,6S)-2,6-dimethylpiperidine-1-carboxamido)-4,4-dimethylpentanamido)-3-(1-(methoxycarbonyl)-1H-indol-3-yl)propanamido)hexanoate
  • BQ 788 sodium salt, ETB receptor antagonist
  • 156161-89-6
  • C34H51N5NaO7
  • C34H50N5O7Na
  • C34H50N5NaO7
  • Endothelin receptor