Basic information Safety Supplier Related

Cyclosporin C

Basic information Safety Supplier Related

Cyclosporin C Basic information

Product Name:
Cyclosporin C
Synonyms:
  • CYCLOSPORIN C
  • Cyclosporine C/Cyclo[L-alanyl-D-alanyl-N-methyl-L-leucyl-N-methyl-L-leucyl-N-methyl-L-valyl-3-hydroxy-N,4-dimethyl-L-2-amino-6-octenoyl-L-threonyl-N-methylglycyl-N-methyl-L-leucyl-L-valyl-N-methyl-L-leucyl]
  • 30-(1-hydroxyethyl)-33-(1-hydroxy-2-methylhex-4-enyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriaconta
  • CS-2545
  • CS-2546
  • cyclo-[MeBmt-Thr-Sar-MeLeu-Val-MeLeu-Ala-D-Ala-MeLeu-MeLeu-MeVal]
  • Cyclosporine EP Impurity C
  • Thr2-cyclosporine
CAS:
59787-61-0
MF:
C62H111N11O13
MW:
1218.61
Product Categories:
  • Intermediates & Fine Chemicals
  • Peptides
  • ACTIVE PHARMACEUTICAL INGREDIENTS
  • Pharmaceuticals
Mol File:
59787-61-0.mol
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Cyclosporin C Chemical Properties

Melting point:
144-1460C
alpha 
D20 -255° (c = 0.5 in chloroform); D20 -182° (c = 0.5 in methanol)
Boiling point:
1316.0±65.0 °C(Predicted)
Density 
1.033±0.06 g/cm3(Predicted)
storage temp. 
Sealed in dry,Store in freezer, under -20°C
solubility 
DMSO: ≥10mg/mL
pka
13.06±0.70(Predicted)
form 
Colorless to off-white crystalline solid.
color 
White to Off-White
InChIKey
JTOKYIBTLUQVQV-PCACHRFWSA-N
CAS DataBase Reference
59787-61-0
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Safety Information

WGK Germany 
3
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Cyclosporin C Usage And Synthesis

Description

Cyclosporin C is a fungal metabolite that has been found in T. inflatum and has diverse biological activities, including antifungal, antiviral, and immunosuppressant properties. It is active against isolates of B. cinerea, A. niger, and Alternaria, Mucor, and Penicillium species (MICs = 0.1-5 μg/ml). Cyclosporin C (15 μg/ml) inhibits vaccinia virus replication in infected BSC40 cells by 98.82%. It inhibits lymphocyte proliferation induced by the mitogens concanavalin A (ConA; ), phytohemagglutinin L (PHA), and pokeweed mitogen (PWM), as well as proliferation induced by alloantigen in mixed lymphocyte culture when used at a concentration of 100 ng/ml. Cyclosporin C (100 ng/ml) inhibits the local graft versus host (GVH) reaction in mice receiving splenocyte grafts.

Chemical Properties

White Solid

Uses

A group of nonpolar cyclic oligopeptides with immunosupppressant activity.

Uses

Cyclosporin C is a minor analogue of the cyclosporin complex produced by a number of fungal species, including Trichoderma, Tolypocladium, Fusarium, Nectria and Acremonium. Cyclosporin C possesses immunosuppressant activity but has been much less extensively investigated than the major analogue, cyclosporin A.

storage

+4°C

Cyclosporin C Preparation Products And Raw materials

Preparation Products

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