Endoxifen Chemical Properties

Melting point:

127-129°C

Boiling point:

519.3±50.0 °C(Predicted)

Density 

1.099±0.06 g/cm3(Predicted)

storage temp. 

Amber Vial, -86°C Freezer, Under Inert Atmosphere

solubility 

DMSO : 50 mg/mL (133.87 mM; Need ultrasonic)H2O : < 0.1 mg/mL (insoluble)

form 

Powder

pka

10.36±0.15(Predicted)

color 

White to off-white

Stability:

Light Sensitive, Temperature Sensitive

Endoxifen Usage And Synthesis

Chemical Properties

Off-White to Pink Solid

Uses

A novel active metabolite of the anti-cancer drug Tamoxifen. It showed potent ER binding property, blocked estrogen stimulated growth of breast cancer cell and half maximal inhibition of estrogen responsive gene expression in ER pos. human breast ca

Uses

A novel active metabolite of the anti-cancer drug Tamoxifen (T006000). It showed potent ER binding property, blocked estrogen stimulated growth of breast cancer cell and half maximal inhibition of estrogen responsive gene expression in ER pos. human breast cancer cell line.

Definition

ChEBI: 4-Hydroxy-N-desmethyltamoxifen is a stilbenoid.

Endoxifen(112093-28-4)Related Product Information

• Endoxifen HCl
• Tamoxifen Impurity 3
• 4-Benzyloxy β-Hydroxy TaMoxifen
• TaMoxifen DiMer
• 1-(4-(2-Dimethylamino)-2-ethoxyphenyl butanone
• N-Desmethyl-4-hydroxy Tamoxifen β-D-Glucuronide (E/Z Mixture)
• 4Hydroxy Tamoxifen
• Tamoxifen EP Impurity D
• (E)-4-Alloxycarboxyl Tamoxifen
• desdimethyltamoxifen
• TAMOXIFEN-N-OXIDE
• Droloxifene
• (E)-4-Acetoxy Tamoxifen
• N-Desmethyl Tamoxifen Methanethiosulfonate
• 2-[4-[(E)-1,2-diphenylbut-1-enyl]phenoxy]-N,N-dimethyl-ethanamine
• alpha-[4-[2-(dimethylamino)ethoxy]phenyl]-beta-ethyl-alpha-phenylphenethyl alcohol
• (E)-4-Hydroxy-N-desmethyl Tamoxifen
• 4-HYDROXYTAMOXIFEN