4-Fluoro-2-methoxyphenylboronic acid Chemical Properties

Melting point:

131-136 °C (lit.)

Boiling point:

294.8±50.0 °C(Predicted)

Density 

1.26±0.1 g/cm3(Predicted)

storage temp. 

Inert atmosphere,Room Temperature

pka

8.69±0.58(Predicted)

form 

Crystalline Powder

color 

White

CAS DataBase Reference

179899-07-1(CAS DataBase Reference)

Safety Information

Hazard Codes 

Xi

Risk Statements 

36/37/38

Safety Statements 

26-36/37/39-36-60-37

WGK Germany 

3

HazardClass 

IRRITANT

HS Code 

29319090

MSDS

• Language:English Provider:SigmaAldrich

4-Fluoro-2-methoxyphenylboronic acid Usage And Synthesis

Uses

suzuki reaction

Uses

Reactant involved in:
Suzuki-Miyaura cross-coupling reactions for synthesis of heterobiaryls
Suzuki and Still coupling for synthesis of antithrombotic drugs
Reactant / precursor used for the synthesis of biologically active molecules including:
2-(4-pyridyl)thienopyridinones for use as GSK-3β inhibitors
Arylheteroarylmethylamines as NR2B subtype of NMDA receptor antagonists with antidepressant activity
Biphenylketones for use as dual modulators of inflammation and bone loss
CB1 antagonists

4-Fluoro-2-methoxyphenylboronic acid(179899-07-1)Related Product Information

• 4-Methoxybenzyl alcohol
• 4-Fluorobenzeneboronic acid
• 4-Methoxybenzoyl chloride
• (4-METHOXYPHENYL)-BORANE
• 3-Methoxyacetophenone
• p-Anisaldehyde
• 4-Methoxybenzyl cyanide
• Anisole
• 2,3,4-Trimethoxybenzaldehyde
• (Trifluoromethoxy)benzene
• 4-Methoxyphenylboronic acid
• Phenylboronic acid
• 2-ETHOXY-4-FLUOROPHENYLBORONIC ACID
• 4-FLUORO-2-PROPOXYPHENYLBORONIC ACID
• 4-FLUORO-2-ISOPROPOXYPHENYLBORONIC ACID
• 4,5-DIFLUORO-2-METHOXYPHENYLBORONIC ACID
• 2-BUTOXY-4-FLUOROPHENYLBORONIC ACID
• Fluorine