ChemicalBook > CAS DataBase List > AMASTATIN HYDROCHLORIDE

AMASTATIN HYDROCHLORIDE

Product Name
AMASTATIN HYDROCHLORIDE
CAS No.
100938-10-1
Chemical Name
AMASTATIN HYDROCHLORIDE
Synonyms
AMASTATIN;AMASTATIN HCL;AMASTATIN HYDROCHLORIDE;AMASTATIN HYDROCHLORIDE HYDRATE;H-(2S,3R)-AHMH-VAL-VAL-ASP-OH HCL;Amastatin hydrate hydrochloride;4-formylphenyl-O-β-d-allopyranoside;N((2S 3R)3-AMINO-2-HXY-5-ME.HEXANOYL)-L&;Amastatinhydrochloridebiochemikasynthetic;(2S,3R)-[3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-VAL-VAL-ASP-OH HCL
CBNumber
CB0194817
Molecular Formula
C21H39ClN4O8
Formula Weight
511.01
MOL File
100938-10-1.mol
More
Less

AMASTATIN HYDROCHLORIDE Property

Melting point:
202-205 °C
storage temp. 
-20°C
solubility 
methanol: 5 mg/mL, clear, colorless
form 
White to off-white powder.
color 
White to off-white
BRN 
8888370
More
Less

Safety

WGK Germany 
3
10
HS Code 
2924190090
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

More
Less

N-Bromosuccinimide Price

Sigma-Aldrich
Product number
A1276
Product name
Amastatin hydrochloride hydrate
Purity
≥97% (HPLC)
Packaging
0.5mg
Price
$177
Updated
2024/03/01
Sigma-Aldrich
Product number
A1276
Product name
Amastatin hydrochloride hydrate
Purity
≥97% (HPLC)
Packaging
1mg
Price
$282
Updated
2024/03/01
Cayman Chemical
Product number
16719
Product name
Amastatin (hydrochloride)
Purity
≥95%
Packaging
500μg
Price
$33
Updated
2024/03/01
Cayman Chemical
Product number
16719
Product name
Amastatin (hydrochloride)
Purity
≥95%
Packaging
1mg
Price
$60
Updated
2024/03/01
Sigma-Aldrich
Product number
A1276
Product name
Amastatin hydrochloride hydrate
Purity
≥97% (HPLC)
Packaging
5mg
Price
$1010
Updated
2024/03/01
More
Less

AMASTATIN HYDROCHLORIDE Chemical Properties,Usage,Production

Uses

Amastatin is a slow, tight binding, competitive aminopeptidase (AP) inhibitor, first described as an inhibitor of human serum AP-A (glutamyl AP; IC50 = 0.54 μg/ml) but not of AP-B (arginine AP). It also inhibits AP-N (AP-M, alanyl AP; Ki = 20-200 nM), leucyl-cystinyl AP (Ki = 20-220 nM), and endoplasmic reticulum AP 1 (Ki = 41.8 μM). Amastatin is without effect on trypsin, papain, chymotrypsin, elastase, pepsin, or thermolysin.[Cayman Chemical]

General Description

Chemical structure: peptide

Biochem/physiol Actions

It inhibits cytosolic leucine aminopeptidase (EC.3.4.11.1), microsomal aminopeptidase M (EC.3.4.11.2) and bacterial leucine aminopeptidase (EC.3.4.11.10). It is less effective against aminopeptidase A (EC 3.4.11.7), the enzyme that converts angiotensin II to angiotensin III. Potentiates the CNS effects of vasopressin and oxytocin in vivo.Effective concentration: 1-10 μM.

storage

+4°C

AMASTATIN HYDROCHLORIDE Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

AMASTATIN HYDROCHLORIDE Suppliers

Alabiotech Inc.
Tel
001-619-354-5251
Fax
001-855-855-6087
Email
sales@alabiotech-e.com
Country
United States
ProdList
972
Advantage
60
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32165
Advantage
58
Alfa Chemistry
Tel
Fax
1-516-927-0118
Email
Info@alfa-chemistry.com
Country
United States
ProdList
24072
Advantage
58
Aladdin Scientific
Tel
+1-+1(833)-552-7181
Email
sales@aladdinsci.com
Country
United States
ProdList
52925
Advantage
58
Cayman Chemical Company
Tel
--
Fax
--
Email
cayman@caymanchem.com
Country
United States
ProdList
6213
Advantage
81
MedChemExpress
Tel
--
Fax
--
Email
sales@medchemexpress.com
Country
United States
ProdList
6398
Advantage
58
Combi-Blocks Inc.
Tel
--
Fax
--
Email
sales@combi-blocks.com
Country
United States
ProdList
6618
Advantage
69
Riedel-de Haen AG
Tel
--
Fax
--
Country
United States
ProdList
6773
Advantage
87
Interchim Inc.
Tel
--
Fax
--
Email
web@interchiminc.com
Country
United States
ProdList
301
Advantage
50
Santa Cruz Biotechnology, Inc.
Tel
--
Fax
--
Email
scbt@scbt.com
Country
United States
ProdList
3597
Advantage
60
LKT Laboratories, Inc.
Tel
--
Fax
--
Email
info@lktlabs.com
Country
United States
ProdList
2164
Advantage
64
2A PharmaChem USA
Tel
--
Fax
--
Email
sales@2apharmachem.com
Country
United States
ProdList
6137
Advantage
39
3B Scientific Corporation
Tel
--
Fax
--
Email
sales@3bsc.com
Country
United States
ProdList
6718
Advantage
47
MP Biomedicals, Inc.
Tel
--
Fax
--
Country
United States
ProdList
6561
Advantage
81
More
Less

View Lastest Price from AMASTATIN HYDROCHLORIDE manufacturers

Career Henan Chemical Co
Product
AMASTATIN HYDROCHLORIDE 100938-10-1
Price
US $1.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
g/kg/Ton
Release date
2020-03-05

100938-10-1, AMASTATIN HYDROCHLORIDERelated Search:


  • [(2S,3R)-3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-VAL-VAL-ASP HYDROCHLORIDE
  • (2S,3R)-[3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-VAL-VAL-ASP-OH HCL
  • AMASTATIN
  • AMASTATIN HCL
  • AMASTATIN HYDROCHLORIDE
  • AMASTATIN HYDROCHLORIDE HYDRATE
  • H-(2S,3R)-AHMH-VAL-VAL-ASP-OH HCL
  • N((2S 3R)3-AMINO-2-HXY-5-ME.HEXANOYL)-L&
  • Amastatinhydrochloridebiochemikasynthetic
  • (2s,3r)-3-amino-2-hydroxy-5-methylhexanoyl-val-val-asp hydrochloride hydrate
  • (Amino-2-hydroxy-5-methyl-hexanoyl)-L-valyl-L-valyl-L-aspartic acid hydrochloride salt
  • (2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl-Val-Val-Asp hydrate hydrochloride
  • Amastatin hydrate hydrochloride
  • L-Aspartic acid,N-[(2S,3R)-3-amino-2-hydroxy-5-methyl-1-oxohexyl]-L-valyl-L-valyl-,monohydrochloride (9CI)
  • 4-formylphenyl-O-β-d-allopyranoside
  • 100938-10-1
  • C21H38N4O8HCl
  • C21H38N4O8HClxH2O
  • C21H38N4O8ClH
  • BioChemical
  • Antibiotics
  • Antibiotics A to Z
  • Antibiotics A-F
  • peptides
  • inhibitor
  • Pepetides