2-Morpholinopyrimidin-5-ylboronic acid
- Product Name
- 2-Morpholinopyrimidin-5-ylboronic acid
- CAS No.
- 870521-33-8
- Chemical Name
- 2-Morpholinopyrimidin-5-ylboronic acid
- Synonyms
- 2-Morpholinopyrimidine-5-boronic acid;2-morpholino-5-pyrimidineboronic acid;2-morpholinopyrimidin-5-ylboronic acid;(2-(Morpholin-4-yl)pyrimidin-5-yl)boronic;2-Morpholinopyrimidin-5-ylboronic acid 95%;2-(Morpholine-4-yl)pyrimidine-5-boronic acid;[2-(4-Morpholinyl)-5-pyrimidinyl]boronic acid;Boronic acid,B-[2-(4-morpholinyl)-5-pyrimidinyl]-;2-Morpholinopyrimidine-5-boronic acid(contains varying amounts of Anhydride)
- CBNumber
- CB11502708
- Molecular Formula
- C8H12BN3O3
- Formula Weight
- 209.01
- MOL File
- 870521-33-8.mol
2-Morpholinopyrimidin-5-ylboronic acid Property
- Boiling point:
- 484.0±55.0 °C(Predicted)
- Density
- 1.37
- storage temp.
- Inert atmosphere,2-8°C
- pka
- 3.02±0.19(Predicted)
- form
- solid
- Appearance
- White to yellow Solid
Safety
- HS Code
- 2934999090
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
H315Causes skin irritation
H319Causes serious eye irritation
H332Harmful if inhaled
H335May cause respiratory irritation
- Precautionary statements
-
P261Avoid breathing dust/fume/gas/mist/vapours/spray.
P280Wear protective gloves/protective clothing/eye protection/face protection.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
N-Bromosuccinimide Price
- Product number
- M733128
- Product name
- 2-Morpholinopyrimidin-5-ylboronicAcid
- Packaging
- 5g
- Price
- $60
- Updated
- 2021/12/16
- Product number
- X1399
- Product name
- 2-(Morpholine-4-yl)pyrimidine-5-boronicacid
- Packaging
- 250mg
- Price
- $105
- Updated
- 2021/12/16
- Product number
- 093052
- Product name
- 2-Morpholinopyrimidin-5-ylboronic acid
- Purity
- 95+%
- Packaging
- 250mg
- Price
- $182
- Updated
- 2021/12/16
- Product number
- BOR0005496
- Product name
- 2-MORPHOLINOPYRIMIDIN-5-YL BORONIC ACID
- Purity
- 95.00%
- Packaging
- 1G
- Price
- $401.1
- Updated
- 2021/12/16
- Product number
- 093052
- Product name
- 2-Morpholinopyrimidin-5-ylboronic acid
- Purity
- 95+%
- Packaging
- 1g
- Price
- $404
- Updated
- 2021/12/16
2-Morpholinopyrimidin-5-ylboronic acid Chemical Properties,Usage,Production
Synthesis
110-91-8
1003845-06-4
870521-33-8
The reaction was carried out with 2-chloropyrimidin-5-ylboronic acid (1 g, 6.32 mmol), morpholine (2.19 mL, 25.26 mmol) and triethylamine (0.88 mL, 6.32 mmol) in ethanol (25 mL) with stirring for 1 hour at 20 °C. After completion of the reaction, water (50 mL) was slowly added to the reaction mixture. The resulting precipitate was collected by filtration and washed with water to finally obtain 2-morpholinopyrimidin-5-ylboronic acid (950 mg, 70% yield) as a milky white solid. The NMR hydrogen spectrum (250 MHz, DMSO-d6) data were as follows: δ 8.63 (s, 2H), 8.05 (s, 2H), 3.68 (ddd, J=23.4,5.7,3.9Hz, 8H).
References
[1] Patent: WO2015/86506, 2015, A1. Location in patent: Page/Page column 131
[2] Patent: WO2015/86512, 2015, A1. Location in patent: Page/Page column 102
[3] Patent: WO2015/86527, 2015, A1. Location in patent: Page/Page column 114; 115
[4] Patent: WO2015/86526, 2015, A1. Location in patent: Page/Page column 147
[5] Patent: WO2015/86525, 2015, A1. Location in patent: Page/Page column 121; 122
2-Morpholinopyrimidin-5-ylboronic acid Preparation Products And Raw materials
Raw materials
Preparation Products
2-Morpholinopyrimidin-5-ylboronic acid Suppliers
- Tel
- 021-31261262/ 49 (0)17662837245
- Fax
- (0)21-33250524
- sales@novochemy.com
- Country
- Germany
- ProdList
- 6328
- Advantage
- 58
View Lastest Price from 2-Morpholinopyrimidin-5-ylboronic acid manufacturers
- Product
- 2-Morpholinopyrimidin-5-ylboronic acid 870521-33-8
- Price
- US $7.00/KG
- Min. Order
- 1KG
- Purity
- 99%
- Supply Ability
- JD 815
- Release date
- 2019-09-02