ChemicalBook > CAS DataBase List > 4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile

4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile

Product Name
4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile
CAS No.
920965-87-3
Chemical Name
4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile
Synonyms
4-Chloro-3-cyano-7-azaindole;4-Chloro-3-cyano-7-azaind...;4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile;1H-Pyrrolo[2,3-b]pyridine-3-carbonitrile, 4-chloro-
CBNumber
CB12471243
Molecular Formula
C8H4ClN3
Formula Weight
177.59
MOL File
920965-87-3.mol
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4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile Property

Density 
1.50±0.1 g/cm3(Predicted)
storage temp. 
under inert gas (nitrogen or Argon) at 2-8°C
pka
10.58±0.40(Predicted)
Appearance
Off-white to yellow Solid
CAS DataBase Reference
920965-87-3
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Safety

RIDADR 
UN3439
HS Code 
2933998090
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P337+P313IF eye irritation persists: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

P403+P233Store in a well-ventilated place. Keep container tightly closed.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

TRC
Product number
C380843
Product name
4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile
Packaging
100mg
Price
$65
Updated
2021/12/16
Biosynth Carbosynth
Product number
FC154467
Product name
4-Chloro-1h-pyrrolo[2,3-b]pyridine-3-carbonitrile
Packaging
250mg
Price
$55
Updated
2021/12/16
Biosynth Carbosynth
Product number
FC154467
Product name
4-Chloro-1h-pyrrolo[2,3-b]pyridine-3-carbonitrile
Packaging
500mg
Price
$100
Updated
2021/12/16
Apolloscientific
Product number
OR928099
Product name
4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile
Purity
95%
Packaging
250mg
Price
$115
Updated
2021/12/16
AK Scientific
Product number
Z5347
Product name
4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile
Packaging
250mg
Price
$117
Updated
2021/12/16
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4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile Chemical Properties,Usage,Production

Synthesis

1004991-98-3

920965-87-3

Step 4: Compound C40 (3.2 g, 16.4 mmol) was suspended in dichloromethane (50 mL) at 25 °C, sulfoxide chloride (1.95 g, 16.4 mmol) was added, heated to reflux and stirred for 4 hours. Upon completion of the reaction, the mixture was cooled to 25 °C and filtered. The resulting solid was suspended in saturated sodium bicarbonate solution (10 mL) and stirred for 15 minutes. The solid was collected by filtration, washed with deionized water (50 mL) and subsequently dried under vacuum for 2 hours. The dried residue was suspended in acetonitrile (20 mL), refluxed for 1 h. The product was cooled to 25 °C, filtered and dried under reduced pressure to afford 4-chloro-3-cyano-1H-pyrrolo[2,3-b]pyridine (C41) as a light brown solid in 70% yield (2 g). The product was confirmed by infrared spectroscopy (KBr press) with major absorption peaks located at 3136, 2857, 2228, 1609, 1573, 1511, 1455, 1398, 1336, and 1312 cm^-1. NMR hydrogen spectra (CDCl3) showed δ: 13.1-13.3 (broad peaks, 1H), 8.6 (single peak, 1H), 8.3- 8.4 (double peak, 1H), 7.4-7.5 (double peak, 1H). Mass spectrometry analysis showed a molecular ion peak (M+H) of 178.2, which is consistent with the theoretically calculated value of C8H4ClN3.

References

[1] Patent: WO2008/12635, 2008, A2. Location in patent: Page/Page column 91

4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile Preparation Products And Raw materials

Raw materials

Preparation Products

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4-Chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonitrile Suppliers

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