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Glucagon Receptor Antagonist I

Product Name
Glucagon Receptor Antagonist I
CAS No.
438618-32-7
Chemical Name
Glucagon Receptor Antagonist I
Synonyms
hGCGR Antagonist;Glucagon Receptor Antagonist I;Butanamide, N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-2-ethyl-;N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
CBNumber
CB23136786
Molecular Formula
C20H30N2OS
Formula Weight
346.53
MOL File
438618-32-7.mol
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Glucagon Receptor Antagonist I Property

Boiling point:
517.8±50.0 °C(Predicted)
Density 
1.07±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: soluble
form 
White crystalline solid.
pka
13.46±0.40(Predicted)
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Cayman Chemical
Product number
21223
Product name
Glucagon Receptor Antagonist I
Purity
≥99%
Packaging
500μg
Price
$74
Updated
2024/03/01
Cayman Chemical
Product number
21223
Product name
Glucagon Receptor Antagonist I
Purity
≥99%
Packaging
1mg
Price
$132
Updated
2024/03/01
Cayman Chemical
Product number
21223
Product name
Glucagon Receptor Antagonist I
Purity
≥99%
Packaging
5mg
Price
$476
Updated
2024/03/01
AK Scientific
Product number
8227CC
Product name
GlucagonReceptorAntagonistI
Packaging
5mg
Price
$583
Updated
2021/12/16
AK Scientific
Product number
8227CC
Product name
GlucagonReceptorAntagonistI
Packaging
1mg
Price
$233
Updated
2021/12/16
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Glucagon Receptor Antagonist I Chemical Properties,Usage,Production

Description

Glucagon receptor antagonist I is a competitive antagonist of the glucagon receptor (GCGR; IC50 = 181 nM). It blocks glucagon-induced glycogenolysis in primary human hepatocytes and isolated liver. Glucagon receptor antagonist I, at 50 mg/kg, reduces the increase in glucose levels observed after intraperitoneal administration of glucagon in humanized mice. Glucagon receptor antagonist inactive control does not prevent glucagon-mediated actions.

Glucagon Receptor Antagonist I Preparation Products And Raw materials

Raw materials

Preparation Products

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Glucagon Receptor Antagonist I Suppliers

China 7 Hungary 1 Russia 1 United Kingdom 1 United States 3 Global 13
Alinda Chemical Ltd.
Tel
+7 (495) 672-17-08
Fax
+7 (495) 672-78-14
Email
sale@alinda.ru
Country
Russia
ProdList
68136
Advantage
55

438618-32-7, Glucagon Receptor Antagonist IRelated Search:

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  • Glucagon Receptor Antagonist I
  • N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
  • Butanamide, N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-2-ethyl-
  • hGCGR Antagonist
  • 438618-32-7