Meptazinol hydrochloride
- Product Name
- Meptazinol hydrochloride
- CAS No.
- 59263-76-2
- Chemical Name
- Meptazinol hydrochloride
- Synonyms
- Meptazinol hcl;Meptazinol-d3 HCl;Meptazinol hydrochlo;WY-22811 hydrochloride;IL-22811 hydrochloride;MEPTAZINOL HYDROCHLORIDE;Meptazinol-d3 hydrochloride;Meptazinol hydrochloride USP/EP/BP;IL-22811 HYDROCHLORIDE;WY-22811 HYDROCHLORIDE;3-(3-ethyl-1-methyl-3-azepanyl)phenol hydrochloride
- CBNumber
- CB4843649
- Molecular Formula
- C15H24ClNO
- Formula Weight
- 269.81
- MOL File
- 59263-76-2.mol
Meptazinol hydrochloride Property
- Melting point:
- 250-252°C
- storage temp.
- Inert atmosphere,2-8°C
- solubility
- H2O: >10mg/mL
- form
- powder
- color
- white to off-white
- Stability:
- Hygroscopic
- InChIKey
- MPJUSISYVXABBH-UHFFFAOYSA-N
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
- Precautionary statements
-
P264Wash hands thoroughly after handling.
P264Wash skin thouroughly after handling.
P270Do not eat, drink or smoke when using this product.
P501Dispose of contents/container to..…
N-Bromosuccinimide Price
- Product number
- M2824
- Product name
- Meptazinol hydrochloride
- Packaging
- 10mg
- Price
- $91.6
- Updated
- 2024/03/01
- Product number
- BP583
- Product name
- Meptazinol hydrochloride
- Purity
- British Pharmacopoeia (BP) Reference Standard
- Packaging
- 100MG
- Price
- $229
- Updated
- 2024/03/01
- Product number
- M2824
- Product name
- Meptazinol hydrochloride
- Packaging
- 50mg
- Price
- $314
- Updated
- 2022/05/15
- Product number
- 3636
- Product name
- Meptazinol hydrochloride
- Purity
- ≥99%(HPLC)
- Packaging
- 50
- Price
- $331
- Updated
- 2021/12/16
- Product number
- 3636
- Product name
- Meptazinol hydrochloride
- Purity
- ≥99%(HPLC)
- Packaging
- 10
- Price
- $83
- Updated
- 2021/12/16
Meptazinol hydrochloride Chemical Properties,Usage,Production
Description
Meptazinol hydrochloride is an injectable narcotic analgesic with antagonist properties; it is similar in potency to meperidine. Meptazinol appears to have a low propensity toward respiratory depression and other opiate-like side effects, possibly due to selective interaction with the mu-1 receptor. Also somewhat unique for an analgesic, it interacts with central cholinergic receptors. An oral form of meptazinol is under development.
Chemical Properties
White Solid
Originator
Wyeth (United Kingdom)
Uses
Analgesic;Opiate receptor agonist
Uses
Mixed opioid agonist-antagonist. Analgesic (narcotic).
brand name
MEPTID
Biological Activity
Centrally active opioid analgesic. Partial agonist at the μ 1 opioid receptor. Also shown to inhibit acetylcholinesterase.
Biochem/physiol Actions
Meptazinol entered the human pharmaceutical market as a racemic mixture in the 1980s for use as an analgesic. Its pharmacology is not completely understood; however, its analgesic properties are mostly due to its partial agonism at the mu1 opioid receptor. Due to its partial agonism, Meptazinol antagonizes morphine dependence in vivo. Its advantage over other opiates is its reduced capacity to cause addition and respiratory depression, also due to its intrinsic activity as a partial agonist. Meptazinol has been found to have additional activity as an acetylcholinesterase (AChE) inhibitor, particularly in its (-) enantiomeric form, which may partially explain its analgesic properties. AChE inhibitors are used to treat Alzheimer′s disease, providing additional interest in this compound.
Meptazinol hydrochloride Preparation Products And Raw materials
Raw materials
Preparation Products
Meptazinol hydrochloride Suppliers
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View Lastest Price from Meptazinol hydrochloride manufacturers
- Product
- Meptazinol hydrochloride 59263-76-2
- Price
- US $1.00-1.00/Kg/Bag
- Min. Order
- 1g
- Purity
- 99%
- Supply Ability
- 50tons
- Release date
- 2020-04-30
- Product
- Meptazinol HCl 59263-76-2
- Price
- US $120.00/KG
- Min. Order
- 1250KG
- Purity
- 99.8%
- Supply Ability
- 330T
- Release date
- 2023-06-05
- Product
- Meptazinol hydrochloride 59263-76-2
- Price
- US $1.10/g
- Min. Order
- 1g
- Purity
- 99.9%
- Supply Ability
- 100 Tons Min
- Release date
- 2021-06-16