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MEQUITAZINE

Product Name
MEQUITAZINE
CAS No.
29216-28-2
Chemical Name
MEQUITAZINE
Synonyms
Butix;LM 209;Mircol;MQ-A-88;Vigigan;Zesulan;Instotal;Primalan;Virginan;Nipolazin
CBNumber
CB5487473
Molecular Formula
C20H22N2S
Formula Weight
322.47
MOL File
29216-28-2.mol
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MEQUITAZINE Property

Melting point:
143-145°C
Boiling point:
469.4±24.0 °C(Predicted)
Density 
1.1330 (rough estimate)
refractive index 
1.5800 (estimate)
storage temp. 
Refrigerator
Water Solubility 
Insoluble in water
solubility 
DMSO : 16 mg/mL (49.62 mM)
form 
powder to crystal
pka
10.43±0.33(Predicted)
color 
White to Almost white
Merck 
14,5864
CAS DataBase Reference
29216-28-2(CAS DataBase Reference)
NIST Chemistry Reference
Mequitazine(29216-28-2)
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Safety

RIDADR 
UN 2811 6.1/PG III
RTECS 
SP5080000
HazardClass 
6.1
PackingGroup 
III
HS Code 
29349990
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H301Toxic if swalloed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

TCI Chemical
Product number
M2807
Product name
Mequitazine
Purity
>98.0%(GC)(T)
Packaging
100mg
Price
$69
Updated
2024/03/01
TCI Chemical
Product number
M2807
Product name
Mequitazine
Purity
>98.0%(GC)(T)
Packaging
1g
Price
$208
Updated
2024/03/01
TRC
Product number
M225110
Product name
Mequitazine
Packaging
100mg
Price
$485
Updated
2021/12/16
TRC
Product number
M225110
Product name
Mequitazine
Packaging
50g
Price
$1090
Updated
2021/12/16
Chem-Impex
Product number
38078
Product name
Mequitazine,≥98%(Assaybytitration,GC)Hazmat
Purity
≥98%(Assaybytitration,GC)
Packaging
100MG
Price
$34.94
Updated
2021/12/16
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MEQUITAZINE Chemical Properties,Usage,Production

Chemical Properties

White Solid

Originator

Primalan,Berk,UK,1976

Uses

It is an antihistamine

Definition

ChEBI: Mequitazine is a member of phenothiazines.

Manufacturing Process

30 g of phenothiazine were added, all at once, to a suspension of 6 g of sodium amide in 240 ml of anhydrous xylene. The mixture was agitated and heated to reflux. When evolution of ammonia ceased (5 hours), 15 g of 3- chloromethyl-quinuclidine hydrochloride were added portionwise over a period of 50 minutes and reflux was then maintained for 22 hours. After cooling to room temperature, 250 ml of distilled water and 250 ml of ethyl acetate were added to the reaction mixture. The aqueous phase was decanted and extracted twice with a total of 250 ml of methyl acetate. The combined organic extracts were extracted three times with a total of 750 ml of a 10% aqueous solution of tartaric acid. The combined acid solutions were treated with 5 g of animal charcoal, filtered and rendered alkaline on an ice bath with 96 ml of 10 N aqueous caustic soda. The oil which separated was extracted three times with a total of 1.500 ml of ethyl acetate. The combined organic extracts were washed to neutrality by washing twice with a total of 1 liter of distilled water, dried over anhydrous magnesium sulfate and evaporated under reduced pressure on a water bath at 45°C. 17 g of oil were obtained which was purified by chromatography on an inert alumina column. 13.3 g of crystallized product were obtained. 10-(3-Quinuclidinyl-methyl)-phenothiazine having a MP of 130°C to 131°C was obtained by recrystallization in boiling acetonitrile.
The 3-chloromethyl-quinuclidine hydrochloride used as starting material in this process can be obtained as described by Grob and coll., Helv. Chim. Acta, 37 (1954),1689.

Therapeutic Function

Antihistaminic

MEQUITAZINE Preparation Products And Raw materials

Raw materials

Preparation Products

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MEQUITAZINE Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
94657
Advantage
76
TCI (Shanghai) Development Co., Ltd.
Tel
021-67121386
Fax
021-67121385
Email
Sales-CN@TCIchemicals.com
Country
China
ProdList
24529
Advantage
81
Adamas Reagent, Ltd.
Tel
400-6009262 16621234537
Fax
021-64823266
Email
chenyj@titansci.com
Country
China
ProdList
14103
Advantage
59
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky(shanghai)International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
Advantage
50
XiaoGan ShenYuan ChemPharm co,ltd
Tel
15527768850
Email
1791901229@qq.com
Country
China
ProdList
8836
Advantage
52
Hangzhou Yuhao Chemical Technology Co., Ltd
Tel
0571-82693216
Fax
+86-571-82880190
Email
info@yuhaochemical.com
Country
China
ProdList
9387
Advantage
52
Wuhan Fortuna Chemical Co., Ltd
Tel
027-59207852 13308628970
Fax
QQ3130921841
Email
buy@fortunachem.com
Country
China
ProdList
2866
Advantage
58
Wisdom Pharmaceutical Co., Ltd.
Tel
0086-15189180296
Fax
0086-513-81292226
Email
l_xu@wisdompharma.com
Country
China
ProdList
221
Advantage
60
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
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View Lastest Price from MEQUITAZINE manufacturers

WUHAN FORTUNA CHEMICAL CO., LTD
Product
Mequitazine 29216-28-2
Price
US $0.00/Kg/Bag
Min. Order
1KG
Purity
98.5%min
Supply Ability
10kg
Release date
2021-08-05
Baoji Guokang Bio-Technology Co., Ltd.
Product
MEQUITAZINE 29216-28-2
Price
US $3015.00/Kg/Bag
Min. Order
1KG
Purity
99%
Supply Ability
5kg
Release date
2021-06-04
Zhuozhou Wenxi import and Export Co., Ltd
Product
MEQUITAZINE 29216-28-2
Price
US $15.00-10.00/KG
Min. Order
1KG
Purity
99%+ HPLC
Supply Ability
Monthly supply of 1 ton
Release date
2021-07-10

29216-28-2, MEQUITAZINERelated Search:


  • 10-(1-Azabicyclo[2.2.2]octan-3-ylmethyl)-10H-phenothiazine
  • 10-(Quinuclidin-3-ylmethyl)-10H-phenothiazine
  • MQ-A-88
  • 10-[(1R,3R)-1-azabicyclo[2.2.2]octan-3-ylMethyl]-10H-phenothiazine
  • 10H-Phenothiazine, 10-(1-azabicyclo[2.2.2]oct-3-ylmethyl)- (9CI)
  • Nipolazin
  • NSC 303612
  • Phenothiazine, 10-(3-quinuclidinylmethyl)- (8CI)
  • Quitadrill
  • 10-(1-Azabicyclo[2.2.2]oct-3-ylmethyl)-10H-phenothiazine
  • 10-(3-Quinuclidinylmethyl)phenothiazine
  • Butix
  • Instotal
  • LM 209
  • Mequitazina
  • Metaplexan
  • Mircol
  • Phenothiazine, 10-(3-quinuclidinylmethyl)-
  • 10-(1-azabicyclo[2.2.2]octan-3-ylmethyl)phenothiazine
  • Primalan
  • Vigigan
  • Virginan
  • Zesulan
  • MEQUITAZINE
  • 10H-PHENOTHIAZINE, 10-(1-AZABICYCLO[2.2.2]OCT-3-YLMETHYL)-
  • MEQUITAZINE USP/EP/BP
  • Indomethacin BP
  • Butix Powder USP Standard
  • 29216-28-2
  • C20H22N2S
  • Heterocyclic Compounds
  • Heterocycles
  • Intermediates & Fine Chemicals
  • Pharmaceuticals