ChemicalBook > CAS DataBase List > 8-AZAGUANINE

8-AZAGUANINE

Product Name: 8-AZAGUANINE
CAS No.: 134-58-7
Chemical Name: 8-AZAGUANINE
Synonyms: Azaguanine;8ag;AZG;8 AG;Azan;B-28;8-AzaG;SF-337;sk1150;NSC-749
CBNumber: CB5752825
Molecular Formula: C4H4N6O
Formula Weight: 152.11
MOL File: 134-58-7.mol

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8-AZAGUANINE Property

Melting point:: >300 °C(lit.)
Boiling point:: 274.55°C (rough estimate)
Density: 1.5579 (rough estimate)
refractive index: 2.3000 (estimate)
storage temp.: Keep in dark place,Inert atmosphere,Store in freezer, under -20°C
solubility: DMSO (Slightly)
pka: 6.75±0.20(Predicted)
form: lyophilized powder
color: White to yellow
Merck: 896
InChIKey: LPXQRXLUHJKZIE-UHFFFAOYSA-N
CAS DataBase Reference: 134-58-7(CAS DataBase Reference)
NIST Chemistry Reference: 8-Azaguanine(134-58-7)
EPA Substance Registry System: 8-Azaguanine (134-58-7)

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Safety

Hazard Codes: Xn
Risk Statements: 22
Safety Statements: 22-24/25
WGK Germany: 3
RTECS: XZ6157000
F: 10-23
HS Code: 29335990
Toxicity: LD50 oral in mouse: 1500mg/kg

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Sigma-Aldrich

Product number: SML2963
Product name: 8-Azaguanine
Purity: ≥98% (HPLC)
Packaging: 10 mg
Price: $56.62
Updated: 2025/07/31

Sigma-Aldrich

Product number: SML2963
Product name: 8-Azaguanine
Purity: ≥98% (HPLC)
Packaging: 50 mg
Price: $231
Updated: 2025/07/31

TRC

Product number: A806065
Product name: 8-Azaguanine
Packaging: 5g
Price: $195
Updated: 2021/12/16

AK Scientific

Product number: J93879
Product name: 8-Azaguanine
Packaging: 1g
Price: $30
Updated: 2021/12/16

Biosynth Carbosynth

Product number: FA07970
Product name: 8-Azaguanine
Packaging: 2g
Price: $60
Updated: 2021/12/16

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8-AZAGUANINE Chemical Properties,Usage,Production

Chemical Properties

yellow powder

Uses

Antineoplastic;Purine antimetabolite

Uses

8-Azaguanine, is a purine analogue which shows antineoplastic activity.

Definition

ChEBI: A triazolopyrimidine that consists of 3,6-dihydro-7H-[1,2,3]triazolo[4,5-d]pyrimidine bearing amino and oxo substituents at positions 5 and 7 respectively.

Hazard

Mitotoic poison.

Biological Activity

8-Azaguanine is a triazole-antimetabolite th at displays varies pharmacological effects including anticancer, antiviral and antifungal. It is easily incorporated into ribonucleic acids including rRNA and tRNA. 8-Azaguanine appears to alter mRNA splicing in SF3B1 mutant cells. 8-Azaguanine novel immunomodulatory drug (IMiD) th at significantly increases the cytotoxicity of NK cells.

Purification Methods

Dissolve it in hot M NH4OH, filter, and cool. Recrystallise it, and wash it with water, then dry it in a vacuum. [Beilstein 26 III/IV 4171.]

8-AZAGUANINE Preparation Products And Raw materials

Raw materials

Nitro Sodium dithionite Congo Red 2,4-Diamino-6-hydroxypyrimidine ,98% Amino

Preparation Products

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View Lastest Price from 8-AZAGUANINE manufacturers

Shanghai UCHEM Inc.

Product: 8-Azaguanine 134-58-7
Price: US $7.00-161.00/g
Min. Order: 1g
Purity: 0.97
Supply Ability: 10kg
Release date: 2024-04-12

Career Henan Chemical Co

Product: 8-AZAGUANINE 134-58-7
Price: US $1.00/ASSAYS
Min. Order: 1ASSAYS
Purity: 98%
Supply Ability: 1kg,2kg,100kg
Release date: 2019-07-09

134-58-7, 8-AZAGUANINERelated Search:

2-Aminopyrimidine 1H-1,2,3-Triazolo[4,5-d]pyrimidin-7-amine Paliperidone Linagliptin Anidulafungin Bexarotene VILAZODONE SB216763 Nexturastat A Clindamycin 5-[2,4-Dihydroxy-6-(4-nitrophenoxy)phenyl]-N-(1-methyl-4-piperidinyl)-3-isoxazolecarboxamide API-2 Bardoxolone Methyl 8-AZAGUANINE 8-AZAHYPOXANTHINE Guanine 1H-[1,2,3]TRIAZOL-4-YLMETHYLAMINE HCL 1H-[1,2,3]TRIAZOLE-4-CARBALDEHYDE

2-Amino-6-hydroxy-8-azapurine, 2-Amino-6-oxy-8-azapurine, Guanazolo

5-aMino-3H,6H,7H-[1,2,3]triazolo[4,5-d]pyriMidin-7-one

5-AMino-1H-[1,2,3]triazolo[4,5-d]pyriMidin-7(6H)-one

5-aMino-3H-[1,2,3]triazolo[4,5-d]pyriMidin-7(6H)-one

8-Azaguanine ,99%

8-Azaguanine,2-Amino-6-hydroxy-8-azapurine, 2-Amino-6-oxy-8-azapurine, 8-AzaG, Guanazolo

7H-1,2,3-Triazolo[4,5-d]pyriMidin-7-one, 5-aMino-3,6-dihydro-

5-AMINO-1H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-7-OL

5-amino-2,3-dihydro-[1,2,3]triazolo[4,5-e]pyrimidin-7-one

5-amino-2,3-dihydrotriazolo[4,5-e]pyrimidin-7-one

5-amino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ol

Prestwick_40

8-AzaG

{7H-1,2,3-

5-Amino-1H-triazolo[d]pyrimidin-7-ol

5-Amino-1H-v-triazolo(d)pyrimidin-7-ol

5-Amino-7-hydroxy-1H-triazolo[d]pyrimidine

5-Amino-7-hydroxy-1H-v-triazolo(d)pyrimidine

5-d)pyrimidin-7-ol,5-amino-v-triazolo(

5-d)pyrimidin-7-one,5-amino-1,6-dihydro-7h-v-triazolo(

7H-1,2,3-Triazolo[4,5-d]pyrimidin-7-one, 5-amino-1,4-dihydro-

7H-v-Triazolo(4,5-d)pyrimidin-7-one, 5-amino-1,6-dihydro-

8 AG

8ag

Azaguanine

Azan

AZG

B-28

Guanazol

NSC-749

Pathocidin

Pathocidine

SF-337

SK 1150

sk1150

Triazoloanalogofguanine

Triazologuanine

v-Triazolo(4,5-d)pyrimidin-7-ol, 5-amino-

5-amino-1H-triazolo[4,5-d]pyrimidin-7-ol

8-AZAGUANINE (50X) HYBRI-MAXGAMMA-IRRADI ATED

8-AZAGUANINE 97%

5-AMINO-1,6-DIHYDRO-7H-1,2,3-TRIAZOLO[4,5-D]PYRIMIDIN-7-ONE

5-AMINO-V-TRIAZOLO(4,5-D)-PYRIMIDIN-7-OL

8-AZAQUANINE

AZAGUANINE, 8-(RG)

GUANAZOLO

AZAGUANINE(8-)

8-AZAGUANINE

5-AMINO-3,6-DIHYDRO-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-7-ONE

5-AMINO-3,6-DIHYDRO-7H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-7-ONE

5-AMINO-1H-VIC-TRIAZOLO[4,5-D]PYRIMIDINE-7-OL

2,3-Triazolo[4,5-d]pyrimidin-7-one,5-amino-1,4-dihydro-7H-1

3-triazolo(4,5-d)pyrimidin-7-one,5-amino-1,4-dihydro-7h-2

5-Amino-1,4-dihydro-7H-1,2,3-triazolo(4,5-d)pyrimidin-7-one

5-Amino-1,6-dihydro-7H-v-triazolo(4,5-d)pyrimidin-7-one

2-AMINO-6-HYDROXY-8-AZAPURINE

2-AMINO-6-OXY-8-AZAPURINE

8-Azaguanine, >98%