Basic information Safety Supplier Related

Coclaurine

Basic information Safety Supplier Related

Coclaurine Basic information

Product Name:
Coclaurine
Synonyms:
  • Coclaurine
  • (1R)-1-(4-Hydroxybenzyl)-6-methoxy-1,2,3,4-tetrahydroisoquinoline-7-ol
  • (R)-1,2,3,4-Tetrahydro-1-(4-hydroxybenzyl)-6-methoxyisoquinolin-7-ol
  • (R)-Coclaurine
  • Sanjoinine K
  • (1R)-1,2,3,4-Tetrahydro-1-[(4-hydroxyphenyl)methyl]-6-methoxy-7-isoquinolinol
  • 7-Isoquinolinol, 1,2,3,4-tetrahydro-1-[(4-hydroxyphenyl)methyl]-6-methoxy-, (1R)-
  • (+)-Coclaurine
CAS:
2196-60-3
MF:
C17H19NO3
MW:
285.34
Mol File:
2196-60-3.mol
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Coclaurine Chemical Properties

Melting point:
222-224 °C
Boiling point:
496.9±45.0 °C(Predicted)
Density 
1.232±0.06 g/cm3(Predicted)
pka
10.00±0.15(Predicted)
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Coclaurine Usage And Synthesis

Chemical Properties

Coclaurine is a white crystalline powder, soluble in methanol, ethanol, DMSO and other organic solvents.

Uses

Coclaurine is a tetrahydroisoquinoline alkaloid with anti-aging activity,used as a nicotinic acetylcholine receptor antagonis.

Definition

ChEBI: (R)-coclaurine is a coclaurine. It is an enantiomer of a (S)-coclaurine.

in vivo

An intracerebroventricular injection of (+)-Coclaurine (d-Coclaurine; 50 μg) produces a slight increase in 3,4-dihydroxyphenylacetic acid level and a significant increase in homovanillic acid level in the mouse striatum. (+)-Coclaurine blocks postsynaptic but not presynaptic dopamine receptors in the mouse striatum[2].

CoclaurineSupplier

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