Basic information Description Clinical Use Safety Supplier Related

Pikamilone

Basic information Description Clinical Use Safety Supplier Related

Pikamilone Basic information

Product Name:
Pikamilone
Synonyms:
  • 4-((Pyridine-3-carbonyl)-amino)-butyric acid
  • Pikamiline
  • PikamiloneHCl
  • 3-[(3-Carboxypropyl)carbamoyl]pyridine
  • PIKAMILON
  • 4-Nicotinoylamino-butylric acid
  • PIKAMILONE HYDROCHLORIDE
  • NICOTINOYL-GABA
CAS:
34562-97-5
MF:
C10H12N2O3
MW:
208.21
EINECS:
1308068-626-2
Product Categories:
  • Other APIs
  • API
  • Heterocycles
  • Chemistry
  • 34562-97-5
Mol File:
34562-97-5.mol
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Pikamilone Chemical Properties

Melting point:
211.0 to 215.0 °C
Boiling point:
522.4±30.0 °C(Predicted)
Density 
1.245
storage temp. 
Inert atmosphere,Room Temperature
solubility 
DMSO (Slightly, Heated), Methanol (Slightly)
form 
Solid
pka
4.60±0.10(Predicted)
color 
White to Off-White
CAS DataBase Reference
34562-97-5(CAS DataBase Reference)
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Safety Information

Hazard Codes 
Xi
HazardClass 
IRRITANT
HS Code 
2933599590
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Pikamilone Usage And Synthesis

Description

Pikamilone is a drug having a central (vegetotropic and vascular) and peripheral (vasodilating) mechanisms of action.

Clinical Use

Pikamilone treatment of benign prostatic hyperplasia
Pikamilone is an original drug of Russian produce having a central (vegetotropic and vascular) and peripheral (vasodilating) mechanisms of action. The drug was tried as monotherapy in elderly patients with benign prostatic hyperplasia who had symptoms of the lower urinary tracts to estimate its effect on local and general mechanisms of nervous and vascular regulation of detruzor function in infravesical obstruction.
https://pubmed.ncbi.nlm.nih.gov/11150159/

Uses

anti-cancer agent

Uses

Nicotinoyl-γ-aminobutyric Acid is a pro-drug of γ-Aminobutyric Acid (A602920). Studies show that Nicotinoyl-γ-aminobutyric Acid is involved in the regulation of the processes in the brain of streptozotocin-induced diabetic rats.

PikamiloneSupplier

Wuhan Senwayer Century Chemical Co.,Ltd Gold
Tel
027-86652399 13627115097;
Email
sales@senwayer.com
TCI (Shanghai) Development Co., Ltd.
Tel
021-67121386
Email
Sales-CN@TCIchemicals.com
Pure Chemistry Scientific Inc.
Tel
001-857-928-2050 or 1-888-588-9418
Email
sales@chemreagents.com
XiaoGan ShenYuan ChemPharm co,ltd
Tel
0712-0712-2580635 15527768850
Email
1791901229@qq.com
Wuhan Fortuna Chemical Co., Ltd
Tel
027-027-59207852 13308628970
Email
buy@fortunachem.com